ONT-093

DB14069

small molecule investigational

Deskripsi

ONT-093 is an orally bioavailable inhibitor of P-glycoprotein (P-gp). In pre-clinical studies, ONT-093 could inhibit P-gp and reverse multidrug resistance at nM concentrations with no effect on paclitaxel pharmacokinetics.

Struktur Molekul 2D

Berat 494.683
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

160 Data
Afatinib The serum concentration of Afatinib can be increased when it is combined with ONT-093.
Bosutinib The serum concentration of Bosutinib can be increased when it is combined with ONT-093.
Brentuximab vedotin The serum concentration of Brentuximab vedotin can be increased when it is combined with ONT-093.
Colchicine The serum concentration of Colchicine can be increased when it is combined with ONT-093.
Edoxaban The serum concentration of Edoxaban can be increased when it is combined with ONT-093.
Ledipasvir The serum concentration of Ledipasvir can be increased when it is combined with ONT-093.
Naloxegol The serum concentration of Naloxegol can be increased when it is combined with ONT-093.
Pazopanib The serum concentration of Pazopanib can be increased when it is combined with ONT-093.
Prucalopride The serum concentration of Prucalopride can be increased when it is combined with ONT-093.
Ranolazine The serum concentration of Ranolazine can be increased when it is combined with ONT-093.
Silodosin The excretion of Silodosin can be decreased when combined with ONT-093.
Topotecan The serum concentration of Topotecan can be increased when it is combined with ONT-093.
Everolimus The serum concentration of Everolimus can be increased when it is combined with ONT-093.
Rifaximin The serum concentration of Rifaximin can be increased when it is combined with ONT-093.
Vincristine The excretion of Vincristine can be decreased when combined with ONT-093.
Doxorubicin The serum concentration of Doxorubicin can be increased when it is combined with ONT-093.
Betrixaban The serum concentration of Betrixaban can be increased when it is combined with ONT-093.
Pravastatin The serum concentration of Pravastatin can be increased when it is combined with ONT-093.
Sildenafil The serum concentration of Sildenafil can be increased when it is combined with ONT-093.
Morphine The serum concentration of Morphine can be increased when it is combined with ONT-093.
Tenofovir disoproxil The serum concentration of Tenofovir disoproxil can be increased when it is combined with ONT-093.
Clobazam The serum concentration of Clobazam can be increased when it is combined with ONT-093.
Quinine The serum concentration of Quinine can be increased when it is combined with ONT-093.
Toremifene The serum concentration of Toremifene can be increased when it is combined with ONT-093.
Bisoprolol The serum concentration of Bisoprolol can be increased when it is combined with ONT-093.
Simvastatin The serum concentration of Simvastatin can be increased when it is combined with ONT-093.
Mannitol The serum concentration of Mannitol can be increased when it is combined with ONT-093.
Loperamide The excretion of Loperamide can be decreased when combined with ONT-093.
Vardenafil The serum concentration of Vardenafil can be increased when it is combined with ONT-093.
Clomifene The serum concentration of Clomifene can be increased when it is combined with ONT-093.
Fexofenadine The serum concentration of Fexofenadine can be increased when it is combined with ONT-093.
Tegaserod The serum concentration of Tegaserod can be increased when it is combined with ONT-093.
Saquinavir The serum concentration of Saquinavir can be increased when it is combined with ONT-093.
Sitagliptin The serum concentration of Sitagliptin can be increased when it is combined with ONT-093.
Posaconazole The serum concentration of Posaconazole can be increased when it is combined with ONT-093.
Paliperidone The serum concentration of Paliperidone can be increased when it is combined with ONT-093.
Belinostat The serum concentration of Belinostat can be increased when it is combined with ONT-093.
Indacaterol The serum concentration of Indacaterol can be increased when it is combined with ONT-093.
Telaprevir The serum concentration of Telaprevir can be increased when it is combined with ONT-093.
Rivaroxaban The serum concentration of Rivaroxaban can be increased when it is combined with ONT-093.
Simeprevir The serum concentration of Simeprevir can be increased when it is combined with ONT-093.
Ambrisentan The serum concentration of Ambrisentan can be increased when it is combined with ONT-093.
Apixaban The serum concentration of Apixaban can be increased when it is combined with ONT-093.
Odanacatib The serum concentration of Odanacatib can be increased when it is combined with ONT-093.
Ticagrelor The serum concentration of Ticagrelor can be increased when it is combined with ONT-093.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with ONT-093.
Mirabegron The serum concentration of Mirabegron can be increased when it is combined with ONT-093.
Canagliflozin The serum concentration of Canagliflozin can be increased when it is combined with ONT-093.
Dolutegravir The serum concentration of Dolutegravir can be increased when it is combined with ONT-093.
Sofosbuvir The serum concentration of Sofosbuvir can be increased when it is combined with ONT-093.
Idelalisib The serum concentration of Idelalisib can be increased when it is combined with ONT-093.
Umeclidinium The serum concentration of Umeclidinium can be increased when it is combined with ONT-093.
Lenvatinib The serum concentration of Lenvatinib can be increased when it is combined with ONT-093.
Nintedanib The serum concentration of Nintedanib can be increased when it is combined with ONT-093.
Technetium Tc-99m sestamibi The serum concentration of Technetium Tc-99m sestamibi can be increased when it is combined with ONT-093.
Dasabuvir The serum concentration of Dasabuvir can be increased when it is combined with ONT-093.
Ombitasvir The serum concentration of Ombitasvir can be increased when it is combined with ONT-093.
Paritaprevir The serum concentration of Paritaprevir can be increased when it is combined with ONT-093.
Selexipag The serum concentration of Selexipag can be increased when it is combined with ONT-093.
Elbasvir The serum concentration of Elbasvir can be increased when it is combined with ONT-093.
Grazoprevir The serum concentration of Grazoprevir can be increased when it is combined with ONT-093.
Velpatasvir The serum concentration of Velpatasvir can be increased when it is combined with ONT-093.
Tezacaftor The serum concentration of Tezacaftor can be increased when it is combined with ONT-093.
Talinolol The serum concentration of Talinolol can be increased when it is combined with ONT-093.
Revefenacin The serum concentration of Revefenacin can be increased when it is combined with ONT-093.
Valspodar The serum concentration of Valspodar can be increased when it is combined with ONT-093.
Duvelisib The serum concentration of Duvelisib can be increased when it is combined with ONT-093.
Glasdegib The serum concentration of Glasdegib can be increased when it is combined with ONT-093.
Elagolix The serum concentration of Elagolix can be increased when it is combined with ONT-093.
Voxilaprevir The serum concentration of Voxilaprevir can be increased when it is combined with ONT-093.
Gilteritinib The serum concentration of Gilteritinib can be increased when it is combined with ONT-093.
Omadacycline The serum concentration of Omadacycline can be increased when it is combined with ONT-093.
Grapiprant The serum concentration of Grapiprant can be increased when it is combined with ONT-093.
Lusutrombopag The serum concentration of Lusutrombopag can be increased when it is combined with ONT-093.
Pibrentasvir The serum concentration of Pibrentasvir can be increased when it is combined with ONT-093.
Glecaprevir The serum concentration of Glecaprevir can be increased when it is combined with ONT-093.
Tenofovir The serum concentration of Tenofovir can be increased when it is combined with ONT-093.
Fedratinib The serum concentration of Fedratinib can be increased when it is combined with ONT-093.
Lasmiditan The serum concentration of Lasmiditan can be increased when it is combined with ONT-093.
Enfortumab vedotin The serum concentration of Enfortumab vedotin can be increased when it is combined with ONT-093.
Darolutamide The serum concentration of Darolutamide can be increased when it is combined with ONT-093.
Tazemetostat The serum concentration of Tazemetostat can be increased when it is combined with ONT-093.
Tipranavir The serum concentration of Tipranavir can be increased when it is combined with ONT-093.
Mibefradil The serum concentration of Mibefradil can be increased when it is combined with ONT-093.
Lemborexant The serum concentration of Lemborexant can be increased when it is combined with ONT-093.
Methylene blue The serum concentration of Methylene blue can be increased when it is combined with ONT-093.
Tucatinib The serum concentration of Tucatinib can be increased when it is combined with ONT-093.
Selumetinib The serum concentration of Selumetinib can be increased when it is combined with ONT-093.
Ripretinib The serum concentration of Ripretinib can be increased when it is combined with ONT-093.
Fostemsavir The serum concentration of Fostemsavir can be increased when it is combined with ONT-093.
Prednisolone phosphate The serum concentration of Prednisolone phosphate can be increased when it is combined with ONT-093.
Belantamab mafodotin The serum concentration of Belantamab mafodotin can be increased when it is combined with ONT-093.
Mefloquine The serum concentration of Mefloquine can be increased when it is combined with ONT-093.
Cethromycin The serum concentration of Cethromycin can be increased when it is combined with ONT-093.
Darunavir The serum concentration of Darunavir can be increased when it is combined with ONT-093.
Voclosporin The serum concentration of Voclosporin can be increased when it is combined with ONT-093.
Trilaciclib The serum concentration of Trilaciclib can be increased when it is combined with ONT-093.
Daptomycin The serum concentration of Daptomycin can be increased when it is combined with ONT-093.
Avanafil The serum concentration of Avanafil can be increased when it is combined with ONT-093.
Tivozanib The serum concentration of Tivozanib can be increased when it is combined with ONT-093.

Target Protein

ATP-dependent translocase ABCB1 ABCB1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16012790
    Chi KN, Chia SK, Dixon R, Newman MJ, Wacher VJ, Sikic B, Gelmon KA: A phase I pharmacokinetic study of the P-glycoprotein inhibitor, ONT-093, in combination with paclitaxel in patients with advanced cancer. Invest New Drugs. 2005 Aug;23(4):311-5. doi: 10.1007/s10637-005-1439-x.

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