Peringatan Keamanan

The administration of more than 50 meq of magnesium daily can produce the development of hypermagnesemia. This can provoke the formation of bladder and renal calculi. There is no known toxicity and the LD50 in animals are higher than 500 mg/kg in humans.T186 It is determined that magnesium silicate is not carcinogenic.L2614

Magnesium silicate

DB13249

small molecule approved

Deskripsi

Magnesium silicate is a compound of magnesium oxide and silicon. It is the magnesium salt of silicic acid containing an unspecified amount of water. The molecular formula can be expressed more clearly as MgSiO3.xH2O.T186 It is known as talc and it presents many uses in the cosmetic industry, food industry and pharmaceutical industry.L2603 Under the FDA, magnesium silicate is determined as a member of the substances generally recognized as safe (GRAS) to be used as an anticaking agent.L2605

Struktur Molekul 2D

Berat 100.387
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.[F26]
Volume Distribusi The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.[F26]
Klirens (Clearance) The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.[F26]

Absorpsi

Orally administered magnesium silicate is rapidly neutralized in the stomach and it forms magnesium chloride and silicon dioxide. From the modified portion, some of the formed magnesium is absorbed.T186 The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.F26

Metabolisme

The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.F26

Rute Eliminasi

The very low absorption of magnesium silicate makes its pharmacokinetic properties not relevant.F26

Interaksi Obat

470 Data
Succinylcholine The therapeutic efficacy of Succinylcholine can be increased when used in combination with Magnesium silicate.
Metocurine iodide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium silicate.
Gallamine triethiodide The therapeutic efficacy of Gallamine triethiodide can be increased when used in combination with Magnesium silicate.
Cisatracurium The therapeutic efficacy of Cisatracurium can be increased when used in combination with Magnesium silicate.
Rocuronium The therapeutic efficacy of Rocuronium can be increased when used in combination with Magnesium silicate.
Atracurium besylate The therapeutic efficacy of Atracurium besylate can be increased when used in combination with Magnesium silicate.
Doxacurium The therapeutic efficacy of Doxacurium can be increased when used in combination with Magnesium silicate.
Mivacurium The therapeutic efficacy of Mivacurium can be increased when used in combination with Magnesium silicate.
Decamethonium The therapeutic efficacy of Decamethonium can be increased when used in combination with Magnesium silicate.
Metocurine The therapeutic efficacy of Metocurine can be increased when used in combination with Magnesium silicate.
Pancuronium The therapeutic efficacy of Pancuronium can be increased when used in combination with Magnesium silicate.
Pipecuronium The therapeutic efficacy of Pipecuronium can be increased when used in combination with Magnesium silicate.
Vecuronium The therapeutic efficacy of Vecuronium can be increased when used in combination with Magnesium silicate.
Rapacuronium The therapeutic efficacy of Rapacuronium can be increased when used in combination with Magnesium silicate.
Pyrantel The therapeutic efficacy of Pyrantel can be increased when used in combination with Magnesium silicate.
Neosaxitoxin The therapeutic efficacy of Neosaxitoxin can be increased when used in combination with Magnesium silicate.
Atracurium The therapeutic efficacy of Atracurium can be increased when used in combination with Magnesium silicate.
Gallamine The therapeutic efficacy of Gallamine can be increased when used in combination with Magnesium silicate.
Alcuronium The therapeutic efficacy of Alcuronium can be increased when used in combination with Magnesium silicate.
Tubocurarine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium silicate.
Atazanavir Magnesium silicate can cause a decrease in the absorption of Atazanavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Bosutinib Magnesium silicate can cause a decrease in the absorption of Bosutinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefditoren The serum concentration of Cefditoren can be decreased when it is combined with Magnesium silicate.
Dabigatran etexilate Magnesium silicate can cause a decrease in the absorption of Dabigatran etexilate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dabrafenib Magnesium silicate can cause a decrease in the absorption of Dabrafenib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dasatinib Magnesium silicate can cause a decrease in the absorption of Dasatinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Delavirdine Magnesium silicate can cause a decrease in the absorption of Delavirdine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Erlotinib Magnesium silicate can cause a decrease in the absorption of Erlotinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gefitinib Magnesium silicate can cause a decrease in the absorption of Gefitinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Itraconazole Magnesium silicate can cause a decrease in the absorption of Itraconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ledipasvir Magnesium silicate can cause a decrease in the absorption of Ledipasvir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methylphenidate Magnesium silicate can cause an increase in the absorption of Methylphenidate resulting in an increased serum concentration and potentially a worsening of adverse effects.
Pazopanib Magnesium silicate can cause a decrease in the absorption of Pazopanib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Riociguat Magnesium silicate can cause a decrease in the absorption of Riociguat resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcitriol The serum concentration of Magnesium silicate can be increased when it is combined with Calcitriol.
Calcifediol The serum concentration of Magnesium silicate can be increased when it is combined with Calcifediol.
Cholecalciferol The serum concentration of Magnesium silicate can be increased when it is combined with Cholecalciferol.
Paricalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Paricalcitol.
Dihydrotachysterol The serum concentration of Magnesium silicate can be increased when it is combined with Dihydrotachysterol.
Alfacalcidol The serum concentration of Magnesium silicate can be increased when it is combined with Alfacalcidol.
Seocalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Seocalcitol.
Inecalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Inecalcitol.
Becocalcidiol The serum concentration of Magnesium silicate can be increased when it is combined with Becocalcidiol.
Eldecalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Eldecalcitol.
1alpha,24S-Dihydroxyvitamin D2 The serum concentration of Magnesium silicate can be increased when it is combined with 1alpha,24S-Dihydroxyvitamin D2.
Elocalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Elocalcitol.
Maxacalcitol The serum concentration of Magnesium silicate can be increased when it is combined with Maxacalcitol.
Doxercalciferol The serum concentration of Magnesium silicate can be increased when it is combined with Doxercalciferol.
Vitamin D The serum concentration of Magnesium silicate can be increased when it is combined with Vitamin D.
1alpha-Hydroxyvitamin D5 The serum concentration of Magnesium silicate can be increased when it is combined with 1alpha-Hydroxyvitamin D5.
Previtamin D(3) The serum concentration of Magnesium silicate can be increased when it is combined with Previtamin D(3).
Deferiprone Magnesium silicate can cause a decrease in the absorption of Deferiprone resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dolutegravir Magnesium silicate can cause a decrease in the absorption of Dolutegravir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Eltrombopag Magnesium silicate can cause a decrease in the absorption of Eltrombopag resulting in a reduced serum concentration and potentially a decrease in efficacy.
Levothyroxine Magnesium silicate can cause a decrease in the absorption of Levothyroxine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tolevamer The risk or severity of adverse effects can be increased when Tolevamer is combined with Magnesium silicate.
Bisacodyl The therapeutic efficacy of Bisacodyl can be decreased when used in combination with Magnesium silicate.
Captopril Magnesium silicate can cause a decrease in the absorption of Captopril resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefpodoxime The serum concentration of Cefpodoxime can be decreased when it is combined with Magnesium silicate.
Cefuroxime The serum concentration of Cefuroxime can be decreased when it is combined with Magnesium silicate.
Chloroquine Magnesium silicate can cause a decrease in the absorption of Chloroquine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Elvitegravir Magnesium silicate can cause a decrease in the absorption of Elvitegravir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gabapentin enacarbil The serum concentration of Gabapentin enacarbil can be decreased when it is combined with Magnesium silicate.
Hyoscyamine Magnesium silicate can cause a decrease in the absorption of Hyoscyamine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rifampin Magnesium silicate can cause a decrease in the absorption of Rifampicin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mecamylamine Magnesium silicate may decrease the excretion rate of Mecamylamine which could result in a higher serum level.
Memantine Magnesium silicate may decrease the excretion rate of Memantine which could result in a higher serum level.
Penicillamine Magnesium silicate can cause a decrease in the absorption of Penicillamine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Quinidine Magnesium silicate may decrease the excretion rate of Quinidine which could result in a higher serum level.
Quinine Magnesium silicate can cause a decrease in the absorption of Quinine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sotalol The serum concentration of Sotalol can be decreased when it is combined with Magnesium silicate.
Sulpiride The therapeutic efficacy of Sulpiride can be increased when used in combination with Magnesium silicate.
Deferasirox Magnesium silicate can cause a decrease in the absorption of Deferasirox resulting in a reduced serum concentration and potentially a decrease in efficacy.
Allopurinol The therapeutic efficacy of Allopurinol can be decreased when used in combination with Magnesium silicate.
Fexofenadine Magnesium silicate can cause a decrease in the absorption of Fexofenadine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Raltegravir Magnesium silicate can cause a decrease in the absorption of Raltegravir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Halofantrine Magnesium silicate can cause a decrease in the absorption of Halofantrine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Misoprostol The risk or severity of adverse effects can be increased when Magnesium silicate is combined with Misoprostol.
Mesalazine Magnesium silicate can cause a decrease in the absorption of Mesalazine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mycophenolic acid The serum concentration of Mycophenolic acid can be decreased when it is combined with Magnesium silicate.
Cysteamine The bioavailability of Cysteamine can be decreased when combined with Magnesium silicate.
Ketoconazole Magnesium silicate can cause a decrease in the absorption of Ketoconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Moxifloxacin Magnesium silicate can cause a decrease in the absorption of Moxifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Grepafloxacin Magnesium silicate can cause a decrease in the absorption of Grepafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Enoxacin Magnesium silicate can cause a decrease in the absorption of Enoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pefloxacin Magnesium silicate can cause a decrease in the absorption of Pefloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Trovafloxacin Magnesium silicate can cause a decrease in the absorption of Trovafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nalidixic acid Magnesium silicate can cause a decrease in the absorption of Nalidixic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rosoxacin Magnesium silicate can cause a decrease in the absorption of Rosoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cinoxacin Magnesium silicate can cause a decrease in the absorption of Cinoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lomefloxacin Magnesium silicate can cause a decrease in the absorption of Lomefloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gatifloxacin Magnesium silicate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Norfloxacin Magnesium silicate can cause a decrease in the absorption of Norfloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Levofloxacin Magnesium silicate can cause a decrease in the absorption of Levofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ofloxacin Magnesium silicate can cause a decrease in the absorption of Ofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sparfloxacin Magnesium silicate can cause a decrease in the absorption of Sparfloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Temafloxacin Magnesium silicate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fleroxacin Magnesium silicate can cause a decrease in the absorption of Fleroxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Technetium Tc-99m ciprofloxacin Magnesium silicate can cause a decrease in the absorption of Technetium Tc-99m ciprofloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Garenoxacin Magnesium silicate can cause a decrease in the absorption of Garenoxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.

Referensi & Sumber

Textbook
  • ISBN: 978-0-12-387667-6
    Rashid I., Nidal H. Daraghmeh M., Omari A., Babur Z., Chowdhry S., Leharne H., Adnan A. (2011). Profiles of drug substances and related methodology. Academic Press.
Attachment

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Formula EC
    Tablet • - • Oral • Canada • Approved

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