Peringatan Keamanan

Mephenesin can produce hemolysis leading to hemoglobinuria with intravenous administration of concentrations greater than 10% A32760. As a central nervous system depressant it can also produce paralysis and respiratory depression.

Mephenesin

DB13583

small molecule approved

Deskripsi

Mephenesin is a synthetic cresol glyceryl ether which produces transient muscle relaxation and paralysis via central nervous system depression A32760. It first entered use in the 1950s.

Struktur Molekul 2D

Berat 182.219
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

16 Data
Cyclobenzaprine The risk or severity of CNS depression can be increased when Cyclobenzaprine is combined with Mephenesin.
Metoclopramide The risk or severity of sedation can be increased when Metoclopramide is combined with Mephenesin.
Lasmiditan The risk or severity of adverse effects can be increased when Lasmiditan is combined with Mephenesin.
Tramadol The risk or severity of CNS depression can be increased when Mephenesin is combined with Tramadol.
Ziprasidone The risk or severity of adverse effects can be increased when Mephenesin is combined with Ziprasidone.
Haloperidol The risk or severity of CNS depression can be increased when Haloperidol is combined with Mephenesin.
Fluoxetine Mephenesin may increase the central nervous system depressant (CNS depressant) activities of Fluoxetine.
Oliceridine The risk or severity of hypotension, sedation, death, somnolence, and respiratory depression can be increased when Mephenesin is combined with Oliceridine.
Ropeginterferon alfa-2b The risk or severity of neuropsychiatric effects can be increased when Ropeginterferon alfa-2b is combined with Mephenesin.
Daridorexant The risk or severity of CNS depression can be increased when Mephenesin is combined with Daridorexant.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Mephenesin.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with Mephenesin.
Midazolam The risk or severity of sedation and CNS depression can be increased when Midazolam is combined with Mephenesin.
Ganaxolone The risk or severity of sedation, somnolence, and CNS depression can be increased when Mephenesin is combined with Ganaxolone.
Zuranolone The risk or severity of CNS depression can be increased when Zuranolone is combined with Mephenesin.
DaxibotulinumtoxinA Mephenesin may increase the neuromuscular blocking activities of DaxibotulinumtoxinA.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15421800
    Authors unspecified: NEW and nonofficial remedies; mephenesin. J Am Med Assoc. 1950 Jun 17;143(7):655.
  • PMID: 15402629
    KAADA BR: Site of action of myanesin in the central nervous system. J Neurophysiol. 1950 Jan;13(1):89-104. doi: 10.1152/jn.1950.13.1.89.
  • PMID: 4855803
    Klee MR, Faber DS: Mephenesin blocks early inward currents and strychnine-induced multiple discharges of aplysia neurons. Pflugers Arch. 1974 Feb 4;346(2):97-106.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Decontractyl Baume
    Ointment • - • Topical • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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