Zanidatamab

DB15471

biotech approved investigational

Deskripsi

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).A264718 It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.A264718

In November 2024, the FDA granted an accelerated approval for zanidatamab for use in previously treated unresectable or metastatic HER2-positive biliary tract cancers.L51908,L51903

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Based on population pharmacokinetic analysis, the estimated half-life of zanidatamab is approximately 21 days.[L51903]
Volume Distribusi Based on population pharmacokinetic analysis, the volume of distribution of zanidatamab is approximately 7.5 liters.[L51903]
Klirens (Clearance) Based on population pharmacokinetic analysis, the estimated clearance of zanidatamab was 0.012 L/h.[L51903]

Absorpsi

Following intravenous administration of zanidatamab, the Cmax is 600 µg/mL, the Ctrough is 178 µg/mL, and the AUC0-336h is 3976 days*µg/mL.L51903 The Cmax of zanidatamab is dose proportional and the total systemic exposure is greater than dose proportional.L51903

Metabolisme

Zanidatamab is likely metabolized via catabolic pathways to smaller peptides and amino acids.L51903

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

372 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Zanidatamab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Zanidatamab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Zanidatamab.
Estrone Estrone may increase the thrombogenic activities of Zanidatamab.
Estradiol Estradiol may increase the thrombogenic activities of Zanidatamab.
Dienestrol Dienestrol may increase the thrombogenic activities of Zanidatamab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Zanidatamab.
Mestranol Mestranol may increase the thrombogenic activities of Zanidatamab.
Estriol Estriol may increase the thrombogenic activities of Zanidatamab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Zanidatamab.
Quinestrol Quinestrol may increase the thrombogenic activities of Zanidatamab.
Hexestrol Hexestrol may increase the thrombogenic activities of Zanidatamab.
Tibolone Tibolone may increase the thrombogenic activities of Zanidatamab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Zanidatamab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Zanidatamab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Zanidatamab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Zanidatamab.
Zeranol Zeranol may increase the thrombogenic activities of Zanidatamab.
Equol Equol may increase the thrombogenic activities of Zanidatamab.
Estetrol Estetrol may increase the thrombogenic activities of Zanidatamab.
Promestriene Promestriene may increase the thrombogenic activities of Zanidatamab.
Methallenestril Methallenestril may increase the thrombogenic activities of Zanidatamab.
Epimestrol Epimestrol may increase the thrombogenic activities of Zanidatamab.
Moxestrol Moxestrol may increase the thrombogenic activities of Zanidatamab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Zanidatamab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Zanidatamab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Zanidatamab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Zanidatamab.
Biochanin A Biochanin A may increase the thrombogenic activities of Zanidatamab.
Formononetin Formononetin may increase the thrombogenic activities of Zanidatamab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Zanidatamab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Zanidatamab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Zanidatamab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Zanidatamab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Zanidatamab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Zanidatamab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Zanidatamab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Zanidatamab.
Trastuzumab The risk or severity of adverse effects can be increased when Trastuzumab is combined with Zanidatamab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Zanidatamab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Zanidatamab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Zanidatamab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Zanidatamab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Zanidatamab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Zanidatamab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Zanidatamab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Zanidatamab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Zanidatamab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Zanidatamab.
Natalizumab The risk or severity of adverse effects can be increased when Natalizumab is combined with Zanidatamab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Zanidatamab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Zanidatamab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Zanidatamab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Zanidatamab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Zanidatamab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Zanidatamab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Zanidatamab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Zanidatamab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Zanidatamab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Zanidatamab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Zanidatamab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Zanidatamab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Zanidatamab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Zanidatamab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Zanidatamab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Zanidatamab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Zanidatamab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Zanidatamab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Zanidatamab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Zanidatamab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Zanidatamab.
Hepatitis B immune globulin The risk or severity of adverse effects can be increased when Hepatitis B immune globulin is combined with Zanidatamab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Zanidatamab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Zanidatamab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Zanidatamab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Zanidatamab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Zanidatamab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Zanidatamab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Zanidatamab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Zanidatamab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Zanidatamab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Zanidatamab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Zanidatamab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Zanidatamab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Zanidatamab.
Trastuzumab emtansine The risk or severity of adverse effects can be increased when Trastuzumab emtansine is combined with Zanidatamab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Zanidatamab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Zanidatamab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Zanidatamab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Zanidatamab.
Stamulumab The risk or severity of adverse effects can be increased when Stamulumab is combined with Zanidatamab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Zanidatamab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Zanidatamab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Zanidatamab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Zanidatamab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Zanidatamab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Zanidatamab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Zanidatamab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Zanidatamab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Zanidatamab.

Target Protein

Receptor tyrosine-protein kinase erbB-2 ERBB2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 39114870
    Harding JJ, Fan J, Oh DY, Choi HJ, Kim JW, Chang HM, Bao L, Sun HC, Macarulla T, Xie F, Metges JP, Ying J, Bridgewater J, Lee MA, Tejani MA, Chen EY, Kim DU, Wasan H, Ducreux M, Bao Y, Lindsey S, Bachini M, Morement H, Boyken L, Ma J, Garfin P, Pant S: A plain language summary of the results from the phase 2b HERIZON-BTC-01 study of zanidatamab in participants with HER2-amplified biliary tract cancer. Future Oncol. 2024;20(31):2319-2329. doi: 10.1080/14796694.2024.2368952. Epub 2024 Aug 8.
  • PMID: 38266541
    Ten Haaft BH, Pedregal M, Prato J, Klumpen HJ, Moreno V, Lamarca A: Revolutionizing anti-HER2 therapies for extrahepatic cholangiocarcinoma and gallbladder cancer: Current advancements and future perspectives. Eur J Cancer. 2024 Mar;199:113564. doi: 10.1016/j.ejca.2024.113564. Epub 2024 Jan 20.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Ziihera
    Injection, powder, lyophilized, for solution • 50 mg/1mL • Intravenous • US • Approved

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