Alaproclate

DB13233

small molecule experimental

Deskripsi

Alaproclate was developed as one of the first selective serotonin reuptake inhibitor (SSRI) antidepressants by Astra AB (now AstraZeneca) in the 1970s. Development was discontinued due to concerns over hepatotoxicity observed in animal studies. Alaproclate has also been found to act as a non-competitive NMDA receptor antagonist although without discriminative stimulus properties similar to phencyclidine.

Struktur Molekul 2D

Berat 255.74
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1089 Data
Cyproheptadine The therapeutic efficacy of Alaproclate can be decreased when used in combination with Cyproheptadine.
Desmopressin The risk or severity of hyponatremia can be increased when Alaproclate is combined with Desmopressin.
Ioflupane I-123 Alaproclate may decrease effectiveness of Ioflupane I-123 as a diagnostic agent.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Alaproclate.
Metyrosine The risk or severity of extrapyramidal symptoms can be increased when Metyrosine is combined with Alaproclate.
Pimozide The risk or severity of QTc prolongation can be increased when Alaproclate is combined with Pimozide.
Buprenorphine Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Hydrocodone Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Magnesium sulfate The therapeutic efficacy of Alaproclate can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Orphenadrine Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Pramipexole Alaproclate may increase the sedative activities of Pramipexole.
Ropinirole Alaproclate may increase the sedative activities of Ropinirole.
Rotigotine Alaproclate may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Alaproclate.
Sodium oxybate Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Thalidomide Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Alaproclate.
Tedizolid phosphate The risk or severity of serotonin syndrome can be increased when Tedizolid phosphate is combined with Alaproclate.
Mirtazapine Alaproclate may increase the serotonergic activities of Mirtazapine.
Morphine The risk or severity of serotonin syndrome can be increased when Morphine is combined with Alaproclate.
Codeine The risk or severity of serotonin syndrome can be increased when Codeine is combined with Alaproclate.
Hydromorphone The risk or severity of serotonin syndrome can be increased when Hydromorphone is combined with Alaproclate.
Meperidine The risk or severity of serotonin syndrome can be increased when Meperidine is combined with Alaproclate.
Oxycodone The risk or severity of serotonin syndrome can be increased when Oxycodone is combined with Alaproclate.
Butorphanol The risk or severity of serotonin syndrome can be increased when Butorphanol is combined with Alaproclate.
Dextropropoxyphene The risk or severity of serotonin syndrome can be increased when Dextropropoxyphene is combined with Alaproclate.
Pentazocine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Alaproclate.
Sufentanil The risk or severity of serotonin syndrome can be increased when Sufentanil is combined with Alaproclate.
Alfentanil The risk or severity of serotonin syndrome can be increased when Alfentanil is combined with Alaproclate.
Fentanyl The risk or severity of serotonin syndrome can be increased when Fentanyl is combined with Alaproclate.
Nalbuphine The risk or severity of serotonin syndrome can be increased when Nalbuphine is combined with Alaproclate.
Levorphanol The risk or severity of serotonin syndrome can be increased when Levorphanol is combined with Alaproclate.
Remifentanil The risk or severity of serotonin syndrome can be increased when Remifentanil is combined with Alaproclate.
Diphenoxylate The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Alaproclate.
Oxymorphone The risk or severity of serotonin syndrome can be increased when Oxymorphone is combined with Alaproclate.
Dezocine The risk or severity of serotonin syndrome can be increased when Dezocine is combined with Alaproclate.
Levacetylmethadol The risk or severity of serotonin syndrome can be increased when Levacetylmethadol is combined with Alaproclate.
Methadyl acetate The risk or severity of serotonin syndrome can be increased when Methadyl acetate is combined with Alaproclate.
Dihydroetorphine The risk or severity of serotonin syndrome can be increased when Dihydroetorphine is combined with Alaproclate.
Diamorphine The risk or severity of serotonin syndrome can be increased when Diamorphine is combined with Alaproclate.
Ethylmorphine The risk or severity of serotonin syndrome can be increased when Ethylmorphine is combined with Alaproclate.
Etorphine The risk or severity of serotonin syndrome can be increased when Etorphine is combined with Alaproclate.
Dextromoramide The risk or severity of serotonin syndrome can be increased when Dextromoramide is combined with Alaproclate.
Desomorphine The risk or severity of serotonin syndrome can be increased when Desomorphine is combined with Alaproclate.
Carfentanil The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Alaproclate.
Dihydrocodeine The risk or severity of serotonin syndrome can be increased when Dihydrocodeine is combined with Alaproclate.
Alphacetylmethadol The risk or severity of serotonin syndrome can be increased when Alphacetylmethadol is combined with Alaproclate.
Dihydromorphine The risk or severity of serotonin syndrome can be increased when Dihydromorphine is combined with Alaproclate.
Ketobemidone The risk or severity of serotonin syndrome can be increased when Ketobemidone is combined with Alaproclate.
DPDPE The risk or severity of serotonin syndrome can be increased when DPDPE is combined with Alaproclate.
Lofentanil The risk or severity of serotonin syndrome can be increased when Lofentanil is combined with Alaproclate.
Opium The risk or severity of serotonin syndrome can be increased when Opium is combined with Alaproclate.
Normethadone The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Alaproclate.
Piritramide The risk or severity of serotonin syndrome can be increased when Piritramide is combined with Alaproclate.
Alphaprodine The risk or severity of serotonin syndrome can be increased when Alphaprodine is combined with Alaproclate.
Meptazinol The risk or severity of serotonin syndrome can be increased when Meptazinol is combined with Alaproclate.
Phenoperidine The risk or severity of serotonin syndrome can be increased when Phenoperidine is combined with Alaproclate.
Phenazocine The risk or severity of serotonin syndrome can be increased when Phenazocine is combined with Alaproclate.
Tilidine The risk or severity of serotonin syndrome can be increased when Tilidine is combined with Alaproclate.
Carfentanil, C-11 The risk or severity of serotonin syndrome can be increased when Carfentanil, C-11 is combined with Alaproclate.
Naltrexone The risk or severity of serotonin syndrome can be increased when Naltrexone is combined with Alaproclate.
Bezitramide The risk or severity of serotonin syndrome can be increased when Bezitramide is combined with Alaproclate.
Eluxadoline The risk or severity of serotonin syndrome can be increased when Eluxadoline is combined with Alaproclate.
Nicomorphine The risk or severity of serotonin syndrome can be increased when Nicomorphine is combined with Alaproclate.
Benzhydrocodone The risk or severity of serotonin syndrome can be increased when Benzhydrocodone is combined with Alaproclate.
Naloxegol The risk or severity of serotonin syndrome can be increased when Naloxegol is combined with Alaproclate.
Iobenguane Alaproclate may decrease effectiveness of Iobenguane as a diagnostic agent.
Methyclothiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Methyclothiazide.
Chlorthalidone The risk or severity of hyponatremia can be increased when Alaproclate is combined with Chlorthalidone.
Bendroflumethiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Bendroflumethiazide.
Metolazone The risk or severity of hyponatremia can be increased when Alaproclate is combined with Metolazone.
Benzthiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Benzthiazide.
Hydroflumethiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Hydroflumethiazide.
Indapamide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Indapamide.
Chlorothiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Chlorothiazide.
Hydrochlorothiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Hydrochlorothiazide.
Trichlormethiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Trichlormethiazide.
Polythiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Polythiazide.
Quinethazone The risk or severity of hyponatremia can be increased when Alaproclate is combined with Quinethazone.
Cyclopenthiazide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Cyclopenthiazide.
Epitizide The risk or severity of hyponatremia can be increased when Alaproclate is combined with Epitizide.
Ethanol Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Alaproclate may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Botulinum toxin type B is combined with Alaproclate.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Botulinum toxin type A is combined with Alaproclate.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Alaproclate.
Ethchlorvynol The risk or severity of adverse effects can be increased when Ethchlorvynol is combined with Alaproclate.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 7996440
    Wilkinson A, Courtney M, Westlind-Danielsson A, Hallnemo G, Akerman KE: Alaproclate acts as a potent, reversible and noncompetitive antagonist of the NMDA receptor coupled ion flow. J Pharmacol Exp Ther. 1994 Dec;271(3):1314-9.
  • PMID: 12851738
    Nicholson KL, Balster RL: Evaluation of the phencyclidine-like discriminative stimulus effects of novel NMDA channel blockers in rats. Psychopharmacology (Berl). 2003 Nov;170(2):215-24. Epub 2003 Jul 8.

Contoh Produk & Brand

Produk: 0 • International brands: 0
Belum ada data produk/brand untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field produk/brand.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul