Navitoclax

DB12340

small molecule investigational

Deskripsi

Navitoclax has been used in trials studying the treatment and basic science of Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies, among others.

Navitoclax is an orally bioavailable small molecule inhibitor of Bcl-2 family proteins. It is a substance being studied in the treatment of lymphomas and other types of cancer. It blocks some of the enzymes that keep cancer cells from dying.

Struktur Molekul 2D

Berat 974.613
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

39 Data
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Navitoclax.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Navitoclax.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Navitoclax.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Navitoclax.
Lidocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Navitoclax.
Ambroxol The risk or severity of methemoglobinemia can be increased when Navitoclax is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Navitoclax is combined with Etrasimod.

Target Protein

Bcl-2-like protein 1 BCL2L1
G1/S-specific cyclin-D1 CCND1
Apoptosis regulator Bcl-2 BCL2
Bcl-2-like protein 2 BCL2L2
Bcl2-associated agonist of cell death BAD

Referensi & Sumber

Artikel (PubMed)
  • PMID: 18085673
    Lock R, Carol H, Houghton PJ, Morton CL, Kolb EA, Gorlick R, Reynolds CP, Maris JM, Keir ST, Wu J, Smith MA: Initial testing (stage 1) of the BH3 mimetic ABT-263 by the pediatric preclinical testing program. Pediatr Blood Cancer. 2008 Jun;50(6):1181-9.

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Sekuens Gen/Protein (FASTA)

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