Peringatan Keamanan

Trolamine produced mild erythema and edema in rabbits with dermally administered doses of 2 g/kg under occlusion A27174. The oral LD50 was found to be 8 g/kg in guinea pigs and 4.19-11.26 g/kg in rats. Repeated oral administration in rats and guinea pigs produced hepatic and renal damage with deaths occurring in rats at doses >0.3 g/kg/day. When inhaled trolamine produced edema and inflammation in rats at doses over 100 mg/m³ after 5 days and at doses over 4.7 mg/m³ after 90 days. There is some evidence of carcinogenicity at high dermal doses (1000 mg/kg/day) in mice. Trolamine is not classified as a carcinogen in humans.

Trolamine

DB13747

small molecule approved

Deskripsi

Trolamine, which is also referred to as triethanolamine (TEA), is a tertiary amine and a triol. It is a bifunctional compound that exhibits both properties of alcohols and amines. Trolamine contains small amounts of diethanolamine and ethanolamine and may also act as an antioxidant against the auto-oxidation of animal and vegetable fats A27174. It is commonly used as a pH adjuster and surfactant in industrial and cosmetic products such as skin and hair conditioning products.

Struktur Molekul 2D

Berat 149.1882
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Dermal absorption of trolamine increases with the dose A27174. This has been found to range from 19-28% in rats with doses of 68-276 mg/kg in 190 ?L of acetone without occlusion and from 60-80% in mice with doses of 79-1120 mg/kg in the same volume of acetone.

Metabolisme

Trolamine is excreted mostly as the unchanged compound A27174. No diethanolamine or ethanolamine has been found. Very small amounts of trolamine glucuronide have been detected but not quantified.

Rute Eliminasi

When orally administered to rats, the 53% of the trolamine dose was found to be excreted in the urine and 20% in the feces A27174. 98% was excreted in the urine with intravenous administration.

Interaksi Obat

1 Data
Tenofovir alafenamide The serum concentration of Tenofovir alafenamide can be increased when it is combined with Trolamine.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 23696578
    Fiume MM, Heldreth B, Bergfeld WF, Belsito DV, Hill RA, Klaassen CD, Liebler D, Marks JG Jr, Shank RC, Slaga TJ, Snyder PW, Andersen FA: Safety assessment of triethanolamine and triethanolamine-containing ingredients as used in cosmetics. Int J Toxicol. 2013 May-Jun;32(3 Suppl):59S-83S. doi: 10.1177/1091581813488804.

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