Ublituximab

DB11850

biotech approved investigational

Deskripsi

CD20, an antigen expressed by various B and T cells, is an attractive therapeutic target in various cancers and autoimmune conditions.A244195, A244200, A244205 Monoclonal antibodies for B cell depletion rely on their binding affinity and ability to clear bound cells through mechanisms such as antibody-dependent cellular cytotoxicity (ADCC), mediated by interactions between an antibody and Fc? receptors on natural killer cells or macrophages.A244210 Ublituximab is a chimeric anti-CD20 IgG1? antibody produced in the rat YB2/0 cell line to target a unique epitope and enhance ADCC compared to other approved anti-CD20 antibodies such as rituximab, ofatumumab, obinutuzumab, and ocrelizumab.A244210, A244215,A241045

Ublituximab was initially developed by LFB Group but was licensed to TG Therapeutics in 2012. It has been investigated for use in numerous B cell-dependent conditions, including chronic lymphocytic leukemia, non-Hodgkin's lymphoma, and relapsing multiple sclerosis.A241045 In December 2022, ublituximab was approved by the US FDA for the treatment of relapsing forms of multiple sclerosis, becoming the first and only anti-CD20 monoclonal antibody for multiple sclerosis allowing for administration in a one-hour infusion twice-a-year following the starting dose.L44508 The next year, June 2023, ublituximab was also approved by the EMA for the treatment of relapsing forms of multiple sclerosis in adult patients.L47486

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The estimated mean terminal half-life of ublituximab-xiiy was 22 days.[L44488]
Volume Distribusi The estimated central volume of distribution of ublituximab-xiiy was 3.18 L.[L44488]
Klirens (Clearance) -

Absorpsi

Following the administration of the approved recommended dosage of ublituximab, the geometric mean steady-state AUC was 3000 mcg/mL per day and the mean Cmax was 139 mcg/mL.L44488 In patients with relapsing multiple sclerosis, ublituximab exposure increases proportionally over a dose range of 150mg to 600mg.L44488

Metabolisme

As with other therapeutic proteins, the metabolism of ublituximab likely occurs via degradation to smaller peptides and amino acids by non-specific proteolytic enzymes.L44488

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

692 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Ublituximab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Ublituximab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Ublituximab.
Estrone Estrone may increase the thrombogenic activities of Ublituximab.
Estradiol Estradiol may increase the thrombogenic activities of Ublituximab.
Dienestrol Dienestrol may increase the thrombogenic activities of Ublituximab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Ublituximab.
Mestranol Mestranol may increase the thrombogenic activities of Ublituximab.
Estriol Estriol may increase the thrombogenic activities of Ublituximab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Ublituximab.
Quinestrol Quinestrol may increase the thrombogenic activities of Ublituximab.
Hexestrol Hexestrol may increase the thrombogenic activities of Ublituximab.
Tibolone Tibolone may increase the thrombogenic activities of Ublituximab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Ublituximab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Ublituximab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Ublituximab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Ublituximab.
Zeranol Zeranol may increase the thrombogenic activities of Ublituximab.
Equol Equol may increase the thrombogenic activities of Ublituximab.
Promestriene Promestriene may increase the thrombogenic activities of Ublituximab.
Methallenestril Methallenestril may increase the thrombogenic activities of Ublituximab.
Epimestrol Epimestrol may increase the thrombogenic activities of Ublituximab.
Moxestrol Moxestrol may increase the thrombogenic activities of Ublituximab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Ublituximab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Ublituximab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Ublituximab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Ublituximab.
Biochanin A Biochanin A may increase the thrombogenic activities of Ublituximab.
Formononetin Formononetin may increase the thrombogenic activities of Ublituximab.
Estetrol Estetrol may increase the thrombogenic activities of Ublituximab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Ublituximab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Ublituximab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Ublituximab.
Adalimumab The risk or severity of infection can be increased when Ublituximab is combined with Adalimumab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Ublituximab.
Gemtuzumab ozogamicin The risk or severity of infection can be increased when Ublituximab is combined with Gemtuzumab ozogamicin.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Ublituximab.
Infliximab The risk or severity of infection can be increased when Ublituximab is combined with Infliximab.
Trastuzumab The risk or severity of neutropenia can be increased when Trastuzumab is combined with Ublituximab.
Rituximab The risk or severity of infection can be increased when Ublituximab is combined with Rituximab.
Basiliximab The risk or severity of infection can be increased when Ublituximab is combined with Basiliximab.
Muromonab The risk or severity of infection can be increased when Ublituximab is combined with Muromonab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Ublituximab.
Ibritumomab tiuxetan The risk or severity of infection can be increased when Ublituximab is combined with Ibritumomab tiuxetan.
Tositumomab The risk or severity of infection can be increased when Ublituximab is combined with Tositumomab.
Alemtuzumab The risk or severity of infection can be increased when Ublituximab is combined with Alemtuzumab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Ublituximab.
Efalizumab The risk or severity of infection can be increased when Ublituximab is combined with Efalizumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of infection can be increased when Ublituximab is combined with Antithymocyte immunoglobulin (rabbit).
Natalizumab The risk or severity of immunosuppression can be increased when Ublituximab is combined with Natalizumab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Ublituximab.
Daclizumab The risk or severity of infection can be increased when Ublituximab is combined with Daclizumab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Ublituximab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Ublituximab.
Eculizumab The risk or severity of infection can be increased when Ublituximab is combined with Eculizumab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Ublituximab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Ublituximab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Ublituximab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Ublituximab.
Afelimomab The risk or severity of infection can be increased when Ublituximab is combined with Afelimomab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Ublituximab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Ublituximab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Ublituximab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Ublituximab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Ublituximab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Ublituximab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Ublituximab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Ublituximab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Ublituximab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Ublituximab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Ublituximab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Ublituximab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Ublituximab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Ublituximab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Ublituximab.
Briakinumab The risk or severity of infection can be increased when Ublituximab is combined with Briakinumab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Ublituximab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Ublituximab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Ublituximab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Ublituximab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Ublituximab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Ublituximab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Ublituximab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Ublituximab.
Trastuzumab emtansine The risk or severity of infection can be increased when Ublituximab is combined with Trastuzumab emtansine.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Ublituximab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Ublituximab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Ublituximab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Ublituximab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Ublituximab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Ublituximab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Ublituximab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Ublituximab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Ublituximab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Ublituximab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Ublituximab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Ublituximab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Ublituximab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Ublituximab.
Lumiliximab The risk or severity of adverse effects can be increased when Lumiliximab is combined with Ublituximab.

Target Protein

B-lymphocyte antigen CD20 MS4A1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 29609506
    Babiker HM, Glode AE, Cooke LS, Mahadevan D: Ublituximab for the treatment of CD20 positive B-cell malignancies. Expert Opin Investig Drugs. 2018 Apr;27(4):407-412. doi: 10.1080/13543784.2018.1459560. Epub 2018 Apr 3.
  • PMID: 33406479
    Graf J, Mares J, Barnett M, Aktas O, Albrecht P, Zamvil SS, Hartung HP: Targeting B Cells to Modify MS, NMOSD, and MOGAD: Part 1. Neurol Neuroimmunol Neuroinflamm. 2020 Dec 16;8(1). pii: 8/1/e918. doi: 10.1212/NXI.0000000000000918. Print 2021 Jan.
  • PMID: 33411674
    Graf J, Mares J, Barnett M, Aktas O, Albrecht P, Zamvil SS, Hartung HP: Targeting B cells to modify MS, NMOSD, and MOGAD: Part 2. Neurol Neuroimmunol Neuroinflamm. 2020 Dec 16;8(1). pii: 8/1/e919. doi: 10.1212/NXI.0000000000000919. Print 2021 Jan.
  • PMID: 32351164
    Fox E, Lovett-Racke AE, Gormley M, Liu Y, Petracca M, Cocozza S, Shubin R, Wray S, Weiss MS, Bosco JA, Power SA, Mok K, Inglese M: A phase 2 multicenter study of ublituximab, a novel glycoengineered anti-CD20 monoclonal antibody, in patients with relapsing forms of multiple sclerosis. Mult Scler. 2021 Mar;27(3):420-429. doi: 10.1177/1352458520918375. Epub 2020 Apr 30.
  • PMID: 18302712
    de Romeuf C, Dutertre CA, Le Garff-Tavernier M, Fournier N, Gaucher C, Glacet A, Jorieux S, Bihoreau N, Behrens CK, Beliard R, Vieillard V, Cazin B, Bourel D, Prost JF, Teillaud JL, Merle-Beral H: Chronic lymphocytic leukaemia cells are efficiently killed by an anti-CD20 monoclonal antibody selected for improved engagement of FcgammaRIIIA/CD16. Br J Haematol. 2008 Mar;140(6):635-43. doi: 10.1111/j.1365-2141.2007.06974.x.
  • PMID: 23958919
    Le Garff-Tavernier M, Herbi L, de Romeuf C, Nguyen-Khac F, Davi F, Grelier A, Boudjoghra M, Maloum K, Choquet S, Urbain R, Vieillard V, Merle-Beral H: Antibody-dependent cellular cytotoxicity of the optimized anti-CD20 monoclonal antibody ublituximab on chronic lymphocytic leukemia cells with the 17p deletion. Leukemia. 2014 Jan;28(1):230-3. doi: 10.1038/leu.2013.240. Epub 2013 Aug 20.
  • PMID: 33459118
    Kaplon H, Reichert JM: Antibodies to watch in 2021. MAbs. 2021 Jan-Dec;13(1):1860476. doi: 10.1080/19420862.2020.1860476.

Contoh Produk & Brand

Produk: 3 • International brands: 0
Produk
  • Briumvi
    Injection, solution, concentrate • 150 mg • Intravenous • EU • Approved
  • Briumvi
    Injection, solution, concentrate • 150 mg • Intravenous • EU • Approved
  • Briumvi
    Injection, solution, concentrate • 150 mg/6mL • Intravenous • US • Approved

Sekuens Gen/Protein (FASTA)

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