Peringatan Keamanan

Acute oral toxicity (LD50): >10000 mg/kg Rat. Lowest Published Toxic Dose (TDL) Man - Route: Oral; Dose: 10 mg/kg/2W intermittent.

Prasterone

DB01708

small molecule approved investigational nutraceutical

Deskripsi

Prasterone, also known as dehydroepiandrosterone (DHEA) is a major C19 steroid produced by the adrenal cortex. It is also produced in small quantities in the testis and the ovary. Dehydroepiandrosterone (DHEA) can be converted to testosterone; androstenedione; estradiol; and estrone. Most of DHEA is sulfated (dehydroepiandrosterone sulfate) before secretion.

In the United States, DHEA or DHEAS have been advertised with claims that they may be beneficial for a wide variety of ailments. DHEA and DHEAS are readily available in the United States, where they are marketed as over-the-counter dietary supplements. In November 2016, DHEA was approved (as Intrarosa) to treat women experiencing moderate to severe pain during sexual intercourse (dyspareunia), a symptom of vulvar and vaginal atrophy (VVA), due to menopause.

In Canada, a prescription is required to buy DHEA.

Struktur Molekul 2D

Berat 288.4244
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 12 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Following a 50-mg DHEA PO dose in cynomolgus monkeys, systemic availability was only 3.1 +/- 0.4%. PMID: 12970301

Metabolisme

Hepatic. As shown by their high conversion ratios (in a study involving cynomolgus monkeys), the major circulating metabolites of DHEA are DHEA-S, androsterone glucuronide, and androstane-3 alpha,17 beta-diol-glucuronide. PMID: 12970301

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

102 Data
Testosterone The serum concentration of Testosterone can be increased when it is combined with Prasterone.
Testosterone propionate The serum concentration of Testosterone propionate can be increased when it is combined with Prasterone.
1-Testosterone The serum concentration of 1-Testosterone can be increased when it is combined with Prasterone.
4-Hydroxytestosterone The serum concentration of 4-Hydroxytestosterone can be increased when it is combined with Prasterone.
Dehydrochloromethyltestosterone The serum concentration of Dehydrochloromethyltestosterone can be increased when it is combined with Prasterone.
Boldenone The serum concentration of Boldenone can be increased when it is combined with Prasterone.
18-methyl-19-nortestosterone The serum concentration of 18-methyl-19-nortestosterone can be increased when it is combined with Prasterone.
Calusterone The serum concentration of Calusterone can be increased when it is combined with Prasterone.
Formebolone The serum concentration of Formebolone can be increased when it is combined with Prasterone.
Methyl-1-testosterone The serum concentration of Methyl-1-testosterone can be increased when it is combined with Prasterone.
5beta-dihydrotestosterone The serum concentration of 5beta-dihydrotestosterone can be increased when it is combined with Prasterone.
Testosterone succinate The serum concentration of Testosterone succinate can be increased when it is combined with Prasterone.
Mibolerone The serum concentration of Mibolerone can be increased when it is combined with Prasterone.
Testosterone cypionate The serum concentration of Testosterone cypionate can be increased when it is combined with Prasterone.
Testosterone enanthate The serum concentration of Testosterone enanthate can be increased when it is combined with Prasterone.
Testosterone undecanoate The serum concentration of Testosterone undecanoate can be increased when it is combined with Prasterone.
Testosterone enantate benzilic acid hydrazone The serum concentration of Testosterone enantate benzilic acid hydrazone can be increased when it is combined with Prasterone.
Stanolone acetate The serum concentration of Stanolone acetate can be increased when it is combined with Prasterone.
Trestolone acetate The serum concentration of Trestolone acetate can be increased when it is combined with Prasterone.
(1,2,6,7-3H)Testosterone The serum concentration of (1,2,6,7-3H)Testosterone can be increased when it is combined with Prasterone.
Drostanolone propionate The serum concentration of Drostanolone propionate can be increased when it is combined with Prasterone.
Stanolone The serum concentration of Stanolone can be increased when it is combined with Prasterone.
Diethylstilbestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Diethylstilbestrol.
Chlorotrianisene The risk or severity of adverse effects can be increased when Prasterone is combined with Chlorotrianisene.
Conjugated estrogens The risk or severity of adverse effects can be increased when Prasterone is combined with Conjugated estrogens.
Estrone The risk or severity of adverse effects can be increased when Prasterone is combined with Estrone.
Estradiol The risk or severity of adverse effects can be increased when Prasterone is combined with Estradiol.
Dienestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Dienestrol.
Ethinylestradiol The risk or severity of adverse effects can be increased when Prasterone is combined with Ethinylestradiol.
Mestranol The risk or severity of adverse effects can be increased when Prasterone is combined with Mestranol.
Estriol The risk or severity of adverse effects can be increased when Prasterone is combined with Estriol.
Estrone sulfate The risk or severity of adverse effects can be increased when Prasterone is combined with Estrone sulfate.
Quinestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Quinestrol.
Hexestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Hexestrol.
Tibolone The risk or severity of adverse effects can be increased when Prasterone is combined with Tibolone.
Synthetic Conjugated Estrogens, A The risk or severity of adverse effects can be increased when Prasterone is combined with Synthetic Conjugated Estrogens, A.
Synthetic Conjugated Estrogens, B The risk or severity of adverse effects can be increased when Prasterone is combined with Synthetic Conjugated Estrogens, B.
Polyestradiol phosphate The risk or severity of adverse effects can be increased when Prasterone is combined with Polyestradiol phosphate.
Esterified estrogens The risk or severity of adverse effects can be increased when Prasterone is combined with Esterified estrogens.
Zeranol The risk or severity of adverse effects can be increased when Prasterone is combined with Zeranol.
Equol The risk or severity of adverse effects can be increased when Prasterone is combined with Equol.
Promestriene The risk or severity of adverse effects can be increased when Prasterone is combined with Promestriene.
Methallenestril The risk or severity of adverse effects can be increased when Prasterone is combined with Methallenestril.
Epimestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Epimestrol.
Moxestrol The risk or severity of adverse effects can be increased when Prasterone is combined with Moxestrol.
Estradiol acetate The risk or severity of adverse effects can be increased when Prasterone is combined with Estradiol acetate.
Estradiol benzoate The risk or severity of adverse effects can be increased when Prasterone is combined with Estradiol benzoate.
Estradiol cypionate The risk or severity of adverse effects can be increased when Prasterone is combined with Estradiol cypionate.
Estradiol valerate The risk or severity of adverse effects can be increased when Prasterone is combined with Estradiol valerate.
Biochanin A The risk or severity of adverse effects can be increased when Prasterone is combined with Biochanin A.
Formononetin The risk or severity of adverse effects can be increased when Prasterone is combined with Formononetin.
Estetrol The risk or severity of adverse effects can be increased when Prasterone is combined with Estetrol.
Lasmiditan The serum concentration of Prasterone can be increased when it is combined with Lasmiditan.
Cenobamate The serum concentration of Prasterone can be decreased when it is combined with Cenobamate.
Tafamidis The serum concentration of Prasterone can be increased when it is combined with Tafamidis.
Ritonavir The serum concentration of Prasterone can be increased when it is combined with Ritonavir.
Haloperidol The serum concentration of Haloperidol can be increased when it is combined with Prasterone.
Tucatinib The metabolism of Tucatinib can be decreased when combined with Prasterone.
Abametapir The serum concentration of Prasterone can be increased when it is combined with Abametapir.
Satralizumab The serum concentration of Prasterone can be decreased when it is combined with Satralizumab.
Filgotinib The serum concentration of Prasterone can be increased when it is combined with Filgotinib.
Febuxostat The excretion of Prasterone can be decreased when combined with Febuxostat.
Sotorasib The serum concentration of Prasterone can be decreased when it is combined with Sotorasib.
Lemborexant The serum concentration of Lemborexant can be increased when it is combined with Prasterone.
Hydroxyzine The metabolism of Hydroxyzine can be decreased when combined with Prasterone.
Clindamycin The metabolism of Clindamycin can be decreased when combined with Prasterone.
Capmatinib The serum concentration of Capmatinib can be increased when it is combined with Prasterone.
Selpercatinib The serum concentration of Selpercatinib can be increased when it is combined with Prasterone.
Somatrogon The metabolism of Prasterone can be increased when combined with Somatrogon.
Roxadustat The serum concentration of Prasterone can be increased when it is combined with Roxadustat.
Pacritinib The serum concentration of Prasterone can be increased when it is combined with Pacritinib.
Oteseconazole The serum concentration of Prasterone can be increased when it is combined with Oteseconazole.
Mavacamten The serum concentration of Prasterone can be decreased when it is combined with Mavacamten.
Viloxazine The metabolism of Prasterone can be decreased when combined with Viloxazine.
Ivosidenib The metabolism of Prasterone can be increased when combined with Ivosidenib.
Dabrafenib The serum concentration of Prasterone can be decreased when it is combined with Dabrafenib.
Stiripentol The metabolism of Prasterone can be decreased when combined with Stiripentol.
Enzalutamide The serum concentration of Prasterone can be decreased when it is combined with Enzalutamide.
Telotristat ethyl The serum concentration of Prasterone can be decreased when it is combined with Telotristat ethyl.
Rilpivirine The serum concentration of Rilpivirine can be increased when it is combined with Prasterone.
Avanafil The serum concentration of Avanafil can be increased when it is combined with Prasterone.
Pretomanid The serum concentration of Prasterone can be increased when it is combined with Pretomanid.
Elacestrant The serum concentration of Prasterone can be increased when it is combined with Elacestrant.
Omaveloxolone The serum concentration of Prasterone can be decreased when it is combined with Omaveloxolone.
Apalutamide The serum concentration of Prasterone can be decreased when it is combined with Apalutamide.
Trofinetide The serum concentration of Prasterone can be increased when it is combined with Trofinetide.
Leniolisib The excretion of Prasterone can be decreased when combined with Leniolisib.
Ivacaftor The serum concentration of Prasterone can be increased when it is combined with Ivacaftor.
Erythromycin The serum concentration of Prasterone can be increased when it is combined with Erythromycin.
Elexacaftor The serum concentration of Prasterone can be increased when it is combined with Elexacaftor.
Epcoritamab The serum concentration of Prasterone can be increased when it is combined with Epcoritamab.
Vadadustat The serum concentration of Prasterone can be increased when it is combined with Vadadustat.
Fedratinib The serum concentration of Prasterone can be increased when it is combined with Fedratinib.
Glofitamab The serum concentration of Prasterone can be increased when it is combined with Glofitamab.
Ritlecitinib The serum concentration of Prasterone can be increased when it is combined with Ritlecitinib.
Momelotinib The serum concentration of Prasterone can be increased when it is combined with Momelotinib.
Bosutinib The serum concentration of Bosutinib can be increased when it is combined with Prasterone.
Encorafenib The serum concentration of Prasterone can be increased when it is combined with Encorafenib.
Danicopan The serum concentration of Prasterone can be increased when it is combined with Danicopan.
Ceftobiprole medocaril The serum concentration of Prasterone can be increased when it is combined with Ceftobiprole medocaril.

Target Protein

Glucose-6-phosphate 1-dehydrogenase G6PD
Estrogen receptor ESR1
Estrogen receptor beta ESR2
GABA(A) Receptor GABRA1
NMDA receptor GRIN1
Androgen receptor AR
Peroxisome proliferator-activated receptor alpha PPARA
Sigma non-opioid intracellular receptor 1 SIGMAR1
Nuclear receptor subfamily 1 group I member 2 NR1I2
Nuclear receptor subfamily 1 group I member 3 NR1I3

Referensi & Sumber

Synthesis reference: Isao Sugimoto, Yoko Sawase, "Stable preparation of water-soluble salts of dehydroepiandrosterone sulfate for parenteral administration." U.S. Patent US4061744, issued January, 1977.
Artikel (PubMed)
  • PMID: 21649617
    Baker WL, Karan S, Kenny AM: Effect of dehydroepiandrosterone on muscle strength and physical function in older adults: a systematic review. J Am Geriatr Soc. 2011 Jun;59(6):997-1002. doi: 10.1111/j.1532-5415.2011.03410.x. Epub 2011 Jun 7.
  • PMID: 19773400
    Alkatib AA, Cosma M, Elamin MB, Erickson D, Swiglo BA, Erwin PJ, Montori VM: A systematic review and meta-analysis of randomized placebo-controlled trials of DHEA treatment effects on quality of life in women with adrenal insufficiency. J Clin Endocrinol Metab. 2009 Oct;94(10):3676-81. doi: 10.1210/jc.2009-0672. Epub 2009 Sep 22.
  • PMID: 15261843
    Arlt W: Dehydroepiandrosterone and ageing. Best Pract Res Clin Endocrinol Metab. 2004 Sep;18(3):363-80.
  • PMID: 10613429
    Wallace MB, Lim J, Cutler A, Bucci L: Effects of dehydroepiandrosterone vs androstenedione supplementation in men. Med Sci Sports Exerc. 1999 Dec;31(12):1788-92.
  • PMID: 17054283
    Grimley Evans J, Malouf R, Huppert F, van Niekerk JK: Dehydroepiandrosterone (DHEA) supplementation for cognitive function in healthy elderly people. Cochrane Database Syst Rev. 2006 Oct 18;(4):CD006221.
  • PMID: 17917157
    Fuller SJ, Tan RS, Martins RN: Androgens in the etiology of Alzheimer's disease in aging men and possible therapeutic interventions. J Alzheimers Dis. 2007 Sep;12(2):129-42.
  • PMID: 14609305
    Thijs L, Fagard R, Forette F, Nawrot T, Staessen JA: Are low dehydroepiandrosterone sulphate levels predictive for cardiovascular diseases? A review of prospective and retrospective studies. Acta Cardiol. 2003 Oct;58(5):403-10.
  • PMID: 2946952
    Barrett-Connor E, Khaw KT, Yen SS: A prospective study of dehydroepiandrosterone sulfate, mortality, and cardiovascular disease. N Engl J Med. 1986 Dec 11;315(24):1519-24.
Menampilkan 8 dari 15 artikel.

Contoh Produk & Brand

Produk: 7 • International brands: 3
Produk
  • Intrarosa
    - • 6.5 mg • - • EU • Approved
  • Intrarosa
    Insert • 6.5 mg/1 • Vaginal • US • Approved
  • Intrarosa
    Insert • 6.5 mg/1 • Vaginal • US • Approved
  • Intrarosa
    Insert • 6.5 mg • Vaginal • Canada • Approved
  • Intrarosa
    Insert • 6.5 mg/1 • Vaginal • US • Approved
  • Intrarosa
    Insert • 6.5 mg/1 • Vaginal • US • Approved
  • Prastera
    Kit • - • Oral • US
International Brands
  • Biolaif
  • Fidelin — Paladin
  • OVIGYN-D — Alembic Pharmaceuicals Ltd

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