Peringatan Keamanan

There is limited information regarding acute toxicity (LD50) of daxibotulinumtoxinA. The estimated human LD50 of botulinum toxins falls ranges from 1 to 3 ng/kg.L47860

Excessive doses of daxibotulinumtoxinA may produce neuromuscular weakness with a variety of symptoms. Respiratory support may be required where excessive doses cause paralysis of the respiratory muscles. In the event of an overdose, the patient should be medically monitored for symptoms of excessive muscle weakness or muscle paralysis. Symptomatic treatment may be necessary. Symptoms of overdose are not likely to be present immediately following injection. Should accidental injection or oral ingestion occur, the person should be medically supervised for several weeks for signs and symptoms of excessive muscle weakness or paralysis. The antitoxin raised against botulinum toxin may be requested through the Centers for Disease Control and Prevention (CDC) in the US; however, the antitoxin will not reverse any botulinum toxin-induced effects already apparent by the time of antitoxin administration.L47840

DaxibotulinumtoxinA

DB17929

biotech approved

Deskripsi

DaxibotulinumtoxinA is an acetylcholine release inhibitor and neuromuscular blocking agent. It is a botulinum toxin without accessory proteins purified from the bacterium Clostridium botulinum type A,L47840 the gram-positive anaerobic bacterium primarily present in soil. C. botulinum is known to produce toxins that can cause botulism in humans.A261075, L47860

DaxibotulinumtoxinA was first approved by the FDA on September 8, 2022, for the temporary improvement of glabellar lines.L47865 On August 14, 2023, the drug was also approved for the treatment of cervical dystonia.L47870 DAXI or DAXXIFY, a product of daxibotulinumtoxinA, incorporates RTP004, a proprietary synthetic stabilizing peptide for enhanced product stability.A261080, A261085

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Using currently available analytical technology, it is not possible to detect daxibotulinumtoxinA in the peripheral blood following intramuscular injection at the recommended dose.L47840 Botulinum toxins are predominantly absorbed at the injection site.L47860

Metabolisme

Botulinum toxins may be degraded by circulating proteases or dislodged and transported via the bloodstream to the liver for cleavage and conjugation.L47860

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

365 Data
Capreomycin The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Capreomycin.
Botulinum toxin type B Botulinum toxin type B may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Botulinum toxin type A Botulinum toxin type A may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Cyclosporine The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Cyclosporine.
Doxycycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Doxycycline.
Lymecycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Lymecycline.
Piperacillin The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Piperacillin.
Framycetin Framycetin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Clomocycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Clomocycline.
Quinine Quinine may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Vancomycin The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Vancomycin.
Tigecycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Tigecycline.
Oxytetracycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Oxytetracycline.
Chloroquine The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Chloroquine.
Demeclocycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Demeclocycline.
Magnesium sulfate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium sulfate.
Mecamylamine Mecamylamine may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Tobramycin Tobramycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Tetracycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Tetracycline.
Gentamicin Gentamicin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Colistin Colistin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Etacrynic acid The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Etacrynic acid.
Quinidine Quinidine may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Metacycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Metacycline.
Netilmicin Netilmicin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Neomycin Neomycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Minocycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Minocycline.
Procainamide The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Procainamide.
Streptomycin Streptomycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Colistimethate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Colistimethate.
Kanamycin Kanamycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Clindamycin The risk or severity of neuromuscular blockade can be increased when Clindamycin is combined with DaxibotulinumtoxinA.
Dantrolene Dantrolene may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Rolitetracycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Rolitetracycline.
Magnesium oxide The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium oxide.
Magnesium cation The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium cation.
Paromomycin Paromomycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Lincomycin The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Lincomycin.
Ribostamycin Ribostamycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Geneticin Geneticin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Apramycin Apramycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Gentamicin C1a Gentamicin C1a may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Neamine Neamine may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Arbekacin Arbekacin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Viomycin The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Viomycin.
Puromycin Puromycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Magnesium hydroxide The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium hydroxide.
Magnesium trisilicate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium trisilicate.
Magnesium chloride The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium chloride.
Magnesium acetate tetrahydrate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium acetate tetrahydrate.
Magnesium carbonate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium carbonate.
Magnesium citrate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium citrate.
Magnesium glycinate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium glycinate.
Magnesium Aluminum Silicate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium Aluminum Silicate.
Dihydrostreptomycin Dihydrostreptomycin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Hygromycin B Hygromycin B may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Sisomicin Sisomicin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Plazomicin Plazomicin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Magnesium silicate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium silicate.
Penimepicycline The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Penimepicycline.
Magnesium aspartate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium aspartate.
Isepamicin Isepamicin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.
Magnesium gluconate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium gluconate.
Magnesium orotate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium orotate.
Magnesium phosphate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium phosphate.
Magnesium acetate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium acetate.
Magnesium stearate The therapeutic efficacy of DaxibotulinumtoxinA can be increased when used in combination with Magnesium stearate.
Digoxin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Digoxin.
Acetyldigitoxin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Acetyldigitoxin.
Deslanoside The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Deslanoside.
Ouabain The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Ouabain.
Digitoxin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Digitoxin.
Oleandrin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Oleandrin.
Cymarin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Cymarin.
Proscillaridin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Proscillaridin.
Metildigoxin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Metildigoxin.
Lanatoside C The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Lanatoside C.
Gitoformate The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Gitoformate.
Acetyldigoxin The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Acetyldigoxin.
Peruvoside The risk or severity of Cardiac Arrhythmia can be increased when DaxibotulinumtoxinA is combined with Peruvoside.
Phenytoin The therapeutic efficacy of DaxibotulinumtoxinA can be decreased when used in combination with Phenytoin.
Fosphenytoin The therapeutic efficacy of DaxibotulinumtoxinA can be decreased when used in combination with Fosphenytoin.
Flunisolide The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Flunisolide.
Fluorometholone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Fluorometholone.
Beclomethasone dipropionate The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Beclomethasone dipropionate.
Betamethasone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Betamethasone.
Desoximetasone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Desoximetasone.
Fluticasone propionate The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Fluticasone propionate.
Fluocinolone acetonide The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Fluocinolone acetonide.
Triamcinolone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Triamcinolone.
Prednisone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Prednisone.
Flumethasone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Flumethasone.
Fludrocortisone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Fludrocortisone.
Hydrocortisone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Hydrocortisone.
Mometasone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Mometasone.
Prednisolone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Prednisolone.
Methylprednisolone The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Methylprednisolone.
Clobetasol propionate The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Clobetasol propionate.
Fluocinonide The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Fluocinonide.
Trilostane The risk or severity of myopathy and weakness can be increased when DaxibotulinumtoxinA is combined with Trilostane.

Target Protein

Synaptosomal-associated protein 25 SNAP25

Referensi & Sumber

Artikel (PubMed)
  • PMID: 37065981
    Mussarat A, Mustafa MS, Azam ST, Nafees Uddin MM, Nasrullah RMU, Siddiq MA: DAXI (DaxibotulinumtoxinA) - An Innovative Approach for Frown Lines. Int J Gen Med. 2023 Apr 10;16:1267-1269. doi: 10.2147/IJGM.S406563. eCollection 2023.
  • PMID: 34787840
    Solish N, Carruthers J, Kaufman J, Rubio RG, Gross TM, Gallagher CJ: Overview of DaxibotulinumtoxinA for Injection: A Novel Formulation of Botulinum Toxin Type A. Drugs. 2021 Dec;81(18):2091-2101. doi: 10.1007/s40265-021-01631-w. Epub 2021 Nov 17.
  • PMID: 31791824
    Bertucci V, Solish N, Kaufman-Janette J, Yoelin S, Shamban A, Schlessinger J, Snyder D, Gallagher C, Liu Y, Shears G, Rubio RG: DaxibotulinumtoxinA for Injection has a prolonged duration of response in the treatment of glabellar lines: Pooled data from two multicenter, randomized, double-blind, placebo-controlled, phase 3 studies (SAKURA 1 and SAKURA 2). J Am Acad Dermatol. 2020 Apr;82(4):838-845. doi: 10.1016/j.jaad.2019.06.1313. Epub 2019 Nov 29.

Contoh Produk & Brand

Produk: 17 • International brands: 0
Produk
  • Botox
    Injection, powder, lyophilized, for solution • 100 [USP'U]/1 • Intradermal; Intramuscular • US • Approved
  • Botox
    Injection, powder, lyophilized, for solution • 200 [USP'U]/1 • Intradermal; Intramuscular • US • Approved
  • BOTOX Cosmetic
    Injection, powder, lyophilized, for solution • 50 [USP'U]/1 • Intramuscular • US • Approved
  • BOTOX Cosmetic
    Injection, powder, lyophilized, for solution • 100 [USP'U]/1 • Intramuscular • US • Approved
  • Daxxify
    Injection, powder, lyophilized, for solution • 100 U/1.2mL • Intramuscular • US • Approved
  • Dysport
    Injection, powder, lyophilized, for solution • 500 U/1 • Intramuscular • US • Approved
  • Dysport
    Injection, powder, lyophilized, for solution • 300 U/1 • Intramuscular • US • Approved
  • Dysport
    Injection, powder, lyophilized, for solution • 300 U/1 • Intramuscular • US • Approved
Menampilkan 8 dari 17 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul