WIN 55212-2

DB13950

small molecule experimental

Deskripsi

WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It is a potent cannabinoid receptor agonist that has been found to be a potent analgesic in a rat model of neuropathic pain. It activates p42 and p44 MAP kinase via receptor-mediated signaling.

Struktur Molekul 2D

Berat 426.516
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1561 Data
Ceritinib WIN 55212-2 may increase the bradycardic activities of Ceritinib.
Ivabradine WIN 55212-2 may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of WIN 55212-2.
Eliglustat The metabolism of Eliglustat can be decreased when combined with WIN 55212-2.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with WIN 55212-2.
Cilostazol The metabolism of Cilostazol can be decreased when combined with WIN 55212-2.
Colchicine The metabolism of Colchicine can be decreased when combined with WIN 55212-2.
Fentanyl The risk or severity of adverse effects can be increased when WIN 55212-2 is combined with Fentanyl.
Iloperidone The metabolism of Iloperidone can be decreased when combined with WIN 55212-2.
Retapamulin The metabolism of Retapamulin can be decreased when combined with WIN 55212-2.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with WIN 55212-2.
Vardenafil The metabolism of Vardenafil can be decreased when combined with WIN 55212-2.
Lovastatin The metabolism of Lovastatin can be decreased when combined with WIN 55212-2.
Cimetidine The serum concentration of WIN 55212-2 can be increased when it is combined with Cimetidine.
Clopidogrel The therapeutic efficacy of Clopidogrel can be decreased when used in combination with WIN 55212-2.
Efavirenz The serum concentration of WIN 55212-2 can be decreased when it is combined with Efavirenz.
Melatonin The therapeutic efficacy of WIN 55212-2 can be decreased when used in combination with Melatonin.
Nafcillin The therapeutic efficacy of WIN 55212-2 can be decreased when used in combination with Nafcillin.
Nitroprusside WIN 55212-2 may increase the hypotensive activities of Nitroprusside.
Dantrolene The risk or severity of hyperkalemia can be increased when Dantrolene is combined with WIN 55212-2.
Lithium citrate The risk or severity of adverse effects can be increased when WIN 55212-2 is combined with Lithium citrate.
Lithium hydroxide The risk or severity of adverse effects can be increased when WIN 55212-2 is combined with Lithium hydroxide.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with WIN 55212-2.
Alprazolam The metabolism of Alprazolam can be decreased when combined with WIN 55212-2.
Cocaine Cocaine may increase the tachycardic activities of WIN 55212-2.
Warfarin The serum concentration of Warfarin can be increased when it is combined with WIN 55212-2.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with WIN 55212-2.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with WIN 55212-2.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with WIN 55212-2.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with WIN 55212-2.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with WIN 55212-2.
Midazolam The serum concentration of Midazolam can be increased when it is combined with WIN 55212-2.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with WIN 55212-2.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with WIN 55212-2.
Boceprevir The serum concentration of WIN 55212-2 can be increased when it is combined with Boceprevir.
Ibutilide Ibutilide may increase the arrhythmogenic activities of WIN 55212-2.
Levosimendan Levosimendan may increase the arrhythmogenic activities of WIN 55212-2.
Procainamide Procainamide may increase the arrhythmogenic activities of WIN 55212-2.
Tocainide Tocainide may increase the arrhythmogenic activities of WIN 55212-2.
Flecainide Flecainide may increase the arrhythmogenic activities of WIN 55212-2.
Encainide Encainide may increase the arrhythmogenic activities of WIN 55212-2.
Ajmaline Ajmaline may increase the arrhythmogenic activities of WIN 55212-2.
Aprindine Aprindine may increase the arrhythmogenic activities of WIN 55212-2.
Azimilide Azimilide may increase the arrhythmogenic activities of WIN 55212-2.
Tedisamil Tedisamil may increase the arrhythmogenic activities of WIN 55212-2.
Vernakalant Vernakalant may increase the arrhythmogenic activities of WIN 55212-2.
Cariporide Cariporide may increase the arrhythmogenic activities of WIN 55212-2.
Sparteine Sparteine may increase the arrhythmogenic activities of WIN 55212-2.
Fasudil Fasudil may increase the arrhythmogenic activities of WIN 55212-2.
Simendan Simendan may increase the arrhythmogenic activities of WIN 55212-2.
Spiradoline Spiradoline may increase the arrhythmogenic activities of WIN 55212-2.
Pilsicainide Pilsicainide may increase the arrhythmogenic activities of WIN 55212-2.
Cicletanine Cicletanine may increase the arrhythmogenic activities of WIN 55212-2.
Cibenzoline Cibenzoline may increase the arrhythmogenic activities of WIN 55212-2.
Nizofenone Nizofenone may increase the arrhythmogenic activities of WIN 55212-2.
Prajmaline Prajmaline may increase the arrhythmogenic activities of WIN 55212-2.
Tiracizine Tiracizine may increase the arrhythmogenic activities of WIN 55212-2.
Ethacizine Ethacizine may increase the arrhythmogenic activities of WIN 55212-2.
Lorajmine Lorajmine may increase the arrhythmogenic activities of WIN 55212-2.
Bunaftine Bunaftine may increase the arrhythmogenic activities of WIN 55212-2.
Lorcainide Lorcainide may increase the arrhythmogenic activities of WIN 55212-2.
Hydroquinine Hydroquinine may increase the arrhythmogenic activities of WIN 55212-2.
Fosfructose Fosfructose may increase the arrhythmogenic activities of WIN 55212-2.
Carteolol WIN 55212-2 may increase the arrhythmogenic activities of Carteolol.
Metipranolol WIN 55212-2 may increase the arrhythmogenic activities of Metipranolol.
Bioallethrin WIN 55212-2 may increase the arrhythmogenic activities of Bioallethrin.
Hydroquinidine WIN 55212-2 may increase the arrhythmogenic activities of Hydroquinidine.
SOR-C13 WIN 55212-2 may increase the arrhythmogenic activities of SOR-C13.
Digoxin Digoxin may increase the arrhythmogenic activities of WIN 55212-2.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of WIN 55212-2.
Deslanoside Deslanoside may increase the arrhythmogenic activities of WIN 55212-2.
Cymarin Cymarin may increase the arrhythmogenic activities of WIN 55212-2.
Metildigoxin Metildigoxin may increase the arrhythmogenic activities of WIN 55212-2.
Acetyldigoxin Acetyldigoxin may increase the arrhythmogenic activities of WIN 55212-2.
Disopyramide Disopyramide may increase the arrhythmogenic activities of WIN 55212-2.
Hyoscyamine Hyoscyamine may increase the arrhythmogenic activities of WIN 55212-2.
Atropine Atropine may increase the arrhythmogenic activities of WIN 55212-2.
Nicardipine Nicardipine may increase the arrhythmogenic activities of WIN 55212-2.
Trimebutine Trimebutine may increase the arrhythmogenic activities of WIN 55212-2.
Otilonium Otilonium may increase the arrhythmogenic activities of WIN 55212-2.
Niguldipine Niguldipine may increase the arrhythmogenic activities of WIN 55212-2.
Bretylium Bretylium may increase the arrhythmogenic activities of WIN 55212-2.
Isradipine Isradipine may increase the arrhythmogenic activities of WIN 55212-2.
Diltiazem Diltiazem may increase the arrhythmogenic activities of WIN 55212-2.
Amlodipine Amlodipine may increase the arrhythmogenic activities of WIN 55212-2.
Nimodipine Nimodipine may increase the arrhythmogenic activities of WIN 55212-2.
Lercanidipine Lercanidipine may increase the arrhythmogenic activities of WIN 55212-2.
Cinnarizine Cinnarizine may increase the arrhythmogenic activities of WIN 55212-2.
Verapamil Verapamil may increase the arrhythmogenic activities of WIN 55212-2.
Losartan Losartan may increase the arrhythmogenic activities of WIN 55212-2.
Levomenthol Levomenthol may increase the arrhythmogenic activities of WIN 55212-2.
Nitrendipine Nitrendipine may increase the arrhythmogenic activities of WIN 55212-2.
Perhexiline Perhexiline may increase the arrhythmogenic activities of WIN 55212-2.
Bepridil Bepridil may increase the arrhythmogenic activities of WIN 55212-2.
Nimesulide Nimesulide may increase the arrhythmogenic activities of WIN 55212-2.
Prenylamine Prenylamine may increase the arrhythmogenic activities of WIN 55212-2.
Cyclandelate Cyclandelate may increase the arrhythmogenic activities of WIN 55212-2.
Clevidipine Clevidipine may increase the arrhythmogenic activities of WIN 55212-2.
Seletracetam Seletracetam may increase the arrhythmogenic activities of WIN 55212-2.
Nylidrin Nylidrin may increase the arrhythmogenic activities of WIN 55212-2.

Target Protein

Cannabinoid receptor 1 CNR1
Cannabinoid receptor 2 CNR2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 29113897
    Perdikaris P, Tsarouchi M, Fanarioti E, Natsaridis E, Mitsacos A, Giompres P: Long lasting effects of chronic WIN55,212-2 treatment on mesostriatal dopaminergic and cannabinoid systems in the rat brain. Neuropharmacology. 2018 Feb;129:1-15. doi: 10.1016/j.neuropharm.2017.11.005. Epub 2017 Nov 4.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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