Peringatan Keamanan

Overdose with a mometasone furoate inhaler may occur with chronic overuseFDA LabelF4292. Symptoms of chronic overuse may present as hypercorticism and adrenal suppression, and patients may not require any more treatment than monitoringFDA LabelF4292.

In animal studies of pregnancy, some fetal toxic effects were seen at or above the maximum recommended human dose, though rodents are more sensitive to these effects than humansFDA LabelF4292,F4295. The benefits and risks of use should be considered in pregnant patientsF4292,F4295

It is unknown if mometasone furoate is excreted in breast milk but other corticosteroids are and therefore caution should be exercised when administering to nursing mothersFDA LabelF4292,F4295.

Safety and effectiveness in pediatric populations has been established through clinical trials, though there may be a reduction in expected growth of about 1cm per year depending on the dose and duration of treatmentFDA Label. Pediatric patients should be titrated to the lowest effective dose for mometasone furoate inhalersFDA Label.

A trial of geriatric patients showed no difference in safety or efficacy compared to younger patients, however patients of an even greater age may still be more sensitive to mometasone furoateFDA LabelF4292,F4295.

The use of a mometasone furoate inhaler in moderate or severe hepatic impairment rarely leads to detectable plasma concentrations though caution may be prudent with increasing degrees of severityFDA LabelF4292.

The effects of mometasone furoate in renal impairment, and across gender and race have not been studiedFDA LabelF4292.

Mometasone furoate

DB14512

small molecule approved investigational vet_approved

Deskripsi

Mometasone furoate is a corticosteroid drug that can be used for the treatment of asthma, rhinitis, and certain skin conditionsFDA LabelF4292,F4295. It has a glucocorticoid receptor binding affinity 22 times stronger than dexamethasone and higher than many other corticosteroids as wellA176906. Mometasone furoate is formulated as a dry powder inhaler, nasal spray, and ointment for its different indicationsFDA LabelF4292,F4295.

Struktur Molekul 2D

Berat 521.429
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The terminal half life of an inhaled dose is approximately 5 hours[FDA Label] though it has been reported as 5.8 hours by other sources[F4292,A176906].
Volume Distribusi Steady state volume of distribution of 152L[FDA Label].
Klirens (Clearance) The clearance rate of mometasone furoate is not readily available[A176900], though it may be close to 90L/h[A176906].

Absorpsi

The mean time to peak concentration is 1.0 to 2.5 hoursFDA Label. Bioavailability has been reported as <1%FDA Label but studies of repeat doses of inhaled corticosteroids suggest a bioavailability of 11%A176918. The 0.1% ointment may have a bioavailability of 0.7%F4295.

Metabolisme

Metabolism of mometasone furoate is largely performed hepatically by cytochrome P450 3A4 producing a number of metabolitesFDA LabelF4292,A176900,A176918. Some of these metabolites include free mometasone and 6-beta-hydroxy-mometasone furoateA176900,A176918,A176879.

Rute Eliminasi

For an inhaled dose, approximately 74% is excreted in the feces and 8% is excreted in the urineFDA LabelF4292.

Interaksi Obat

1191 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Mometasone furoate.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Mometasone furoate.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Mometasone furoate.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Mometasone furoate.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Mometasone furoate.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Mometasone furoate.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Mometasone furoate.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Mometasone furoate.
Pegaspargase The serum concentration of Mometasone furoate can be increased when it is combined with Pegaspargase.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Mometasone furoate.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mometasone furoate.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Mometasone furoate.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Mometasone furoate.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Mometasone furoate.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Mometasone furoate.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Mometasone furoate.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Mometasone furoate.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Mometasone furoate.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Mometasone furoate.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Mometasone furoate.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Mometasone furoate.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Mometasone furoate.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Mometasone furoate.
Cladribine Mometasone furoate may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Mometasone furoate.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Mometasone furoate.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Mometasone furoate.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Mometasone furoate.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Mometasone furoate.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Mometasone furoate.
Bexarotene The risk or severity of adverse effects can be increased when Bexarotene is combined with Mometasone furoate.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Mometasone furoate.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Mometasone furoate.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Mometasone furoate.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Mometasone furoate.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Mometasone furoate.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Mometasone furoate.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Mometasone furoate.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Mometasone furoate.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Mometasone furoate.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Mometasone furoate.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Mometasone furoate.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Mometasone furoate.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Mometasone furoate.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Mometasone furoate.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Mometasone furoate.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Mometasone furoate.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Mometasone furoate.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mycophenolate mofetil is combined with Mometasone furoate.
Tretinoin The metabolism of Tretinoin can be increased when combined with Mometasone furoate.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Mometasone furoate.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Mometasone furoate.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Mometasone furoate.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Mometasone furoate.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Mometasone furoate.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Mometasone furoate.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Mometasone furoate.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Mometasone furoate.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Mometasone furoate.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Mometasone furoate.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Mometasone furoate.
Thalidomide The risk or severity of adverse effects can be increased when Thalidomide is combined with Mometasone furoate.
Melphalan The risk or severity of adverse effects can be increased when Melphalan is combined with Mometasone furoate.
Fludarabine The risk or severity of adverse effects can be increased when Fludarabine is combined with Mometasone furoate.
Flucytosine The risk or severity of adverse effects can be increased when Flucytosine is combined with Mometasone furoate.
Capecitabine The risk or severity of adverse effects can be increased when Capecitabine is combined with Mometasone furoate.
Procarbazine The risk or severity of adverse effects can be increased when Procarbazine is combined with Mometasone furoate.
Arsenic trioxide The risk or severity of adverse effects can be increased when Arsenic trioxide is combined with Mometasone furoate.
Idarubicin The risk or severity of adverse effects can be increased when Idarubicin is combined with Mometasone furoate.
Estramustine The risk or severity of adverse effects can be increased when Estramustine is combined with Mometasone furoate.
Mitoxantrone The risk or severity of adverse effects can be increased when Mitoxantrone is combined with Mometasone furoate.
Lomustine The risk or severity of adverse effects can be increased when Lomustine is combined with Mometasone furoate.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Mometasone furoate.
Decitabine The risk or severity of adverse effects can be increased when Decitabine is combined with Mometasone furoate.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Mometasone furoate.
Stepronin The risk or severity of adverse effects can be increased when Stepronin is combined with Mometasone furoate.
Hydroxychloroquine The risk or severity of adverse effects can be increased when Hydroxychloroquine is combined with Mometasone furoate.
Castanospermine The risk or severity of adverse effects can be increased when Castanospermine is combined with Mometasone furoate.
Vorinostat The risk or severity of adverse effects can be increased when Vorinostat is combined with Mometasone furoate.
2-Methoxyethanol The risk or severity of adverse effects can be increased when 2-Methoxyethanol is combined with Mometasone furoate.
Brequinar The risk or severity of adverse effects can be increased when Brequinar is combined with Mometasone furoate.
Pirfenidone The risk or severity of adverse effects can be increased when Pirfenidone is combined with Mometasone furoate.
Interferon alfa The risk or severity of adverse effects can be increased when Interferon alfa is combined with Mometasone furoate.
Glatiramer The risk or severity of adverse effects can be increased when Glatiramer is combined with Mometasone furoate.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Mometasone furoate.
Human interferon omega-1 The risk or severity of adverse effects can be increased when Human interferon omega-1 is combined with Mometasone furoate.
Mepolizumab The risk or severity of adverse effects can be increased when Mepolizumab is combined with Mometasone furoate.
Abetimus The risk or severity of adverse effects can be increased when Abetimus is combined with Mometasone furoate.
Belatacept The risk or severity of adverse effects can be increased when Belatacept is combined with Mometasone furoate.
Bendamustine The risk or severity of adverse effects can be increased when Bendamustine is combined with Mometasone furoate.
Pralatrexate The risk or severity of adverse effects can be increased when Pralatrexate is combined with Mometasone furoate.
Wortmannin The risk or severity of adverse effects can be increased when Wortmannin is combined with Mometasone furoate.
Eribulin The risk or severity of adverse effects can be increased when Eribulin is combined with Mometasone furoate.
Belimumab The risk or severity of adverse effects can be increased when Belimumab is combined with Mometasone furoate.
Teriflunomide The risk or severity of adverse effects can be increased when Teriflunomide is combined with Mometasone furoate.
Carfilzomib The risk or severity of adverse effects can be increased when Carfilzomib is combined with Mometasone furoate.
Dimethyl fumarate The risk or severity of adverse effects can be increased when Dimethyl fumarate is combined with Mometasone furoate.
Obinutuzumab The risk or severity of adverse effects can be increased when Obinutuzumab is combined with Mometasone furoate.
Vedolizumab The risk or severity of adverse effects can be increased when Vedolizumab is combined with Mometasone furoate.
Blinatumomab The risk or severity of adverse effects can be increased when Blinatumomab is combined with Mometasone furoate.

Target Protein

Glucocorticoid receptor NR3C1
Progesterone receptor PGR

Referensi & Sumber

Artikel (PubMed)
  • PMID: 11449203
    Szefler SJ: Pharmacokinetics of intranasal corticosteroids. J Allergy Clin Immunol. 2001 Jul;108(1 Suppl):S26-31.
  • PMID: 16054538
    Hubner M, Hochhaus G, Derendorf H: Comparative pharmacology, bioavailability, pharmacokinetics, and pharmacodynamics of inhaled glucocorticosteroids. Immunol Allergy Clin North Am. 2005 Aug;25(3):469-88. doi: 10.1016/j.iac.2005.05.004.
  • PMID: 11589253
    Crim C, Pierre LN, Daley-Yates PT: A review of the pharmacology and pharmacokinetics of inhaled fluticasone propionate and mometasone furoate. Clin Ther. 2001 Sep;23(9):1339-54.
  • PMID: 14595701
    Teng XW, Cutler DJ, Davies NM: Mometasone furoate degradation and metabolism in human biological fluids and tissues. Biopharm Drug Dispos. 2003 Nov;24(8):321-33. doi: 10.1002/bdd.362.

Contoh Produk & Brand

Produk: 197 • International brands: 6
Produk
  • Allergy
    Spray, metered • 50 ug/1 • Nasal • US • OTC • Approved
  • Allergy Nasal
    Spray, metered • 50 ug/1 • Nasal • US • OTC • Approved
  • Apo-mometasone
    Spray, metered • 50 mcg / act • Nasal • Canada • Generic • Approved
  • Asmanex
    Inhalant • 220 ug/1 • Respiratory (inhalation) • US • Approved
  • Asmanex
    Inhalant • 220 ug/1 • Respiratory (inhalation) • US • Approved
  • Asmanex
    Inhalant • 110 ug/1 • Respiratory (inhalation) • US • Approved
  • Asmanex
    Inhalant • 220 ug/1 • Respiratory (inhalation) • US • Approved
  • Asmanex
    Inhalant • 110 ug/1 • Respiratory (inhalation) • US • Approved
Menampilkan 8 dari 197 produk.
International Brands
  • Ecural — Essex pharma
  • Elocom — Merck
  • Elomet — Schering-Plough
  • Eziwin — Intas
  • mometAid — Progreś Laboratories
  • Novasone — Schering-Plough

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul