Abexinostat

DB12565

small molecule investigational

Deskripsi

Abexinostat has been used in trials studying the treatment of Sarcoma, Lymphoma, Leukemia, Lymphocytic, and Hodgkin Disease, among others. It is a novel, broad-spectrum hydroxamic acid-based inhibitor of histone deacetylase (HDAC) with potential antineoplastic activity.

Struktur Molekul 2D

Berat 397.431
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

404 Data
Ivabradine Ivabradine may increase the QTc-prolonging activities of Abexinostat.
Vorinostat The risk or severity of gastrointestinal bleeding and thrombocytopenia can be increased when Abexinostat is combined with Vorinostat.
Dofetilide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Dofetilide.
Citalopram The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Citalopram.
Anagrelide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Anagrelide.
Disopyramide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Disopyramide.
Clemastine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Clemastine.
Ibutilide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Ibutilide.
Valproic acid The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Valproic acid.
Terfenadine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Terfenadine.
Grepafloxacin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Grepafloxacin.
Quinine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Quinine.
Sotalol The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Sotalol.
Erlotinib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Erlotinib.
Toremifene The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Toremifene.
Cisapride The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Cisapride.
Imatinib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Imatinib.
Astemizole The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Astemizole.
Thioridazine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Thioridazine.
Trovafloxacin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Trovafloxacin.
Mifepristone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Mifepristone.
Cocaine The risk or severity of methemoglobinemia can be increased when Abexinostat is combined with Cocaine.
Quinidine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Quinidine.
Procainamide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Procainamide.
Pimozide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Pimozide.
Amiodarone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Amiodarone.
Arsenic trioxide The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Arsenic trioxide.
Escitalopram The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Escitalopram.
Domperidone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Domperidone.
Sparfloxacin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Sparfloxacin.
Halofantrine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Halofantrine.
Bepridil The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Bepridil.
Paliperidone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Paliperidone.
Lithium cation The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Lithium cation.
Temafloxacin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Temafloxacin.
Zuclopenthixol The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Zuclopenthixol.
Tetrabenazine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Tetrabenazine.
Dronedarone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Dronedarone.
Nilotinib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Nilotinib.
Iloperidone The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Iloperidone.
Vandetanib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Vandetanib.
Romidepsin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Romidepsin.
Asenapine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Asenapine.
Artemether The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Artemether.
Lumefantrine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Lumefantrine.
Vemurafenib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Vemurafenib.
Eliglustat The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Eliglustat.
Ribociclib The risk or severity of QTc prolongation can be increased when Ribociclib is combined with Abexinostat.
Glasdegib The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Glasdegib.
Deutetrabenazine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Deutetrabenazine.
Macimorelin The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Macimorelin.
Terodiline The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Terodiline.
Leuprolide The risk or severity of QTc prolongation can be increased when Leuprolide is combined with Abexinostat.
Goserelin The risk or severity of QTc prolongation can be increased when Goserelin is combined with Abexinostat.
Erythromycin The risk or severity of QTc prolongation can be increased when Erythromycin is combined with Abexinostat.
Azithromycin The risk or severity of QTc prolongation can be increased when Azithromycin is combined with Abexinostat.
Moxifloxacin The risk or severity of QTc prolongation can be increased when Moxifloxacin is combined with Abexinostat.
Ranolazine The risk or severity of QTc prolongation can be increased when Ranolazine is combined with Abexinostat.
Sulfisoxazole The risk or severity of QTc prolongation can be increased when Sulfisoxazole is combined with Abexinostat.
Amitriptyline The risk or severity of QTc prolongation can be increased when Amitriptyline is combined with Abexinostat.
Methadone The risk or severity of QTc prolongation can be increased when Methadone is combined with Abexinostat.
Diltiazem The risk or severity of QTc prolongation can be increased when Diltiazem is combined with Abexinostat.
Clozapine The risk or severity of QTc prolongation can be increased when Abexinostat is combined with Clozapine.
Sulpiride The risk or severity of QTc prolongation can be increased when Sulpiride is combined with Abexinostat.
Nimodipine The risk or severity of QTc prolongation can be increased when Nimodipine is combined with Abexinostat.
Promazine The risk or severity of QTc prolongation can be increased when Promazine is combined with Abexinostat.
Prochlorperazine The risk or severity of QTc prolongation can be increased when Prochlorperazine is combined with Abexinostat.
Droperidol The risk or severity of QTc prolongation can be increased when Droperidol is combined with Abexinostat.
Imipramine The risk or severity of QTc prolongation can be increased when Imipramine is combined with Abexinostat.
Chlorpromazine The risk or severity of QTc prolongation can be increased when Chlorpromazine is combined with Abexinostat.
Oxaliplatin The risk or severity of QTc prolongation can be increased when Oxaliplatin is combined with Abexinostat.
Ciprofloxacin The risk or severity of QTc prolongation can be increased when Ciprofloxacin is combined with Abexinostat.
Fluorouracil The risk or severity of QTc prolongation can be increased when Fluorouracil is combined with Abexinostat.
Perflutren The risk or severity of QTc prolongation can be increased when Perflutren is combined with Abexinostat.
Cinnarizine The risk or severity of QTc prolongation can be increased when Cinnarizine is combined with Abexinostat.
Atropine The risk or severity of QTc prolongation can be increased when Atropine is combined with Abexinostat.
Chloroquine The risk or severity of QTc prolongation can be increased when Chloroquine is combined with Abexinostat.
Efavirenz The risk or severity of QTc prolongation can be increased when Efavirenz is combined with Abexinostat.
Adenosine The risk or severity of QTc prolongation can be increased when Adenosine is combined with Abexinostat.
Pentamidine The risk or severity of QTc prolongation can be increased when Pentamidine is combined with Abexinostat.
Gadobenic acid The risk or severity of QTc prolongation can be increased when Gadobenic acid is combined with Abexinostat.
Carbinoxamine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Abexinostat.
Dolasetron The risk or severity of QTc prolongation can be increased when Dolasetron is combined with Abexinostat.
Roxithromycin The risk or severity of QTc prolongation can be increased when Roxithromycin is combined with Abexinostat.
Nalidixic acid The risk or severity of QTc prolongation can be increased when Nalidixic acid is combined with Abexinostat.
Cinoxacin The risk or severity of QTc prolongation can be increased when Cinoxacin is combined with Abexinostat.
Loperamide The risk or severity of QTc prolongation can be increased when Loperamide is combined with Abexinostat.
Granisetron The risk or severity of QTc prolongation can be increased when Granisetron is combined with Abexinostat.
Ondansetron The risk or severity of QTc prolongation can be increased when Ondansetron is combined with Abexinostat.
Levosimendan The risk or severity of QTc prolongation can be increased when Levosimendan is combined with Abexinostat.
Mesoridazine The risk or severity of QTc prolongation can be increased when Mesoridazine is combined with Abexinostat.
Desloratadine The risk or severity of QTc prolongation can be increased when Desloratadine is combined with Abexinostat.
Telithromycin The risk or severity of QTc prolongation can be increased when Telithromycin is combined with Abexinostat.
Lomefloxacin The risk or severity of QTc prolongation can be increased when Lomefloxacin is combined with Abexinostat.
Dimenhydrinate The risk or severity of QTc prolongation can be increased when Dimenhydrinate is combined with Abexinostat.
Primaquine The risk or severity of QTc prolongation can be increased when Primaquine is combined with Abexinostat.
Papaverine The risk or severity of QTc prolongation can be increased when Papaverine is combined with Abexinostat.
Chlorpheniramine The risk or severity of QTc prolongation can be increased when Chlorpheniramine is combined with Abexinostat.
Nifedipine The risk or severity of QTc prolongation can be increased when Nifedipine is combined with Abexinostat.
Levofloxacin The risk or severity of QTc prolongation can be increased when Levofloxacin is combined with Abexinostat.

Target Protein

Histone deacetylase 1 HDAC1
Histone deacetylase HDAC1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16731764
    Buggy JJ, Cao ZA, Bass KE, Verner E, Balasubramanian S, Liu L, Schultz BE, Young PR, Dalrymple SA: CRA-024781: a novel synthetic inhibitor of histone deacetylase enzymes with antitumor activity in vitro and in vivo. Mol Cancer Ther. 2006 May;5(5):1309-17.

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Sekuens Gen/Protein (FASTA)

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