Peringatan Keamanan

Overdosage of letibotulinumtoxinA is likely to result in excessive neuromuscular weakness with a variety of associated symptoms. Patients should be monitored closely in the event of an overdose, and may require respiratory support if respiratory paralysis occurs.L42330

Symptoms of overdosage are not likely to be present immediately following injection, and patients should be medically supervised for several weeks for signs and symptoms of excessive muscle weakness or paralysis.L42330

LetibotulinumtoxinA

DB16820

biotech approved

Deskripsi

The aesthetic utility of botulinum toxin was discovered incidentally following its initial use in the treatment of facial spasmodic disorders in the early 1970s.A249920 The first aesthetic use of botulinum toxin was reported in 1989, when onabotulinumtoxinA (Botox) was used as a treatment for facial asymmetry resulting from iatrogenic facial nerve damage.A249920 It was subsequently approved by the FDA in 1992 for use in aesthetic procedures and has since become one of the most popular cosmetic procedures worldwide.A249920

LetibotulinumtoxinA is a type A botulinum neurotoxin produced from fermentation of Clostridium botulinum strain CBFC26.L42330 It is a 900 kDa multimeric complex comprising a 150 kDa toxin, a 130 kDa non-toxic non-haemagglutinating protein, and various other haemagglutinins.L42330 LetibotulinumtoxinA has been a market-leading cosmetic product in South Korea for a number of years and was subsequently approved in the European Union.L42335 It was approved for use in the treatment of glabellar lines in Canada in June 2022L42330,L42335 and in the US in March 2024.L50291,L50296

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Pharmacokinetic studies of letibotulinumtoxinA are not feasible due to an extremely high affinity for its pre-synaptic cholinergic binding sites - as affinity is in the picomolar range, no detectable amount of toxin appears in the blood following administration.L42330

Metabolisme

As with other exogenously administered proteins, letibotulinumtoxinA is expected to undergo non-specific enzymatic degradation to smaller peptides and amino acids.L42330

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

174 Data
Capreomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Capreomycin.
Botulinum toxin type B The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Botulinum toxin type B.
Botulinum toxin type A The risk or severity of neuromuscular blockade can be increased when Botulinum toxin type A is combined with Letibotulinumtoxina.
Cyclosporine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Cyclosporine.
Doxycycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Doxycycline.
Lymecycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Lymecycline.
Piperacillin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Piperacillin.
Framycetin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Framycetin.
Clomocycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Clomocycline.
Quinine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Quinine.
Vancomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Vancomycin.
Tigecycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Tigecycline.
Oxytetracycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Oxytetracycline.
Chloroquine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Chloroquine.
Demeclocycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Demeclocycline.
Magnesium sulfate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium sulfate.
Mecamylamine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Mecamylamine.
Tobramycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Tobramycin.
Tetracycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Tetracycline.
Gentamicin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Gentamicin.
Colistin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Colistin.
Etacrynic acid The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Etacrynic acid.
Quinidine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Quinidine.
Metacycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Metacycline.
Netilmicin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Netilmicin.
Neomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Neomycin.
Minocycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Minocycline.
Procainamide The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Procainamide.
Streptomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Streptomycin.
Colistimethate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Colistimethate.
Kanamycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Kanamycin.
Clindamycin The risk or severity of neuromuscular blockade can be increased when Clindamycin is combined with Letibotulinumtoxina.
Dantrolene The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Dantrolene.
Rolitetracycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Rolitetracycline.
Magnesium oxide The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium oxide.
Magnesium cation The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium cation.
Paromomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Paromomycin.
Lincomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Lincomycin.
Ribostamycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Ribostamycin.
Geneticin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Geneticin.
Apramycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Apramycin.
Gentamicin C1a The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Gentamicin C1a.
Neamine The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Neamine.
Arbekacin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Arbekacin.
Viomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Viomycin.
Puromycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Puromycin.
Magnesium hydroxide The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium hydroxide.
Magnesium trisilicate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium trisilicate.
Magnesium chloride The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium chloride.
Magnesium acetate tetrahydrate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium acetate tetrahydrate.
Magnesium carbonate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium carbonate.
Magnesium citrate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium citrate.
Magnesium glycinate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium glycinate.
Magnesium Aluminum Silicate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium Aluminum Silicate.
Dihydrostreptomycin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Dihydrostreptomycin.
Hygromycin B The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Hygromycin B.
Sisomicin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Sisomicin.
Plazomicin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Plazomicin.
Magnesium silicate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium silicate.
Penimepicycline The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Penimepicycline.
Magnesium aspartate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium aspartate.
Isepamicin The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Isepamicin.
Magnesium gluconate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium gluconate.
Magnesium orotate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium orotate.
Magnesium phosphate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium phosphate.
Magnesium acetate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium acetate.
Magnesium stearate The therapeutic efficacy of Letibotulinumtoxina can be increased when used in combination with Magnesium stearate.
Digoxin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Digoxin.
Acetyldigitoxin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Acetyldigitoxin.
Deslanoside The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Deslanoside.
Ouabain The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Ouabain.
Digitoxin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Digitoxin.
Oleandrin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Oleandrin.
Cymarin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Cymarin.
Proscillaridin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Proscillaridin.
Metildigoxin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Metildigoxin.
Lanatoside C The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Lanatoside C.
Gitoformate The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Gitoformate.
Acetyldigoxin The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Acetyldigoxin.
Peruvoside The risk or severity of Cardiac Arrhythmia can be increased when Letibotulinumtoxina is combined with Peruvoside.
Phenytoin The therapeutic efficacy of Letibotulinumtoxina can be decreased when used in combination with Phenytoin.
Fosphenytoin The therapeutic efficacy of Letibotulinumtoxina can be decreased when used in combination with Fosphenytoin.
Flunisolide The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Flunisolide.
Fluorometholone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Fluorometholone.
Beclomethasone dipropionate The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Beclomethasone dipropionate.
Betamethasone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Betamethasone.
Desoximetasone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Desoximetasone.
Fluticasone propionate The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Fluticasone propionate.
Fluocinolone acetonide The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Fluocinolone acetonide.
Triamcinolone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Triamcinolone.
Prednisone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Prednisone.
Flumethasone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Flumethasone.
Fludrocortisone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Fludrocortisone.
Hydrocortisone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Hydrocortisone.
Mometasone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Mometasone.
Prednisolone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Prednisolone.
Methylprednisolone The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Methylprednisolone.
Clobetasol propionate The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Clobetasol propionate.
Fluocinonide The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Fluocinonide.
Trilostane The risk or severity of myopathy and weakness can be increased when Letibotulinumtoxina is combined with Trilostane.

Target Protein

Synaptosomal-associated protein 25 SNAP25

Contoh Produk & Brand

Produk: 4 • International brands: 0
Produk
  • Letybo
    Injection, powder, lyophilized, for solution • 50 U/1 • Intramuscular • US • Approved
  • Letybo
    Injection, powder, lyophilized, for solution • 100 U/1 • Intramuscular • US • Approved
  • Letybo
    Powder, for solution • 50 unit / vial • Intramuscular • Canada • Approved
  • Letybo
    Powder, for solution • 100 unit / vial • Intramuscular • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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