Hasil Filter

48

Total database: 17430
Struktur (SMILES)
48 (100.0%)
Target
32 (66.7%)
Genomik
3 (6.2%)
Referensi
48 (100.0%)

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Hasil Pencarian (48)

small molecule | CAS: 1986-47-6

A propylamine formed from the cyclization of the side chain of amphetamine. This monoamine oxidase inhibitor is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It also is useful in panic and phobic disorders. (From…

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22004-32-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +5
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 185562-00-9

2,5-Dimethoxy-4-ethylthioamphetamine (ALEPH-2) is a phenylisopropylamine derivative with alleged anxiolytic and hallucinogenic properties.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +10
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2801-68-5

Deskripsi belum tersedia.

Kategori:
AminesEthylaminesPhenethylamines
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1082-88-8

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 74698-37-6

MDI-P has demonstrated potent anti-HIV activity. MDI-P has been shown to be effective in killing HIV in cell culture. HIV is the virus that causes acquired immune deficiency syndrome (AIDS). MDI-P is also a potential therapeutic agent for the treatment of the…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 32156-26-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +13
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 64-13-1

Deskripsi belum tersedia.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +12
Target Protein:
Sodium-dependent dopamine transporterAlpha-1D adrenergic receptorSodium-dependent serotonin transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15588-95-1

A psychedelic phenyl isopropylamine derivative, commonly called DOM, whose mood-altering effects and mechanism of action may be similar to those of LSD.

Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amfecloral DB08924
small molecule | CAS: 5581-35-1

Amfecloral is a stimulant drug of the phenethylamine and amphetamine chemical classes. For a short period of time, it was available under the brand Acutran and indicated as an appetite suppressant, but this product no longer exists. It acts as a prodrug which…

Waktu Paruh-
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Genetik -
Aminorex DB01490
small molecule | CAS: 2207-50-3

Aminorex is an amphetamine-like anorectic agent. It may cause pulmonary hypertension.

Kategori:
Oxazoles
Waktu Paruh-
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Genetik -
Amphetamine Approved DB00182
small molecule | CAS: 300-62-9

Amphetamine, a compound discovered over 100 years ago, is one of the more restricted controlled drugs. It was previously used for a large variety of conditions and this changed until this point where its use is highly restricted. Amphetamine, with the chemica…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +31
Target Protein:
Synaptic vesicular amine transporterSodium-dependent dopamine transporterCocaine- and amphetamine-regulated transcript protein +8
Waktu ParuhThe half-life of am…
Vol. DistribusiAmphetamine is repo…
KlirensThe reported normal…
Genetik -
Atomoxetine Approved DB00289
small molecule | CAS: 83015-26-3

Atomoxetine is a selective norepinephrine (NE) reuptake inhibitor used for the treatment of attention deficit hyperactivity disorder (ADHD). Also known as the marketed product Strattera, atomoxetine is used with other treatment modalities (psychological, educ…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterNMDA receptor +2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe clearance rate …
Genetik 6 Varian
Barbexaclone DB09001
small molecule | CAS: 4388-82-3

Barbexaclone, a salt compound of propylhexedrine and phenobarbital, is a potent antiepileptic. By weight, barbexaclone is 40% propylhexedrine and 60% phenobarbital. While barbexaclone has sedative properties, propylhexedrine has psychostimulant properties in…

Kategori:
AnticonvulsantsBarbituratesBarbiturates and Derivatives +8
Waktu ParuhAfter IV administra…
Vol. DistribusiIn mice, the volume…
Klirens-
Genetik -
Benzphetamine Approved DB00865
small molecule | CAS: 156-08-1

A sympathomimetic agent with properties similar to dextroamphetamine. It is used in the treatment of obesity. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1222)

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +28
Target Protein:
Synaptic vesicular amine transporterAlpha-2A adrenergic receptorAlpha-1A adrenergic receptor +1
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Cathine DB01486
small molecule | CAS: 492-39-7

Cathine, also known as d-norpseudoephedrine and (+)-norpseudoephedrine, is a psychoactive drug with stimulant properties. It belongs to the phenethylamine and amphetamine chemical classes. In the United States, it is classified as a Schedule IV controlled sub…

Kategori:
AlcoholsAlimentary Tract and MetabolismAmines +7
Waktu Paruh5.2 +/- 3.4 hours
Vol. Distribusi-
Klirens-
Genetik -
Cathinone DB01560
small molecule | CAS: 71031-15-7

Cathinone is a monoamine alkaloid found in the shrub Catha edulis (Khat). Closely related to ephedrine, cathine and other amphetamines, it is probably the main contributor to the stimulant effect of Catha edulis. Cathinone differs from many other amphetamines…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCentral Nervous System Stimulants +1
Waktu Paruh-
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Genetik -
small molecule | CAS: 461-78-9

A sympathomimetic agent that was formerly used as an anorectic. It has properties similar to those of dextroamphetamine. It has been implicated in lipid storage disorders and pulmonary hypertension. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1223)

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +7
Target Protein:
Sodium-dependent serotonin transporter
Waktu Paruh40 hours
Vol. Distribusi-
Klirens-
Genetik -
Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Dextroamphetamine Approved DB01576
small molecule | CAS: 51-64-9

Dextroamphetamine is the dextrorotatory enantiomer of amphetamine[A2505]. Dextroamphetamine was approved by the FDA in 2001 for the treatment of attention deficit hyperactivity disorder[L6010,Label].

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +19
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +3
Waktu Paruh11.75 hours.[Label]…
Vol. Distribusi195L.[A177247]
Klirens17L/h.[A177247]
Genetik -
Etilamfetamine DB13285
small molecule | CAS: 457-87-4

Etilamfetamine is also known as N-ethylamphetamine and is in the Canadian Legislation - The Controlled Drugs and Substances Act, and is a Schedule 1 controlled drug. Like other amphetamines, this amphetamine analog was used as an appetite suppressant in the 1…

Kategori:
Alimentary Tract and MetabolismAntiobesity Preparations, Excl. Diet ProductsCentrally Acting Antiobesity Products
Waktu Paruh-
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Genetik -
Etryptamine DB01546
small molecule | CAS: 2235-90-7

In the 1960's, alpha-ethyltryptamine (?ET), a non hydrazine reversible monoamine oxidase inhibitor, was developed in the United States by the Upjohn chemical company for use as an antidepressant. ?ET was an FDA approved antidepressant under the name Monase. H…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
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Genetik -
Famprofazone DB16702
small molecule | CAS: 22881-35-2

Famprofazone is a nonsteroidal anti-inflammatory agent found in combination products such as ‘Gewodin’ which is marketed in Taiwan.[L34724] It is important to note that the drug is metabolized to [methamphetamine] and [amphetamine] in the body and can lead to…

Kategori:
AminesAmphetaminesAnalgesics +7
Waktu Paruh-
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Genetik -
Fencamfamin DB01463
small molecule | CAS: 1209-98-9

Fencamfamin (Glucoenergan, Reactivan) is a stimulant which was developed in the 1960s as an appetite suppressant, but was later withdrawn for this application due to problems with dependence and abuse. It is around half the potency of [dexamphetamine], and is…

Kategori:
Bridged-Ring CompoundsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Sodium-dependent dopamine transporterD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenproporex DB01550
small molecule | CAS: 16397-28-7

Fenproporex is an orally active stimulant drug, which was developed in the 1960s. It is used as an appetite suppressant and a treatment for obesity. It is listed as an illicit substance in many countries due to addiction issues and listed as a prohibited subs…

Kategori:
AminesDrugs that are Mainly Renally ExcretedEthylamines +2
Waktu Paruh-
Vol. Distribusi-
KlirensThe amphetamine met…
Genetik -
Hydroxyamphetamine Approved DB09352
small molecule | CAS: 103-86-6

Hydroxyamphetamine is a derivative of amphetamines. Hydroxyamphetamine is intended mainly as local eye drops for diagnostic purposes. It is indirect sympathomimetic agent which cause dilation of the eye pupil before diagnostic test. Among the minor side effe…

Kategori:
Adrenergic AgonistsAminesAmphetamines +7
Target Protein:
Trace amine-associated receptor 1
Waktu Paruh-
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Indopan DB01446
small molecule | CAS: 299-26-3

Indopan (alpha-methyltryptamine) is a stimulant and psychoactive drug which produces effects similar to 3,4-methylenedioxy-N-methylamphetamine (MDMA), despite being structurally dissimilar. It was developed in the 1960's by Upjohn with the intention for use a…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
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Genetik -
Levmetamfetamine Approved DB09571
small molecule | CAS: 33817-09-3

Levomethamphetamine, the L-enantiomer of methamphetamine is a sympathomimetic vasoconstrictor used in some over-the-counter (OTC) nasal decongestant inhalers in the United States.

Waktu ParuhThe elimination hal…
Vol. Distribusi-
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Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Mazindol Approved DB00579
small molecule | CAS: 22232-71-9

Mazindol is a tricyclic anorexigenic agent that is unrelated to and less toxic than [amphetamine], but with some similar side effects. It inhibits uptake of catecholamines and blocks the binding of cocaine to the dopamine uptake transporter. Mazindol is only …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlimentary Tract and Metabolism +19
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporterSodium-dependent serotonin transporter +1
Waktu Paruh10-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Mephedrone DB13108
small molecule | CAS: 1189805-46-6

Mephedrone has been investigated in Alcohol-Related Disorders and Amphetamine-Related Disorders.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mephentermine Approved DB01365
small molecule | CAS: 100-92-5

A sympathomimetic agent with mainly indirect effects on adrenergic receptors. It is used to maintain blood pressure in hypotensive states, for example, following spinal anesthesia. Although the central stimulant effects of mephentermine are much less than tho…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
Alpha adrenergic receptorD(2) dopamine receptorBeta adrenergic receptor
Waktu Paruh17 to 18 hours.
Vol. Distribusi-
Klirens-
Genetik -
Metamfetamine Approved DB01577
small molecule | CAS: 537-46-2

Metamfetamine (methamphetamine) is a psychostimulant and sympathomimetic drug, and a member of the amphetamine group of sympathomimetic amines. Methamphetamine can induce effects such as euphoria, increased alertness and energy, and enhanced self-esteem. It i…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +33
Target Protein:
D(2) dopamine receptorAlpha-1B adrenergic receptorSodium-dependent dopamine transporter +10
Gen Terkait:
PICK1
Waktu ParuhThe biological half…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Methoxyphenamine Approved DB13624
small molecule | CAS: 93-30-1

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +12
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 82801-81-8

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAminesAmphetamines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylphenidate Approved DB00422
small molecule | CAS: 113-45-1

Methylphenidate is a central nervous system stimulant used most commonly in the treatment of Attention-Deficit/Hyperactivity Disorder (ADHD) and for narcolepsy. Also known as the marketed products Ritalin, Concerta, or Biphentin, methylphenidate is used with …

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +17
Target Protein:
Sodium-dependent dopamine transporter5-hydroxytryptamine receptor 1ASodium-dependent noradrenaline transporter
Waktu ParuhConcerta: The half-…
Vol. DistribusiConcerta: Plasma me…
KlirensThe apparent mean s…
Genetik -
Midomafetamine DB01454
small molecule | CAS: 42542-10-9

An N-substituted amphetamine analog. It is a widely abused drug classified as a hallucinogen and causes marked, long-lasting changes in brain serotonergic systems. It is commonly referred to as MDMA or ecstasy. It is a widely abused drug classified as a hallu…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +20
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter +4
Waktu Paruh6–10 (though durati…
Vol. Distribusi-
Klirens-
Genetik -
MMDA DB01442
small molecule | CAS: 13674-05-0

MMDA, or 3-methoxy-4,5-methylenedioxyamphetamine, is a member of the amphetamine drug class with stimulant and psychedelic properties. It also acts as an entheogen and an entactogen. MMDA bears resemblance to the psychopharmacologically active essential oils …

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +11
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent dopamine transporterSodium-dependent serotonin transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naloxone Approved DB01183
small molecule | CAS: 465-65-6

Naloxone is an opioid antagonist medication used to block or reverse the effects of opioid drugs, particularly within the setting of drug overdoses which are rapidly becoming a leading cause of death worldwide.[A234594] More specifically, naloxone has a high …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnalgesics +27
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe mean half life …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of na…
Genetik -
Phendimetrazine Approved DB01579
small molecule | CAS: 634-03-7

Phendimetrazine is a weight loss medication. Phendimetrazine is chemically related to amphetamines and is a Schedule III drug under the Convention on Psychotropic Substances and in the US since 1970.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Alpha-1A adrenergic receptorSodium-dependent noradrenaline transporterAlpha-1B adrenergic receptor
Waktu Paruh19-24 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenmetrazine Approved DB00830
small molecule | CAS: 134-49-6

A sympathomimetic drug used primarily as an appetite depressant. Its actions and mechanisms are similar to dextroamphetamine.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnti-Obesity Agents +8
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Phentermine Approved DB00191
small molecule | CAS: 122-09-8

Phentermine is a sympathomimetic amine anorectic agent and it was introduced in 1959 as part of an anti-obesity combination drug.[A174361, A174364] It is chemically related to amphetamine and it is commonly referred to as an atypical amphetamine.[A174370] Phe…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +22
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Phenylacetic acid Approved DB09269
small molecule | CAS: 103-82-2

Phenylacetic acid is an organic compound containing a phenyl functional group and a carboxylic acid functional group. It is a white solid with a disagreeable odor. Because it is used in the illicit production of phenylacetone (used in the manufacture of subst…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmmonium Ion Binding Activity +5
Waktu Paruh-
Vol. Distribusi19.2 ± 3.3 L.
Klirens-
Genetik -
Serdexmethylphenidate Approved DB16629
small molecule | CAS: 1996626-29-9

Attention Deficit Hyperactivity Disorder (ADHD) is an early-onset neurodevelopmental disorder that often extends into adulthood and is characterized by developmentally inappropriate and impaired attention, impulsivity, and motor hyperactivity.[A230698, A23070…

Kategori:
Agents that produce hypertensionCentral Nervous System AgentsCentral Nervous System Stimulants +12
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 1A
Waktu ParuhFollowing a single …
Vol. DistribusiSerdexmethylphenida…
KlirensSerdexmethylphenida…
Genetik -
Sibutramine Approved DB01105
small molecule | CAS: 106650-56-0

Sibutramine (trade name Meridia in the USA, Reductil in Europe and other countries), usually as sibutramide hydrochloride monohydrate, is an orally administered agent for the treatment of obesity. It is a centrally acting stimulant chemically related to amphe…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +23
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Gen Terkait:
GNB3
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens* Oral cl=1750 L/h …
Genetik 1 Varian
Tenamfetamine DB01509
small molecule | CAS: 4764-17-4

An amphetamine derivative that inhibits uptake of catecholamine neurotransmitters. It is a hallucinogen. It is less toxic than its methylated derivative but in sufficient doses may still destroy serotonergic neurons and has been used for that purpose experime…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tranylcypromine Approved DB00752
small molecule | CAS: 155-09-9

A propylamine formed from the cyclization of the side chain of amphetamine. This monoamine oxidase inhibitor is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It also is useful in panic and phobic disorders (From …

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +32
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh1.5-3.2 hours in pa…
Vol. Distribusi1.1-5.7 L/kg
Klirens-
Genetik -
Tropicamide Approved DB00809
small molecule | CAS: 1508-75-4

Tropicamide is an alkaloid atropine?derived anticholinergic drug and a non?selective antagonist of muscarinic acetylcholine (mACh) receptors.[A230103] Usually available in ophthalmic formulations, tropicamide is used to cause mydriasis and cycloplegia for eye…

Kategori:
Anticholinergic AgentsAutonomic AgentsCholinergic Agents +8
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhTropicamide has a p…
Vol. DistribusiNo information can …
KlirensNo information can …
Genetik -