MRK-409

DB13993

small molecule experimental

Deskripsi

MRK-409 is a GABA-A receptor agonist A31972.

Struktur Molekul 2D

Berat 397.39
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

663 Data
Buprenorphine MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Hydrocodone MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Magnesium sulfate The therapeutic efficacy of MRK-409 can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine MRK-409 may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Mirtazapine MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Orphenadrine MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Pramipexole MRK-409 may increase the sedative activities of Pramipexole.
Ropinirole MRK-409 may increase the sedative activities of Ropinirole.
Rotigotine MRK-409 may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with MRK-409.
Sodium oxybate MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Thalidomide MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Yohimbine The therapeutic efficacy of MRK-409 can be increased when used in combination with Yohimbine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with MRK-409.
Ethanol MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine MRK-409 may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Fluvoxamine The risk or severity of adverse effects can be increased when MRK-409 is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when MRK-409 is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when MRK-409 is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when MRK-409 is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when MRK-409 is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when MRK-409 is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when MRK-409 is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when MRK-409 is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when MRK-409 is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when MRK-409 is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when MRK-409 is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when MRK-409 is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when MRK-409 is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when MRK-409 is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when MRK-409 is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when MRK-409 is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when MRK-409 is combined with Alaproclate.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with MRK-409.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with MRK-409.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with MRK-409.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with MRK-409.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with MRK-409.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with MRK-409.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with MRK-409.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with MRK-409.
Desipramine The risk or severity of CNS depression can be increased when Desipramine is combined with MRK-409.
Pizotifen The risk or severity of CNS depression can be increased when Pizotifen is combined with MRK-409.
Dosulepin The risk or severity of CNS depression can be increased when Dosulepin is combined with MRK-409.
Zopiclone The risk or severity of adverse effects can be increased when MRK-409 is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with MRK-409.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with MRK-409.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with MRK-409.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of MRK-409.
Lorazepam The risk or severity of CNS depression can be increased when Lorazepam is combined with MRK-409.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with MRK-409.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with MRK-409.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with MRK-409.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with MRK-409.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with MRK-409.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with MRK-409.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with MRK-409.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with MRK-409.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with MRK-409.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with MRK-409.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with MRK-409.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with MRK-409.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with MRK-409.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with MRK-409.
Venlafaxine The risk or severity of CNS depression can be increased when Venlafaxine is combined with MRK-409.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with MRK-409.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with MRK-409.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with MRK-409.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with MRK-409.
Valproic acid The risk or severity of CNS depression can be increased when Valproic acid is combined with MRK-409.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with MRK-409.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with MRK-409.
Dihydroergotamine The risk or severity of CNS depression can be increased when Dihydroergotamine is combined with MRK-409.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with MRK-409.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with MRK-409.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with MRK-409.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with MRK-409.
Protriptyline The risk or severity of CNS depression can be increased when Protriptyline is combined with MRK-409.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with MRK-409.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with MRK-409.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with MRK-409.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with MRK-409.
Meprobamate The risk or severity of CNS depression can be increased when Meprobamate is combined with MRK-409.
Thiethylperazine The risk or severity of CNS depression can be increased when Thiethylperazine is combined with MRK-409.
Palonosetron The risk or severity of CNS depression can be increased when Palonosetron is combined with MRK-409.
Sulpiride The risk or severity of CNS depression can be increased when Sulpiride is combined with MRK-409.
Alprazolam The risk or severity of CNS depression can be increased when Alprazolam is combined with MRK-409.

Target Protein

Gamma-aminobutyric acid receptor subunit alpha-2 GABRA2
Gamma-aminobutyric acid receptor subunit alpha-3 GABRA3

Referensi & Sumber

Artikel (PubMed)
  • PMID: 20147571
    Atack JR, Wafford KA, Street LJ, Dawson GR, Tye S, Van Laere K, Bormans G, Sanabria-Bohorquez SM, De Lepeleire I, de Hoon JN, Van Hecken A, Burns HD, McKernan RM, Murphy MG, Hargreaves RJ: MRK-409 (MK-0343), a GABAA receptor subtype-selective partial agonist, is a non-sedating anxiolytic in preclinical species but causes sedation in humans. J Psychopharmacol. 2011 Mar;25(3):314-28. doi: 10.1177/0269881109354927. Epub 2010 Feb 10.

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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