Peringatan Keamanan

The LD50 in rat following oral and intraperitoneal administration is 3370 mg/kg and 805 mg/kg, respectively MSDS. Subcutaneous LD50 in mouse is >5000 mg/kg MSDS. Mild skin irritation was seen in rabbits following dermal application of 750 mg/30d(l) MSDS. Non-steroidal anti-inflammatory drug (NSAID) overdose may produce nausea, vomiting, indigestion and upper abdominal pain. Other effects may include drowsiness, dizziness, confusion, disorientation, lethargy MSDS.

Bufexamac

DB13346

small molecule approved withdrawn

Deskripsi

Bufexamac is a non-steroidal anti-inflammatory drug (NSAID) under the market name Droxaryl, Malipuran, Paraderm and Parfenac. It is typically administered topically for the treatment of subacute and chronic eczema of the skin, including atopic eczema and other inflammatory dermatoses, as well as sunburn and other minor burns, and itching. It has also been used in suppositories in combination with local anaesthetics indicated for haemorrhoids. The use of bufexamac has been discontinued in Canada and the United States, which may be due to undetermined clinical efficacy and a high prevalence of contact sensitization A32822. Bufexamac was also withdrawn by the EMA in April 2010.

Struktur Molekul 2D

Berat 223.272
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) No data available.
Volume Distribusi No data available.
Klirens (Clearance) No data available.

Absorpsi

Method of application affects the extent of cutaneous absorption A27192. Following rectal administration as suppositories, the systemic absorption was reported to be low A32823.

Metabolisme

No data available.

Rute Eliminasi

Following topical administration of 5% bufexamac, the recovery in the urine was 3.5% of the applied dose within 144 hours A27192. Studies in healthy volunteers receiving an oral dose of 125 to 500 mg indicate that an average of 80% of the total dose is excreted in the urine within 48 hours A27192.

Interaksi Obat

156 Data
Aminosalicylic acid The therapeutic efficacy of Aminosalicylic acid can be decreased when used in combination with Bufexamac.
Mesalazine The risk or severity of nephrotoxicity can be increased when Mesalazine is combined with Bufexamac.
Sulfasalazine The therapeutic efficacy of Sulfasalazine can be decreased when used in combination with Bufexamac.
Diflunisal The therapeutic efficacy of Diflunisal can be decreased when used in combination with Bufexamac.
Acetylsalicylic acid The therapeutic efficacy of Acetylsalicylic acid can be decreased when used in combination with Bufexamac.
Balsalazide The therapeutic efficacy of Balsalazide can be decreased when used in combination with Bufexamac.
Olsalazine The risk or severity of nephrotoxicity can be increased when Bufexamac is combined with Olsalazine.
Bismuth subsalicylate The therapeutic efficacy of Bismuth subsalicylate can be decreased when used in combination with Bufexamac.
Dersalazine The therapeutic efficacy of Dersalazine can be decreased when used in combination with Bufexamac.
Phenyl aminosalicylate The therapeutic efficacy of Phenyl aminosalicylate can be decreased when used in combination with Bufexamac.
Methyl salicylate The therapeutic efficacy of Methyl salicylate can be decreased when used in combination with Bufexamac.
Trolamine salicylate The therapeutic efficacy of Trolamine salicylate can be decreased when used in combination with Bufexamac.
Nitroaspirin The therapeutic efficacy of Nitroaspirin can be decreased when used in combination with Bufexamac.
Aloxiprin The therapeutic efficacy of Aloxiprin can be decreased when used in combination with Bufexamac.
Guacetisal The therapeutic efficacy of Guacetisal can be decreased when used in combination with Bufexamac.
Carbaspirin calcium The therapeutic efficacy of Carbaspirin calcium can be decreased when used in combination with Bufexamac.
Choline salicylate The therapeutic efficacy of Choline salicylate can be decreased when used in combination with Bufexamac.
Thiosalicylic acid The therapeutic efficacy of Thiosalicylic acid can be decreased when used in combination with Bufexamac.
Diclofenac The risk or severity of adverse effects can be increased when Diclofenac is combined with Bufexamac.
Flurbiprofen The risk or severity of adverse effects can be increased when Flurbiprofen is combined with Bufexamac.
Bromfenac The risk or severity of adverse effects can be increased when Bromfenac is combined with Bufexamac.
Nepafenac The risk or severity of adverse effects can be increased when Nepafenac is combined with Bufexamac.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Bufexamac.
Nabumetone The risk or severity of adverse effects can be increased when Nabumetone is combined with Bufexamac.
Tenoxicam The risk or severity of adverse effects can be increased when Tenoxicam is combined with Bufexamac.
Celecoxib The risk or severity of adverse effects can be increased when Celecoxib is combined with Bufexamac.
Tolmetin The risk or severity of adverse effects can be increased when Tolmetin is combined with Bufexamac.
Rofecoxib The risk or severity of adverse effects can be increased when Rofecoxib is combined with Bufexamac.
Piroxicam The risk or severity of adverse effects can be increased when Piroxicam is combined with Bufexamac.
Fenoprofen The risk or severity of adverse effects can be increased when Fenoprofen is combined with Bufexamac.
Valdecoxib The risk or severity of adverse effects can be increased when Valdecoxib is combined with Bufexamac.
Sulindac The risk or severity of adverse effects can be increased when Sulindac is combined with Bufexamac.
Etodolac The risk or severity of adverse effects can be increased when Etodolac is combined with Bufexamac.
Mefenamic acid The risk or severity of adverse effects can be increased when Mefenamic acid is combined with Bufexamac.
Naproxen The risk or severity of adverse effects can be increased when Naproxen is combined with Bufexamac.
Phenylbutazone The risk or severity of adverse effects can be increased when Phenylbutazone is combined with Bufexamac.
Meloxicam The risk or severity of adverse effects can be increased when Meloxicam is combined with Bufexamac.
Carprofen The risk or severity of adverse effects can be increased when Carprofen is combined with Bufexamac.
Suprofen The risk or severity of adverse effects can be increased when Suprofen is combined with Bufexamac.
Salicylic acid The risk or severity of adverse effects can be increased when Salicylic acid is combined with Bufexamac.
Meclofenamic acid The risk or severity of adverse effects can be increased when Meclofenamic acid is combined with Bufexamac.
Oxaprozin The risk or severity of adverse effects can be increased when Oxaprozin is combined with Bufexamac.
Ketoprofen The risk or severity of adverse effects can be increased when Ketoprofen is combined with Bufexamac.
Ibuprofen The risk or severity of adverse effects can be increased when Ibuprofen is combined with Bufexamac.
Lumiracoxib The risk or severity of adverse effects can be increased when Lumiracoxib is combined with Bufexamac.
Magnesium salicylate The risk or severity of adverse effects can be increased when Magnesium salicylate is combined with Bufexamac.
Salsalate The risk or severity of adverse effects can be increased when Salsalate is combined with Bufexamac.
Choline magnesium trisalicylate The risk or severity of adverse effects can be increased when Choline magnesium trisalicylate is combined with Bufexamac.
Antipyrine The risk or severity of adverse effects can be increased when Antipyrine is combined with Bufexamac.
Tiaprofenic acid The risk or severity of adverse effects can be increased when Tiaprofenic acid is combined with Bufexamac.
Etoricoxib The risk or severity of adverse effects can be increased when Etoricoxib is combined with Bufexamac.
Oxyphenbutazone The risk or severity of adverse effects can be increased when Oxyphenbutazone is combined with Bufexamac.
Niflumic acid The risk or severity of adverse effects can be increased when Niflumic acid is combined with Bufexamac.
Nimesulide The risk or severity of adverse effects can be increased when Nimesulide is combined with Bufexamac.
Benoxaprofen The risk or severity of adverse effects can be increased when Benoxaprofen is combined with Bufexamac.
Zomepirac The risk or severity of adverse effects can be increased when Zomepirac is combined with Bufexamac.
Lornoxicam The risk or severity of adverse effects can be increased when Lornoxicam is combined with Bufexamac.
Aceclofenac The risk or severity of adverse effects can be increased when Aceclofenac is combined with Bufexamac.
Zaltoprofen The risk or severity of adverse effects can be increased when Zaltoprofen is combined with Bufexamac.
Azapropazone The risk or severity of adverse effects can be increased when Azapropazone is combined with Bufexamac.
Felbinac The risk or severity of adverse effects can be increased when Felbinac is combined with Bufexamac.
Parecoxib The risk or severity of adverse effects can be increased when Parecoxib is combined with Bufexamac.
Salicylamide The risk or severity of adverse effects can be increased when Salicylamide is combined with Bufexamac.
Kebuzone The risk or severity of adverse effects can be increased when Kebuzone is combined with Bufexamac.
Isoxicam The risk or severity of adverse effects can be increased when Isoxicam is combined with Bufexamac.
Indoprofen The risk or severity of adverse effects can be increased when Indoprofen is combined with Bufexamac.
Ibuproxam The risk or severity of adverse effects can be increased when Ibuproxam is combined with Bufexamac.
Floctafenine The risk or severity of adverse effects can be increased when Floctafenine is combined with Bufexamac.
Fenbufen The risk or severity of adverse effects can be increased when Fenbufen is combined with Bufexamac.
Etofenamate The risk or severity of adverse effects can be increased when Etofenamate is combined with Bufexamac.
Epirizole The risk or severity of adverse effects can be increased when Epirizole is combined with Bufexamac.
Loxoprofen The risk or severity of adverse effects can be increased when Loxoprofen is combined with Bufexamac.
Droxicam The risk or severity of adverse effects can be increased when Droxicam is combined with Bufexamac.
Tolfenamic acid The risk or severity of adverse effects can be increased when Tolfenamic acid is combined with Bufexamac.
Clonixin The risk or severity of adverse effects can be increased when Clonixin is combined with Bufexamac.
Propacetamol The risk or severity of adverse effects can be increased when Propacetamol is combined with Bufexamac.
Tepoxalin The risk or severity of adverse effects can be increased when Tepoxalin is combined with Bufexamac.
Flunixin The risk or severity of adverse effects can be increased when Flunixin is combined with Bufexamac.
Indobufen The risk or severity of adverse effects can be increased when Indobufen is combined with Bufexamac.
Tinoridine The risk or severity of adverse effects can be increased when Tinoridine is combined with Bufexamac.
Alclofenac The risk or severity of adverse effects can be increased when Alclofenac is combined with Bufexamac.
Fentiazac The risk or severity of adverse effects can be increased when Fentiazac is combined with Bufexamac.
Suxibuzone The risk or severity of adverse effects can be increased when Suxibuzone is combined with Bufexamac.
Bumadizone The risk or severity of adverse effects can be increased when Bumadizone is combined with Bufexamac.
Alminoprofen The risk or severity of adverse effects can be increased when Alminoprofen is combined with Bufexamac.
Feprazone The risk or severity of adverse effects can be increased when Bufexamac is combined with Feprazone.
Difenpiramide The risk or severity of adverse effects can be increased when Bufexamac is combined with Difenpiramide.
Nifenazone The risk or severity of adverse effects can be increased when Bufexamac is combined with Nifenazone.
Lonazolac The risk or severity of adverse effects can be increased when Bufexamac is combined with Lonazolac.
Tenidap The risk or severity of adverse effects can be increased when Bufexamac is combined with Tenidap.
Bendazac The risk or severity of adverse effects can be increased when Bufexamac is combined with Bendazac.
Pranoprofen The risk or severity of adverse effects can be increased when Bufexamac is combined with Pranoprofen.
Propyphenazone The risk or severity of adverse effects can be increased when Bufexamac is combined with Propyphenazone.
Proglumetacin The risk or severity of adverse effects can be increased when Bufexamac is combined with Proglumetacin.
Ethenzamide The risk or severity of adverse effects can be increased when Bufexamac is combined with Ethenzamide.
Mofebutazone The risk or severity of adverse effects can be increased when Bufexamac is combined with Mofebutazone.
Proquazone The risk or severity of adverse effects can be increased when Bufexamac is combined with Proquazone.
Benorilate The risk or severity of adverse effects can be increased when Bufexamac is combined with Benorilate.
Pirprofen The risk or severity of adverse effects can be increased when Bufexamac is combined with Pirprofen.
Acemetacin The risk or severity of adverse effects can be increased when Bufexamac is combined with Acemetacin.

Target Protein

Prostaglandin G/H synthase 1 PTGS1
Prostaglandin G/H synthase 2 PTGS2
Histone deacetylase 6 HDAC6
Polyamine deacetylase HDAC10 HDAC10

Referensi & Sumber

Artikel (PubMed)

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Norfemac Cream - 5%
    Cream • 5 % • Topical • Canada • OTC • Approved
  • Norfemac Ointment - 5%
    Ointment • 5 % • Topical • Canada • OTC • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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