Dexamethasone acetate

DB14649

small molecule approved investigational vet_approved

Deskripsi

Commonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions.T797,L10695,L14348 Developed in 1957, dexamethasone is structurally similar to other corticosteroids such as hydrocortisone and prednisolone.A188724 Dexamethasone acetate has largely been replaced by dexamethasone phosphate and continues to be administered for a large variety of inflammatory conditions.L10701

Recently, dexamethasone has been a drug of interest in the treatment of COVID-19. In a June 16 2020 press release highlighting early results of a clinical trial, Randomized Evaluation of COVID-19 Therapy (RECOVERY), it was reported that dexamethasone reduced COVID-19 deaths by approximately one-fifth and one-third in patients on oxygen therapy and mechanical ventilation, respectively. Dexamethasone was therefore recommended as a life-saving treatment for COVID-19 patients experiencing severe respiratory symptoms.L14318

Struktur Molekul 2D

Berat 434.4977
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1059 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Dexamethasone acetate.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be increased when combined with Dexamethasone acetate.
Afatinib The serum concentration of Afatinib can be decreased when it is combined with Dexamethasone acetate.
Brentuximab vedotin The serum concentration of Brentuximab vedotin can be decreased when it is combined with Dexamethasone acetate.
Dabigatran etexilate The serum concentration of Dabigatran etexilate can be decreased when it is combined with Dexamethasone acetate.
Linagliptin The serum concentration of Linagliptin can be decreased when it is combined with Dexamethasone acetate.
Paliperidone The serum concentration of Paliperidone can be decreased when it is combined with Dexamethasone acetate.
Sofosbuvir The serum concentration of Sofosbuvir can be decreased when it is combined with Dexamethasone acetate.
Daclatasvir The metabolism of Daclatasvir can be increased when combined with Dexamethasone acetate.
Aspartame The excretion of Dexamethasone acetate can be decreased when combined with Aspartame.
Pravastatin The excretion of Dexamethasone acetate can be decreased when combined with Pravastatin.
Pantoprazole The excretion of Dexamethasone acetate can be decreased when combined with Pantoprazole.
Cefotiam The excretion of Dexamethasone acetate can be decreased when combined with Cefotiam.
Liothyronine The excretion of Dexamethasone acetate can be decreased when combined with Liothyronine.
Conjugated estrogens The excretion of Dexamethasone acetate can be decreased when combined with Conjugated estrogens.
Valproic acid The excretion of Dexamethasone acetate can be decreased when combined with Valproic acid.
Indomethacin The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Indomethacin.
Aminohippuric acid The excretion of Dexamethasone acetate can be decreased when combined with Aminohippuric acid.
Lansoprazole The excretion of Dexamethasone acetate can be decreased when combined with Lansoprazole.
Cefalotin The excretion of Dexamethasone acetate can be decreased when combined with Cefalotin.
Tenoxicam The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Tenoxicam.
Cefotaxime The excretion of Dexamethasone acetate can be decreased when combined with Cefotaxime.
Zidovudine The excretion of Dexamethasone acetate can be decreased when combined with Zidovudine.
Cimetidine The excretion of Dexamethasone acetate can be decreased when combined with Cimetidine.
Guanidine The excretion of Dexamethasone acetate can be decreased when combined with Guanidine.
Piroxicam The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Piroxicam.
Cephalexin The excretion of Dexamethasone acetate can be decreased when combined with Cephalexin.
Enalapril The excretion of Dexamethasone acetate can be decreased when combined with Enalapril.
Diclofenac The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Diclofenac.
Oxytetracycline The excretion of Dexamethasone acetate can be decreased when combined with Oxytetracycline.
Leucovorin The excretion of Dexamethasone acetate can be decreased when combined with Leucovorin.
Furosemide The excretion of Dexamethasone acetate can be decreased when combined with Furosemide.
Esomeprazole The excretion of Dexamethasone acetate can be decreased when combined with Esomeprazole.
Tetracycline The excretion of Dexamethasone acetate can be decreased when combined with Tetracycline.
Acyclovir The excretion of Dexamethasone acetate can be decreased when combined with Acyclovir.
Phenylbutazone The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Phenylbutazone.
Cefaclor The excretion of Dexamethasone acetate can be decreased when combined with Cefaclor.
Bumetanide The excretion of Dexamethasone acetate can be decreased when combined with Bumetanide.
Dinoprostone The excretion of Dexamethasone acetate can be decreased when combined with Dinoprostone.
Famotidine The excretion of Dexamethasone acetate can be decreased when combined with Famotidine.
Salicylic acid The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Salicylic acid.
Acetylsalicylic acid The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Acetylsalicylic acid.
Ganciclovir The excretion of Dexamethasone acetate can be decreased when combined with Ganciclovir.
Ketoprofen The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Ketoprofen.
Minocycline The excretion of Dexamethasone acetate can be decreased when combined with Minocycline.
Probenecid The excretion of Dexamethasone acetate can be decreased when combined with Probenecid.
Mercaptopurine The excretion of Dexamethasone acetate can be decreased when combined with Mercaptopurine.
Ibuprofen The risk or severity of gastrointestinal irritation can be increased when Dexamethasone acetate is combined with Ibuprofen.
Novobiocin The excretion of Dexamethasone acetate can be decreased when combined with Novobiocin.
Benzylpenicillin The excretion of Dexamethasone acetate can be decreased when combined with Benzylpenicillin.
Melatonin The excretion of Dexamethasone acetate can be decreased when combined with Melatonin.
Ouabain The excretion of Dexamethasone acetate can be decreased when combined with Ouabain.
Rosuvastatin The excretion of Dexamethasone acetate can be decreased when combined with Rosuvastatin.
Cefadroxil The excretion of Dexamethasone acetate can be decreased when combined with Cefadroxil.
Ceftriaxone The excretion of Dexamethasone acetate can be decreased when combined with Ceftriaxone.
Gemfibrozil The excretion of Dexamethasone acetate can be decreased when combined with Gemfibrozil.
Cefamandole The excretion of Dexamethasone acetate can be decreased when combined with Cefamandole.
Cefazolin The excretion of Dexamethasone acetate can be decreased when combined with Cefazolin.
Cefoperazone The excretion of Dexamethasone acetate can be decreased when combined with Cefoperazone.
Ceftizoxime The excretion of Dexamethasone acetate can be decreased when combined with Ceftizoxime.
Cefacetrile The excretion of Dexamethasone acetate can be decreased when combined with Cefacetrile.
Ceftibuten The excretion of Dexamethasone acetate can be decreased when combined with Ceftibuten.
Liotrix The excretion of Dexamethasone acetate can be decreased when combined with Liotrix.
Cilastatin The excretion of Dexamethasone acetate can be decreased when combined with Cilastatin.
Tazobactam The excretion of Dexamethasone acetate can be decreased when combined with Tazobactam.
trans-2-hydroxycinnamic acid The excretion of Dexamethasone acetate can be decreased when combined with trans-2-hydroxycinnamic acid.
Topiroxostat The excretion of Dexamethasone acetate can be decreased when combined with Topiroxostat.
Cholic Acid The excretion of Dexamethasone acetate can be decreased when combined with Cholic Acid.
Glutaric Acid The excretion of Dexamethasone acetate can be decreased when combined with Glutaric Acid.
Benzoic acid The therapeutic efficacy of Benzoic acid can be decreased when used in combination with Dexamethasone acetate.
Taurocholic acid The excretion of Dexamethasone acetate can be decreased when combined with Taurocholic acid.
Caprylic acid The excretion of Dexamethasone acetate can be decreased when combined with Caprylic acid.
Ataluren The excretion of Dexamethasone acetate can be decreased when combined with Ataluren.
Teriflunomide The excretion of Dexamethasone acetate can be decreased when combined with Teriflunomide.
Dolutegravir The excretion of Dexamethasone acetate can be decreased when combined with Dolutegravir.
Cefaloridine The excretion of Dexamethasone acetate can be decreased when combined with Cefaloridine.
Lenvatinib The excretion of Dexamethasone acetate can be decreased when combined with Lenvatinib.
Tafamidis The excretion of Dexamethasone acetate can be decreased when combined with Tafamidis.
Cabotegravir The excretion of Dexamethasone acetate can be decreased when combined with Cabotegravir.
Letermovir The metabolism of Dexamethasone acetate can be decreased when combined with Letermovir.
Rucaparib Dexamethasone acetate may decrease the excretion rate of Rucaparib which could result in a higher serum level.
Favipiravir The excretion of Dexamethasone acetate can be decreased when combined with Favipiravir.
Pradigastat The excretion of Dexamethasone acetate can be decreased when combined with Pradigastat.
Linezolid The excretion of Dexamethasone acetate can be decreased when combined with Linezolid.
Ifosfamide The metabolism of Ifosfamide can be increased when combined with Dexamethasone acetate.
Ledipasvir The serum concentration of Ledipasvir can be decreased when it is combined with Dexamethasone acetate.
Perampanel The metabolism of Perampanel can be increased when combined with Dexamethasone acetate.
Warfarin Dexamethasone acetate may increase the anticoagulant activities of Warfarin.
Acenocoumarol Dexamethasone acetate may increase the anticoagulant activities of Acenocoumarol.
(R)-warfarin Dexamethasone acetate may increase the anticoagulant activities of (R)-warfarin.
R,S-Warfarin alcohol The metabolism of R,S-Warfarin alcohol can be increased when combined with Dexamethasone acetate.
S,R-Warfarin alcohol The metabolism of S,R-Warfarin alcohol can be increased when combined with Dexamethasone acetate.
(S)-Warfarin Dexamethasone acetate may increase the anticoagulant activities of (S)-Warfarin.
Doxorubicin The serum concentration of Doxorubicin can be decreased when it is combined with Dexamethasone acetate.
Vincristine The serum concentration of Vincristine can be decreased when it is combined with Dexamethasone acetate.
Rolapitant The metabolism of Rolapitant can be increased when combined with Dexamethasone acetate.
Erlotinib The serum concentration of Erlotinib can be decreased when it is combined with Dexamethasone acetate.
Diethylstilbestrol The serum concentration of Dexamethasone acetate can be increased when it is combined with Diethylstilbestrol.
Etonogestrel The serum concentration of Dexamethasone acetate can be increased when it is combined with Etonogestrel.
Desogestrel The serum concentration of Dexamethasone acetate can be increased when it is combined with Desogestrel.

Target Protein

Glucocorticoid receptor NR3C1
Annexin A1 ANXA1
Nitric oxide synthase, inducible NOS2
Nuclear receptor subfamily 0 group B member 1 NR0B1
Nuclear receptor subfamily 1 group I member 2 NR1I2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 13560344
    BUNIM JJ, BLACK RL, LUTWAK L, PETERSON RE, WHEDON GD: Studies on dexamethasone, a new synthetic steroid, in rheurheumatoid arthritis: a preliminary report; adrenal cortical, metabolic and early clinical effects. Arthritis Rheum. 1958 Aug;1(4):313-31. doi: 10.1002/art.1780010404.
Textbook
  • Susan J. Dreyer MD, William Jeremy Beckworth MD (2011). Pain procedures in clinical practice: Commonly Used Medications in Procedures (3rd ed.). Elsevier.

Contoh Produk & Brand

Produk: 1 • International brands: 1
Produk
  • Dexamethasone Acetate Micro
    Powder • 1 g/1g • Not applicable • US
International Brands
  • Decadron-LA

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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