Peringatan Keamanan

Symptoms of mazindol overdose may be associated with restlessness, tremor, rapid breathing, confusion, hallucinations, panic, aggressiveness, nausea, vomiting, diarrhea, an irregular heartbeat, and seizures.

Mazindol

DB00579

small molecule approved investigational

Deskripsi

Mazindol is a tricyclic anorexigenic agent that is unrelated to and less toxic than amphetamine, but with some similar side effects. It inhibits uptake of catecholamines and blocks the binding of cocaine to the dopamine uptake transporter. Mazindol is only approved in the United States for the treatment of Duchenne muscular dystrophy, and is not marketed or available in the United States for use in the treatment of obesity.

Struktur Molekul 2D

Berat 284.74
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 10-13 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with or without food. Preferably take 1 hour before a meal. Taking with food may reduce GI disturbance.

Interaksi Obat

728 Data
Buprenorphine Mazindol may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Hydrocodone Mazindol may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Magnesium sulfate The therapeutic efficacy of Mazindol can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Mazindol may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Mazindol may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Orphenadrine Mazindol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Mazindol may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Pramipexole Mazindol may increase the sedative activities of Pramipexole.
Ropinirole Mazindol may increase the sedative activities of Ropinirole.
Rotigotine Mazindol may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Mazindol.
Sodium oxybate Mazindol may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Mazindol may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Thalidomide Mazindol may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Mazindol may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Mazindol.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Mazindol.
Dicoumarol The risk or severity of adverse effects can be increased when Mazindol is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Mazindol is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Mazindol is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Mazindol is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Mazindol is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Mazindol is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Mazindol is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Mazindol is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Mazindol is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Mazindol is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Mazindol is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Mazindol is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Mazindol is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Mazindol is combined with (S)-Warfarin.
Tedizolid phosphate The risk or severity of serotonin syndrome can be increased when Tedizolid phosphate is combined with Mazindol.
Mirtazapine Mazindol may increase the serotonergic activities of Mirtazapine.
Ethanol Mazindol may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Mazindol may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Mazindol.
Fluvoxamine The risk or severity of adverse effects can be increased when Mazindol is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Mazindol is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Mazindol is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when Mazindol is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Mazindol is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Mazindol is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Mazindol is combined with Nefazodone.
Zimelidine The risk or severity of adverse effects can be increased when Mazindol is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Mazindol is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Mazindol is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Mazindol.
Seproxetine The risk or severity of adverse effects can be increased when Mazindol is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Mazindol is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when Mazindol is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Mazindol is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Mazindol is combined with Alaproclate.
Methylene blue Mazindol may increase the serotonergic activities of Methylene blue.
Iobenguane Mazindol can cause a decrease in the absorption of Iobenguane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zopiclone The risk or severity of adverse effects can be increased when Mazindol is combined with Zopiclone.
Reserpine The risk or severity of adverse effects can be increased when Mazindol is combined with Reserpine.
Clozapine The risk or severity of adverse effects can be increased when Mazindol is combined with Clozapine.
Thiethylperazine The risk or severity of adverse effects can be increased when Mazindol is combined with Thiethylperazine.
Sulpiride The risk or severity of adverse effects can be increased when Mazindol is combined with Sulpiride.
Remoxipride The risk or severity of adverse effects can be increased when Mazindol is combined with Remoxipride.
Prochlorperazine The risk or severity of adverse effects can be increased when Mazindol is combined with Prochlorperazine.
Triflupromazine The risk or severity of adverse effects can be increased when Mazindol is combined with Triflupromazine.
Fluphenazine The risk or severity of adverse effects can be increased when Mazindol is combined with Fluphenazine.
Moricizine The risk or severity of adverse effects can be increased when Mazindol is combined with Moricizine.
Trifluoperazine The risk or severity of adverse effects can be increased when Mazindol is combined with Trifluoperazine.
Perphenazine The risk or severity of adverse effects can be increased when Mazindol is combined with Perphenazine.
Mesoridazine The risk or severity of adverse effects can be increased when Mazindol is combined with Mesoridazine.
Acetophenazine The risk or severity of adverse effects can be increased when Mazindol is combined with Acetophenazine.
Pimozide The risk or severity of adverse effects can be increased when Mazindol is combined with Pimozide.
Chlorprothixene The risk or severity of adverse effects can be increased when Mazindol is combined with Chlorprothixene.
Alimemazine The risk or severity of adverse effects can be increased when Mazindol is combined with Alimemazine.
Periciazine The risk or severity of adverse effects can be increased when Mazindol is combined with Periciazine.
Acepromazine The risk or severity of adverse effects can be increased when Mazindol is combined with Acepromazine.
Aceprometazine The risk or severity of adverse effects can be increased when Mazindol is combined with Aceprometazine.
Molindone The risk or severity of adverse effects can be increased when Mazindol is combined with Molindone.
Pipotiazine The risk or severity of adverse effects can be increased when Mazindol is combined with Pipotiazine.
Thioproperazine The risk or severity of adverse effects can be increased when Mazindol is combined with Thioproperazine.
Thiothixene The risk or severity of adverse effects can be increased when Mazindol is combined with Thiothixene.
Osanetant The risk or severity of adverse effects can be increased when Mazindol is combined with Osanetant.
Bifeprunox The risk or severity of adverse effects can be increased when Mazindol is combined with Bifeprunox.
BL-1020 The risk or severity of adverse effects can be increased when Mazindol is combined with BL-1020.
Lumateperone The risk or severity of adverse effects can be increased when Mazindol is combined with Lumateperone.
Amisulpride The risk or severity of adverse effects can be increased when Mazindol is combined with Amisulpride.
Perospirone The risk or severity of adverse effects can be increased when Mazindol is combined with Perospirone.
Amperozide The risk or severity of adverse effects can be increased when Mazindol is combined with Amperozide.
Cyamemazine The risk or severity of adverse effects can be increased when Mazindol is combined with Cyamemazine.
Melperone The risk or severity of adverse effects can be increased when Mazindol is combined with Melperone.
Brilaroxazine The risk or severity of adverse effects can be increased when Mazindol is combined with Brilaroxazine.
Azaperone The risk or severity of adverse effects can be increased when Mazindol is combined with Azaperone.
Propiopromazine The risk or severity of adverse effects can be increased when Mazindol is combined with Propiopromazine.
Tetrahydropalmatine The risk or severity of adverse effects can be increased when Mazindol is combined with Tetrahydropalmatine.
Ecopipam The risk or severity of adverse effects can be increased when Mazindol is combined with Ecopipam.

Target Protein

Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent dopamine transporter SLC6A3
Sodium-dependent serotonin transporter SLC6A4
Synaptic vesicular amine transporter SLC18A2

Referensi & Sumber

Synthesis reference: U.S. Patents 3,597,445 and 3,763,178.

Contoh Produk & Brand

Produk: 2 • International brands: 4
Produk
  • Sanorex
    Tablet • 1 mg • Oral • Canada • Approved
  • Sanorex
    Tablet • 2 mg • Oral • Canada • Approved
International Brands
  • Dimagrir — Gador
  • Fagolip Plus — Cetus
  • Mazanor — Kwang Dong
  • Teronac — Novartis

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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