Loprazolam

DB13643

small molecule experimental

Deskripsi

Loprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent nocturnal awakenings. Loprazolam is recommended as a short-term therapy only, due to adverse events associated with the drug including dependence and withdrawal symptoms. It is a positive modulator of GABA-A receptor that enhances the inhibitory neurotransmission. It is not an FDA-approved drug.

Struktur Molekul 2D

Berat 464.904
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

718 Data
Buprenorphine Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Hydrocodone Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Magnesium sulfate The therapeutic efficacy of Loprazolam can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Loprazolam may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Mirtazapine Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Orphenadrine Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Pramipexole Loprazolam may increase the sedative activities of Pramipexole.
Ropinirole Loprazolam may increase the sedative activities of Ropinirole.
Rotigotine Loprazolam may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Loprazolam.
Suvorexant Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Thalidomide Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Clozapine The risk or severity of adverse effects can be increased when Loprazolam is combined with Clozapine.
Methadone Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Methadone.
Olanzapine The risk or severity of adverse effects can be increased when Loprazolam is combined with Olanzapine.
Phenytoin The serum concentration of Phenytoin can be increased when it is combined with Loprazolam.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with Loprazolam.
Sodium oxybate Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Teduglutide The serum concentration of Loprazolam can be increased when it is combined with Teduglutide.
Yohimbine The therapeutic efficacy of Loprazolam can be increased when used in combination with Yohimbine.
Flumazenil Flumazenil may decrease the sedative activities of Loprazolam.
Ethanol Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Loprazolam may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Zimelidine The risk or severity of adverse effects can be increased when Loprazolam is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Loprazolam is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Loprazolam is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Loprazolam is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Loprazolam is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Loprazolam is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Loprazolam is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Loprazolam is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Loprazolam is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Loprazolam is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Loprazolam is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Loprazolam is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Loprazolam is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Loprazolam is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Loprazolam.
Indalpine The risk or severity of adverse effects can be increased when Loprazolam is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Loprazolam is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Loprazolam is combined with Alaproclate.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Loprazolam.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Loprazolam.
Zopiclone The risk or severity of adverse effects can be increased when Loprazolam is combined with Zopiclone.
Caffeine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Caffeine.
Theophylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Theophylline.
Dyphylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Dyphylline.
Pentoxifylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Pentoxifylline.
Mercaptopurine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Mercaptopurine.
Aminophylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Aminophylline.
Oxtriphylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Oxtriphylline.
Theobromine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Theobromine.
Fenethylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Fenethylline.
8-azaguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 8-azaguanine.
7,9-Dimethylguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 7,9-Dimethylguanine.
Xanthine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Xanthine.
7-Deazaguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 7-Deazaguanine.
Guanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Guanine.
9-Methylguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 9-Methylguanine.
Peldesine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Peldesine.
Hypoxanthine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Hypoxanthine.
9-Deazaguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 9-Deazaguanine.
Propentofylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Propentofylline.
Valomaciclovir The therapeutic efficacy of Loprazolam can be decreased when used in combination with Valomaciclovir.
3-isobutyl-1-methyl-7H-xanthine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 3-isobutyl-1-methyl-7H-xanthine.
Uric acid The therapeutic efficacy of Loprazolam can be decreased when used in combination with Uric acid.
Doxofylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Doxofylline.
6-O-benzylguanine The therapeutic efficacy of Loprazolam can be decreased when used in combination with 6-O-benzylguanine.
Lisofylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Lisofylline.
Lobucavir The therapeutic efficacy of Loprazolam can be decreased when used in combination with Lobucavir.
Cafedrine The therapeutic efficacy of Loprazolam can be decreased when used in combination with Cafedrine.
Theodrenaline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Theodrenaline.
Bamifylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Bamifylline.
Proxyphylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Proxyphylline.
Acefylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Acefylline.
Etamiphylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Etamiphylline.
Pentifylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Pentifylline.
Bufylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Bufylline.
Bromotheophylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Bromotheophylline.
Furafylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with Furafylline.
8-chlorotheophylline The therapeutic efficacy of Loprazolam can be decreased when used in combination with 8-chlorotheophylline.
PCS-499 The therapeutic efficacy of Loprazolam can be decreased when used in combination with PCS-499.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Loprazolam.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Loprazolam.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Loprazolam.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Loprazolam.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Loprazolam.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Loprazolam.

Target Protein

GABA(A) Receptor GABRA1
GABA(A) Receptor Benzodiazepine Binding Site GABRA1

Referensi & Sumber

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Contoh Produk & Brand

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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