Bifeprunox

DB04888

small molecule investigational

Deskripsi

Bifeprunox is a novel atypical antipsychotic agent which, along with SLV313, aripiprazole and SSR-181507 combines minimal D2 receptor agonism with 5-HT receptor agonism.

Struktur Molekul 2D

Berat 385.4583
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

755 Data
Buprenorphine Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Hydrocodone Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Magnesium sulfate The therapeutic efficacy of Bifeprunox can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Bifeprunox may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Mirtazapine Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Orphenadrine Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Pramipexole Bifeprunox may increase the sedative activities of Pramipexole.
Ropinirole Bifeprunox may increase the sedative activities of Ropinirole.
Rotigotine Bifeprunox may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Bifeprunox.
Sodium oxybate Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Thalidomide Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Bifeprunox may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Bifeprunox is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Bifeprunox is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Bifeprunox.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Bifeprunox.
Sulpiride Bifeprunox may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Bifeprunox.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Bifeprunox.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Bifeprunox.
Mequitazine Bifeprunox may increase the arrhythmogenic activities of Mequitazine.
Tetrabenazine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Tetrabenazine.
Deutetrabenazine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Deutetrabenazine.
Ethanol Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Bifeprunox may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Bifeprunox.
Fluvoxamine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Bifeprunox is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Bifeprunox is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Bifeprunox is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Bifeprunox is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Bifeprunox is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Bifeprunox is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Seproxetine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Bifeprunox.
Indalpine The risk or severity of adverse effects can be increased when Bifeprunox is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Bifeprunox is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Bifeprunox is combined with Alaproclate.
Carbidopa The therapeutic efficacy of Carbidopa can be decreased when used in combination with Bifeprunox.
Benzatropine The therapeutic efficacy of Benzatropine can be decreased when used in combination with Bifeprunox.
Cabergoline The therapeutic efficacy of Cabergoline can be decreased when used in combination with Bifeprunox.
Tolcapone The therapeutic efficacy of Tolcapone can be decreased when used in combination with Bifeprunox.
Metixene The therapeutic efficacy of Metixene can be decreased when used in combination with Bifeprunox.
Trihexyphenidyl The therapeutic efficacy of Trihexyphenidyl can be decreased when used in combination with Bifeprunox.
Procyclidine The therapeutic efficacy of Procyclidine can be decreased when used in combination with Bifeprunox.
Profenamine The therapeutic efficacy of Profenamine can be decreased when used in combination with Bifeprunox.
Entacapone The therapeutic efficacy of Entacapone can be decreased when used in combination with Bifeprunox.
Lisuride The therapeutic efficacy of Lisuride can be decreased when used in combination with Bifeprunox.
Apomorphine The therapeutic efficacy of Apomorphine can be decreased when used in combination with Bifeprunox.
Biperiden The therapeutic efficacy of Biperiden can be decreased when used in combination with Bifeprunox.
Progabide The therapeutic efficacy of Progabide can be decreased when used in combination with Bifeprunox.
Amantadine The therapeutic efficacy of Amantadine can be decreased when used in combination with Bifeprunox.
Selegiline The therapeutic efficacy of Selegiline can be decreased when used in combination with Bifeprunox.
Memantine The therapeutic efficacy of Memantine can be decreased when used in combination with Bifeprunox.
Pergolide The therapeutic efficacy of Pergolide can be decreased when used in combination with Bifeprunox.
Bromocriptine The therapeutic efficacy of Bromocriptine can be decreased when used in combination with Bifeprunox.
Levodopa The therapeutic efficacy of Levodopa can be decreased when used in combination with Bifeprunox.
Rasagiline The therapeutic efficacy of Rasagiline can be decreased when used in combination with Bifeprunox.
3,5-Dinitrocatechol The therapeutic efficacy of 3,5-Dinitrocatechol can be decreased when used in combination with Bifeprunox.
Etilevodopa The therapeutic efficacy of Etilevodopa can be decreased when used in combination with Bifeprunox.
Safinamide The therapeutic efficacy of Safinamide can be decreased when used in combination with Bifeprunox.
Ifenprodil The therapeutic efficacy of Ifenprodil can be decreased when used in combination with Bifeprunox.
Dexetimide The therapeutic efficacy of Dexetimide can be decreased when used in combination with Bifeprunox.
Opicapone The therapeutic efficacy of Opicapone can be decreased when used in combination with Bifeprunox.
Piribedil The therapeutic efficacy of Piribedil can be decreased when used in combination with Bifeprunox.
Benserazide The therapeutic efficacy of Benserazide can be decreased when used in combination with Bifeprunox.
Tropatepine The therapeutic efficacy of Tropatepine can be decreased when used in combination with Bifeprunox.
Melevodopa The therapeutic efficacy of Melevodopa can be decreased when used in combination with Bifeprunox.
Dihydroergocryptine The therapeutic efficacy of Dihydroergocryptine can be decreased when used in combination with Bifeprunox.
Phenglutarimide The therapeutic efficacy of Phenglutarimide can be decreased when used in combination with Bifeprunox.
Mazaticol The therapeutic efficacy of Mazaticol can be decreased when used in combination with Bifeprunox.
Etybenzatropine The therapeutic efficacy of Etybenzatropine can be decreased when used in combination with Bifeprunox.
Budipine The therapeutic efficacy of Budipine can be decreased when used in combination with Bifeprunox.
Bornaprine The therapeutic efficacy of Bornaprine can be decreased when used in combination with Bifeprunox.
Etanautine The therapeutic efficacy of Etanautine can be decreased when used in combination with Bifeprunox.
Dexpramipexole The therapeutic efficacy of Dexpramipexole can be decreased when used in combination with Bifeprunox.
Amitriptyline The risk or severity of adverse effects can be increased when Amitriptyline is combined with Bifeprunox.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Bifeprunox.
Imipramine The risk or severity of adverse effects can be increased when Imipramine is combined with Bifeprunox.
Nortriptyline The risk or severity of adverse effects can be increased when Nortriptyline is combined with Bifeprunox.
Amoxapine The risk or severity of adverse effects can be increased when Amoxapine is combined with Bifeprunox.

Target Protein

5-hydroxytryptamine receptor 1A HTR1A
D(2) dopamine receptor DRD2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17659474
    Newman-Tancredi A, Cussac D, Depoortere R: Neuropharmacological profile of bifeprunox: merits and limitations in comparison with other third-generation antipsychotics. Curr Opin Investig Drugs. 2007 Jul;8(7):539-54.
  • PMID: 17692841
    Tadori Y, Kitagawa H, Forbes RA, McQuade RD, Stark A, Kikuchi T: Differences in agonist/antagonist properties at human dopamine D(2) receptors between aripiprazole, bifeprunox and SDZ 208-912. Eur J Pharmacol. 2007 Nov 28;574(2-3):103-11. Epub 2007 Aug 10.

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