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Total database: 17430
Struktur (SMILES)
15 (78.9%)
Target
12 (63.2%)
Genomik
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19 (100.0%)

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Hasil Pencarian (19)

Alovudine F-18 DB14930
small molecule | CAS: 287114-80-1

Alovudine F-18 is under investigation in clinical trial NCT02819024 (Dexamethasone Effects in Patients With Refractory Non-Small Cell Lung Cancer Using FLT Positron Emission Tomography).

Kategori:
Anti-Infective AgentsAntiviral AgentsDeoxyribonucleosides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anifrolumab Approved DB11976
biotech | CAS: 1326232-46-5

Anifrolumab, or MEDI-546, is a type 1 interferon receptor (IFNAR) inhibiting IgG1? monoclonal antibody indicated in the treatment of adults with moderate to severe systemic lupus erythematosus.[A237074,L34929] The standard therapy for systemic lupus erythemat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe serum eliminati…
Vol. DistribusiBased on population…
KlirensFollowing the admin…
Genetik -
biotech | CAS: 1826819-58-2

Azintuxizumab vedotin is under investigation in clinical trial NCT02951117 (A Study of Venetoclax and ABBV-838 Combination Therapy With Dexamethasone in Participants With Multiple Myeloma Whose Cancer Has Come Back or Had No Response to Recent Cancer Treatmen…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Beclomethasone dipropionate Approved DB00394
small molecule | CAS: 5534-09-8

Beclomethasone dipropionate is a second-generation[A179842] synthetic corticosteroid and diester of beclomethasone, which is structurally similar to [dexamethasone].[L6871] It is a prodrug of an active metabolite beclomethasone 17-monopropionate (17-BMP)[A179…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +40
Target Protein:
Glucocorticoid receptor
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Betamethasone Approved DB00443
small molecule | CAS: 378-44-9

Betamethasone is a long-acting corticosteroid with immunosuppressive and antiinflammatory properties.[A192444] It can be used topically to manage inflammatory skin conditions such as eczema, and parenterally to manage several disease states including autoimmu…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +52
Target Protein:
Glucocorticoid receptor
Waktu ParuhIn a study that inc…
Vol. DistribusiIn a study that inc…
KlirensIn a study that inc…
Genetik -
small molecule | CAS: 97011-16-0

NA-831 (Traneurocin), is under investigation in two clinical trials: NCT03538522 (completed, for mild cognitive impairment and Alzheimer’s disease) and NCT04452565 (unknown status, combination therapy with Atazanavir and Dexamethasone for COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitinase B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexamethasone Approved DB01234
small molecule | CAS: 50-02-2

Dexamethasone, or MK-125, is a corticosteroid fluorinated at position 9 used to treat endocrine, rheumatic, collagen, dermatologic, allergic, ophthalmic, gastrointestinal, respiratory, hematologic, neoplastic, edematous, and other conditions.[L10701] Develope…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +74
Target Protein:
Glucocorticoid receptorNuclear receptor subfamily 0 group B member 1Annexin A1 +2
Waktu ParuhThe mean terminal h…
Vol. DistribusiA 1.5mg oral dose o…
KlirensA 20mg oral tablet …
Genetik -
Dexamethasone acetate Approved DB14649
small molecule | CAS: 1177-87-3

Commonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions.[T797,L10695,L14348] Developed in 1957, dexamethasone is struct…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Glucocorticoid receptorAnnexin A1Nitric oxide synthase, inducible +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2265-64-7

Dexamethasone isonicotinate is an anti-inflammatory, anti-allergic glucocorticoid that can be administered orally, by inhalation, topically, and parenterally. Its unintended mineralocorticoid action may cause salt and water retention.

Kategori:
Adrenal Cortex HormonesAnti-Allergic AgentsAnti-Inflammatory Agents +25
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 16978-57-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14899-36-6

Dexamethasone palmitate is under investigation in clinical trial NCT05693467 (Preemptive Co-infiltration of Dexamethasone Palmitate With Ropivacaine for Postoperative Pain in Major Spinal Surgery).

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +3
Target Protein:
Steroid hormone receptor ERR1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elotuzumab Approved DB06317
biotech | CAS: 915296-00-3

Elotuzumab is a humanized IgG1 (Immunoglobulin G) monoclonal antibody indicated in combination with lenalidomide and dexamethasone for the treatment of patients with multiple myeloma who have received one to three prior therapies. Elotuzumab targets SLAMF7, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
SLAM family member 7
Waktu Paruh-
Vol. Distribusi-
KlirensThe clearance of el…
Genetik -
Marbofloxacin DB11426
small molecule | CAS: 115550-35-1

Marbofloxacin is a carboxylic acid, part of the third generation of antibiotic fluoroquinolones. It is used in veterinary medicine. A formulation of marbofloxacin combined with clotrimazole and dexamethasone is available under the name Aurizon.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melphalan flufenamide Approved DB16627
small molecule | CAS: 380449-51-4

Melphalan flufenamide, also known as melflufen or J1, is a prodrug of [melphalan].[A230123,L32173] Melphalan flufenamide is more readily uptaken by cells than melphalan, and is cleaved to the active metabolite by aminopeptidases.[A230123] _In vitro_ models sh…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +12
Target Protein:
DNA
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Mometasone furoate Approved DB14512
small molecule | CAS: 83919-23-7

Mometasone furoate is a corticosteroid drug that can be used for the treatment of asthma, rhinitis, and certain skin conditions[FDA Label][F4292,F4295]. It has a glucocorticoid receptor binding affinity 22 times stronger than [dexamethasone] and higher than m…

Kategori:
Adrenal Cortex HormonesAdrenalsAdrenergics, Inhalants +28
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiSteady state volume…
KlirensThe clearance rate …
Genetik -
Narazaciclib DB19038
small molecule | CAS: 1357470-29-1

Narazaciclib is under investigation in clinical trial NCT06351644 (On 123300 (Narazaciclib) and Dexamethasone in Patients With Relapsed And/or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
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Neomycin Approved DB00994
small molecule | CAS: 1404-04-2

Neomycin is a broad-spectrum aminoglycoside antibiotic drug that is derived from the metabolic products of _Streptomyces fradiae_.[L11979] Neomycin is a complex comprised of three components, neomycin A, B, and C.[A191529] Neomycin B, also known as [framyceti…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAminoglycoside Antibacterials +28
Target Protein:
30S ribosomal protein S1216S ribosomal RNAExtracellular calcium-sensing receptor
Waktu ParuhThere is limited in…
Vol. DistribusiThe small fraction …
KlirensThere is limited in…
Genetik -
Selinexor Approved DB11942
small molecule | CAS: 1393477-72-9

Selinexor is a first-in-class selective inhibitor of nuclear transport (SINE) compound. Selinexor, in combination with [bortezomib] and [dexamethasone], is currently approved for the treatment of multiple myeloma, a type of cancer formed from antibody-produci…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP3A Substrates +4
Target Protein:
Exportin-1
Waktu ParuhSelinexor has a mea…
Vol. DistribusiThe mean apparent v…
KlirensSelinexor has a mea…
Genetik -
VLX-1570 DB16030
small molecule | CAS: 1956378-23-6

VLX-1570 is under investigation in clinical trial NCT02372240 (A Study of VLX1570 and Dexamethasone in Myeloma Patients).

Kategori:
Benzene Derivatives
Waktu Paruh-
Vol. Distribusi-
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Genetik -