Peringatan Keamanan

Single doses of up to 640mg given both intravenously and subcutaneously have been administered in clinical studies without evidence of dose-limiting toxicities.L39665 If overdosage of bimekizumab is suspected, monitor the patient for adverse reactions and institute symptomatic treatment as clinically indicated.

Bimekizumab

DB12917

biotech approved investigational

Deskripsi

Bimekizumab is a humanized monoclonal antibody directed towards IL-17, which was approved for use in the EU on August 20, 2021, for the treatment of plaque psoriasis.L39665,L39680 It is the first IL-17 inhibitor to target both IL-17A and IL-17F.A244455 It has demonstrated superior efficacy as compared to another IL-17 inhibitor, secukinumab, as well as ustekinumab (an IL-12/23 inhibitor) and adalimumab (a TNF inhibitor) in the treatment of moderate-to-severe psoriasis,A244450,A244455 likely owing to its dual inhibition of both IL-17A and IL-17F. Bimekizumab was also granted FDA approval on October 18, 2023.L48551

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The mean terminal elimination half-life of bimekizumab in patients with plaque psoriasis was 23 days.[L39665]
Volume Distribusi In patients with plaque psoriasis, the median volume of distribution at steady-state was 11.2 L.[L39665]
Klirens (Clearance) The median apparent clearance of bimekuzmab in patients with plaque psoriasis was 0.337 L/day.[L39665]

Absorpsi

In healthy volunteers, the absolute bioavailability of bimekizumab following subcutaneous injection was 70.1%.L39665

Metabolisme

As a monoclonal antibody, bimekizumab is likely degraded into smaller peptides and amino acids via catabolic processes.L39665

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1334 Data
Diethylstilbestrol The metabolism of Diethylstilbestrol can be increased when combined with Bimekizumab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Bimekizumab.
Conjugated estrogens The metabolism of Conjugated estrogens can be increased when combined with Bimekizumab.
Estrone Estrone may increase the thrombogenic activities of Bimekizumab.
Estradiol The metabolism of Estradiol can be increased when combined with Bimekizumab.
Dienestrol Dienestrol may increase the thrombogenic activities of Bimekizumab.
Ethinylestradiol The metabolism of Ethinylestradiol can be increased when combined with Bimekizumab.
Mestranol The metabolism of Mestranol can be increased when combined with Bimekizumab.
Estriol Estriol may increase the thrombogenic activities of Bimekizumab.
Estrone sulfate The metabolism of Estrone sulfate can be increased when combined with Bimekizumab.
Quinestrol Quinestrol may increase the thrombogenic activities of Bimekizumab.
Hexestrol Hexestrol may increase the thrombogenic activities of Bimekizumab.
Tibolone Tibolone may increase the thrombogenic activities of Bimekizumab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Bimekizumab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Bimekizumab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Bimekizumab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Bimekizumab.
Zeranol Zeranol may increase the thrombogenic activities of Bimekizumab.
Equol Equol may increase the thrombogenic activities of Bimekizumab.
Promestriene Promestriene may increase the thrombogenic activities of Bimekizumab.
Methallenestril Methallenestril may increase the thrombogenic activities of Bimekizumab.
Epimestrol Epimestrol may increase the thrombogenic activities of Bimekizumab.
Moxestrol Moxestrol may increase the thrombogenic activities of Bimekizumab.
Estradiol acetate The metabolism of Estradiol acetate can be increased when combined with Bimekizumab.
Estradiol benzoate The metabolism of Estradiol benzoate can be increased when combined with Bimekizumab.
Estradiol cypionate The metabolism of Estradiol cypionate can be increased when combined with Bimekizumab.
Estradiol valerate The metabolism of Estradiol valerate can be increased when combined with Bimekizumab.
Biochanin A Biochanin A may increase the thrombogenic activities of Bimekizumab.
Formononetin Formononetin may increase the thrombogenic activities of Bimekizumab.
Estetrol The metabolism of Estetrol can be increased when combined with Bimekizumab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Bimekizumab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Bimekizumab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Bimekizumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Bimekizumab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Bimekizumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Bimekizumab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Bimekizumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Bimekizumab.
Trastuzumab The risk or severity of neutropenia can be increased when Trastuzumab is combined with Bimekizumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Bimekizumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Bimekizumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Bimekizumab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Bimekizumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Bimekizumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Bimekizumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Bimekizumab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Bimekizumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Bimekizumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Bimekizumab.
Natalizumab The risk or severity of immunosuppression can be increased when Bimekizumab is combined with Natalizumab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Bimekizumab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Bimekizumab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Bimekizumab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Bimekizumab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Bimekizumab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Bimekizumab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Bimekizumab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Bimekizumab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Bimekizumab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Bimekizumab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Bimekizumab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Bimekizumab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Bimekizumab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Bimekizumab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Bimekizumab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Bimekizumab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Bimekizumab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Bimekizumab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Bimekizumab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Bimekizumab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Bimekizumab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Bimekizumab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Bimekizumab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Bimekizumab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Bimekizumab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Bimekizumab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Bimekizumab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Bimekizumab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Bimekizumab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Bimekizumab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Bimekizumab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Bimekizumab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Bimekizumab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Bimekizumab.
Trastuzumab emtansine The metabolism of Trastuzumab emtansine can be increased when combined with Bimekizumab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Bimekizumab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Bimekizumab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Bimekizumab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Bimekizumab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Bimekizumab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Bimekizumab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Bimekizumab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Bimekizumab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Bimekizumab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Bimekizumab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Bimekizumab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Bimekizumab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Bimekizumab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Bimekizumab.
Lumiliximab The risk or severity of adverse effects can be increased when Lumiliximab is combined with Bimekizumab.

Target Protein

Interleukin-17A IL17A
Interleukin-17F IL17F

Referensi & Sumber

Synthesis reference: Adams R, Maroof A, Baker T, Lawson ADG, Oliver R, Paveley R, Rapecki S, Shaw S, Vajjah P, West S, Griffiths M: Bimekizumab, a Novel Humanized IgG1 Antibody That Neutralizes Both IL-17A and IL-17F. Front Immunol. 2020 Aug 21;11:1894. doi: 10.3389/fimmu.2020.01894. eCollection 2020.
Artikel (PubMed)
  • PMID: 34884596
    Singh R, Koppu S, Perche PO, Feldman SR: The Cytokine Mediated Molecular Pathophysiology of Psoriasis and Its Clinical Implications. Int J Mol Sci. 2021 Nov 26;22(23). pii: ijms222312793. doi: 10.3390/ijms222312793.
  • PMID: 34178093
    Freitas E, Torres T: Bimekizumab: the new drug in the biologics armamentarium for psoriasis. Drugs Context. 2021 Jun 8;10. pii: dic-2021-4-1. doi: 10.7573/dic.2021-4-1. eCollection 2021.
  • PMID: 33727793
    Oliveira DG, Faria R, Torres T: An Overview of Bimekizumab for the Treatment of Psoriatic Arthritis: The Evidence so Far. Drug Des Devel Ther. 2021 Mar 9;15:1045-1053. doi: 10.2147/DDDT.S267405. eCollection 2021.

Contoh Produk & Brand

Produk: 17 • International brands: 0
Produk
  • Bimzelx
    Injection, solution • 320 mg/2mL • Subcutaneous • US • Approved
  • Bimzelx
    Injection, solution • 320 mg/2mL • Subcutaneous • US • Approved
  • Bimzelx
    Solution • 160 mg / mL • Subcutaneous • Canada • Approved
  • Bimzelx
    Solution • 160 mg / mL • Subcutaneous • Canada • Approved
  • Bimzelx
    Injection, solution • 160 mg • Subcutaneous • EU • Approved
  • Bimzelx
    Injection, solution • 160 mg • Subcutaneous • EU • Approved
  • Bimzelx
    Injection, solution • 160 mg • Subcutaneous • EU • Approved
  • Bimzelx
    Injection, solution • 160 mg • Subcutaneous • EU • Approved
Menampilkan 8 dari 17 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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