Peringatan Keamanan

Bamlanivimab has been administered at doses of 7000 mg (ten times the authorized dose) during phase 2 clinical trials without any observed dose-limiting toxicity. In the event of an overdose, the recommended treatment is symptomatic and supportive measures; there is no antidote for bamlanivimab overdose.L20979

Bamlanivimab

DB15718

biotech approved investigational

Deskripsi

Bamlanivimab (LY-CoV555, also known as LY3819253), is a synthetic monoclonal antibody (mAb) derived from one of the first blood samples in the United States from a patient who recovered from COVID-19.A224039, L15311, L15316 Bamlanivimab is a neutralizing IgG1? mAb directed against the SARS-CoV-2 spike (S) protein, which is described to block viral entry into human cells.A224039, L15311, L15316, L20979

AbCellera initially discovered bamlanivimab in collaboration with the National Institute of Allergy and Infectious Diseases (NIAID), and subsequently further developed it in collaboration with Eli Lilly and Company. Bamlanivimab consists of two identical light chains of 214 amino acids and two identical heavy chains of 455 amino acids each; the Fc region is unmodified.L20979 Bamlanivimab is produced in Chinese Hamster Ovary (CHO) cells.L20979 Based on phase 2 clinical trial (BLAZE-1) interim results, bamlanivimab was granted Emergency Use Authorization (EUA) by the FDA on November 10, 2020.A224044, L20974 It is set to enter phase 3 clinical trials.L15316, L15321

Under the EUA granted in February 2021, bamlanivimab is used in combination with etesevimab to treat mild to moderate COVID-19 in adults and pediatric patients who are at high risk for progressing to severe COVID-19:L40179 this EUA later expanded in December 2021 to include all younger children at high risk, including newborns.L40174 The EUA currently allows bamlanivimab and etesevimab for post-exposure prophylaxis of COVID-19 in adults and children.L40179

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

As a monoclonal antibody, it is expected that bamlanivimab will be degraded by proteases in various locations throughout the body. Bamlanivimab is not metabolized by cytochrome P450 enzymes, making drug interactions unlikely.L20979

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

387 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Bamlanivimab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Bamlanivimab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Bamlanivimab.
Estrone Estrone may increase the thrombogenic activities of Bamlanivimab.
Estradiol Estradiol may increase the thrombogenic activities of Bamlanivimab.
Dienestrol Dienestrol may increase the thrombogenic activities of Bamlanivimab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Bamlanivimab.
Mestranol Mestranol may increase the thrombogenic activities of Bamlanivimab.
Estriol Estriol may increase the thrombogenic activities of Bamlanivimab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Bamlanivimab.
Quinestrol Quinestrol may increase the thrombogenic activities of Bamlanivimab.
Hexestrol Hexestrol may increase the thrombogenic activities of Bamlanivimab.
Tibolone Tibolone may increase the thrombogenic activities of Bamlanivimab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Bamlanivimab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Bamlanivimab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Bamlanivimab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Bamlanivimab.
Zeranol Zeranol may increase the thrombogenic activities of Bamlanivimab.
Equol Equol may increase the thrombogenic activities of Bamlanivimab.
Promestriene Promestriene may increase the thrombogenic activities of Bamlanivimab.
Methallenestril Methallenestril may increase the thrombogenic activities of Bamlanivimab.
Epimestrol Epimestrol may increase the thrombogenic activities of Bamlanivimab.
Moxestrol Moxestrol may increase the thrombogenic activities of Bamlanivimab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Bamlanivimab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Bamlanivimab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Bamlanivimab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Bamlanivimab.
Biochanin A Biochanin A may increase the thrombogenic activities of Bamlanivimab.
Formononetin Formononetin may increase the thrombogenic activities of Bamlanivimab.
Estetrol Estetrol may increase the thrombogenic activities of Bamlanivimab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Bamlanivimab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Bamlanivimab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Bamlanivimab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Bamlanivimab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Bamlanivimab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Bamlanivimab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Bamlanivimab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Bamlanivimab.
Trastuzumab The risk or severity of adverse effects can be increased when Trastuzumab is combined with Bamlanivimab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Bamlanivimab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Bamlanivimab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Bamlanivimab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Bamlanivimab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Bamlanivimab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Bamlanivimab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Bamlanivimab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Bamlanivimab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Bamlanivimab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Bamlanivimab.
Natalizumab The risk or severity of adverse effects can be increased when Natalizumab is combined with Bamlanivimab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Bamlanivimab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Bamlanivimab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Bamlanivimab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Bamlanivimab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Bamlanivimab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Bamlanivimab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Bamlanivimab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Bamlanivimab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Bamlanivimab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Bamlanivimab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Bamlanivimab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Bamlanivimab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Bamlanivimab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Bamlanivimab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Bamlanivimab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Bamlanivimab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Bamlanivimab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Bamlanivimab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Bamlanivimab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Bamlanivimab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Bamlanivimab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Bamlanivimab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Bamlanivimab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Bamlanivimab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Bamlanivimab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Bamlanivimab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Bamlanivimab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Bamlanivimab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Bamlanivimab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Bamlanivimab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Bamlanivimab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Bamlanivimab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Bamlanivimab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Bamlanivimab.
Trastuzumab emtansine The risk or severity of adverse effects can be increased when Trastuzumab emtansine is combined with Bamlanivimab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Bamlanivimab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Bamlanivimab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Bamlanivimab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Bamlanivimab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Bamlanivimab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Bamlanivimab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Bamlanivimab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Bamlanivimab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Bamlanivimab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Bamlanivimab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Bamlanivimab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Bamlanivimab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Bamlanivimab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Bamlanivimab.
Lumiliximab The risk or severity of adverse effects can be increased when Lumiliximab is combined with Bamlanivimab.

Target Protein

Spike glycoprotein S

Referensi & Sumber

Artikel (PubMed)
  • PMID: 33024963
    Jones BE, Brown-Augsburger PL, Corbett KS, Westendorf K, Davies J, Cujec TP, Wiethoff CM, Blackbourne JL, Heinz BA, Foster D, Higgs RE, Balasubramaniam D, Wang L, Bidshahri R, Kraft L, Hwang Y, Zentelis S, Jepson KR, Goya R, Smith MA, Collins DW, Hinshaw SJ, Tycho SA, Pellacani D, Xiang P, Muthuraman K, Sobhanifar S, Piper MH, Triana FJ, Hendle J, Pustilnik A, Adams AC, Berens SJ, Baric RS, Martinez DR, Cross RW, Geisbert TW, Borisevich V, Abiona O, Belli HM, de Vries M, Mohamed A, Dittmann M, Samanovic M, Mulligan MJ, Goldsmith JA, Hsieh CL, Johnson NV, Wrapp D, McLellan JS, Barnhart BC, Graham BS, Mascola JR, Hansen CL, Falconer E: LY-CoV555, a rapidly isolated potent neutralizing antibody, provides protection in a non-human primate model of SARS-CoV-2 infection. bioRxiv. 2020 Oct 1. doi: 10.1101/2020.09.30.318972.
  • PMID: 33113295
    Chen P, Nirula A, Heller B, Gottlieb RL, Boscia J, Morris J, Huhn G, Cardona J, Mocherla B, Stosor V, Shawa I, Adams AC, Van Naarden J, Custer KL, Shen L, Durante M, Oakley G, Schade AE, Sabo J, Patel DR, Klekotka P, Skovronsky DM: SARS-CoV-2 Neutralizing Antibody LY-CoV555 in Outpatients with Covid-19. N Engl J Med. 2020 Oct 28. doi: 10.1056/NEJMoa2029849.

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Bamlanivimab
    Solution • 700 mg / 20 mL • Intravenous • Canada • Approved
  • Bamlanivimab
    Injection, solution • 35 mg/1mL • Intravenous • US

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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