Fasinumab

DB12157

biotech investigational

Deskripsi

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic painA241045 and has demonstrated significantly greater pain relief and functional improvement as compared to standard therapy (i.e. NSAIDs and/or opioids) in this patient population.A241165

NGF was first discovered in the 1950sA241180 and was the first neurotrophic factor to be identified and biochemically characterized.A241190 It has since been recognized for its role in nociceptive signaling transduction and has thus become an attractive target in the treatment of chronic pain conditions.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

373 Data
Diethylstilbestrol Diethylstilbestrol may increase the thrombogenic activities of Fasinumab.
Chlorotrianisene Chlorotrianisene may increase the thrombogenic activities of Fasinumab.
Conjugated estrogens Conjugated estrogens may increase the thrombogenic activities of Fasinumab.
Estrone Estrone may increase the thrombogenic activities of Fasinumab.
Estradiol Estradiol may increase the thrombogenic activities of Fasinumab.
Dienestrol Dienestrol may increase the thrombogenic activities of Fasinumab.
Ethinylestradiol Ethinylestradiol may increase the thrombogenic activities of Fasinumab.
Mestranol Mestranol may increase the thrombogenic activities of Fasinumab.
Estriol Estriol may increase the thrombogenic activities of Fasinumab.
Estrone sulfate Estrone sulfate may increase the thrombogenic activities of Fasinumab.
Quinestrol Quinestrol may increase the thrombogenic activities of Fasinumab.
Hexestrol Hexestrol may increase the thrombogenic activities of Fasinumab.
Tibolone Tibolone may increase the thrombogenic activities of Fasinumab.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may increase the thrombogenic activities of Fasinumab.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may increase the thrombogenic activities of Fasinumab.
Polyestradiol phosphate Polyestradiol phosphate may increase the thrombogenic activities of Fasinumab.
Esterified estrogens Esterified estrogens may increase the thrombogenic activities of Fasinumab.
Zeranol Zeranol may increase the thrombogenic activities of Fasinumab.
Equol Equol may increase the thrombogenic activities of Fasinumab.
Promestriene Promestriene may increase the thrombogenic activities of Fasinumab.
Methallenestril Methallenestril may increase the thrombogenic activities of Fasinumab.
Epimestrol Epimestrol may increase the thrombogenic activities of Fasinumab.
Moxestrol Moxestrol may increase the thrombogenic activities of Fasinumab.
Estradiol acetate Estradiol acetate may increase the thrombogenic activities of Fasinumab.
Estradiol benzoate Estradiol benzoate may increase the thrombogenic activities of Fasinumab.
Estradiol cypionate Estradiol cypionate may increase the thrombogenic activities of Fasinumab.
Estradiol valerate Estradiol valerate may increase the thrombogenic activities of Fasinumab.
Biochanin A Biochanin A may increase the thrombogenic activities of Fasinumab.
Formononetin Formononetin may increase the thrombogenic activities of Fasinumab.
Estetrol Estetrol may increase the thrombogenic activities of Fasinumab.
Cetuximab The risk or severity of adverse effects can be increased when Cetuximab is combined with Fasinumab.
Human immunoglobulin G The risk or severity of adverse effects can be increased when Human immunoglobulin G is combined with Fasinumab.
Omalizumab The risk or severity of adverse effects can be increased when Omalizumab is combined with Fasinumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Fasinumab.
Abciximab The risk or severity of adverse effects can be increased when Abciximab is combined with Fasinumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Fasinumab.
Indium In-111 satumomab pendetide The risk or severity of adverse effects can be increased when Indium In-111 satumomab pendetide is combined with Fasinumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Fasinumab.
Trastuzumab The risk or severity of adverse effects can be increased when Trastuzumab is combined with Fasinumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Fasinumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Fasinumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Fasinumab.
Digoxin Immune Fab (Ovine) The risk or severity of adverse effects can be increased when Digoxin Immune Fab (Ovine) is combined with Fasinumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Fasinumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Fasinumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Fasinumab.
Capromab pendetide The risk or severity of adverse effects can be increased when Capromab pendetide is combined with Fasinumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Fasinumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Fasinumab.
Natalizumab The risk or severity of adverse effects can be increased when Natalizumab is combined with Fasinumab.
Palivizumab The risk or severity of adverse effects can be increased when Palivizumab is combined with Fasinumab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Fasinumab.
Bevacizumab The risk or severity of adverse effects can be increased when Bevacizumab is combined with Fasinumab.
Technetium Tc-99m arcitumomab The risk or severity of adverse effects can be increased when Technetium Tc-99m arcitumomab is combined with Fasinumab.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Fasinumab.
Panitumumab The risk or severity of adverse effects can be increased when Panitumumab is combined with Fasinumab.
Ranibizumab The risk or severity of adverse effects can be increased when Ranibizumab is combined with Fasinumab.
Galiximab The risk or severity of adverse effects can be increased when Galiximab is combined with Fasinumab.
Pexelizumab The risk or severity of adverse effects can be increased when Pexelizumab is combined with Fasinumab.
Afelimomab The risk or severity of adverse effects can be increased when Afelimomab is combined with Fasinumab.
Epratuzumab The risk or severity of adverse effects can be increased when Epratuzumab is combined with Fasinumab.
Bectumomab The risk or severity of adverse effects can be increased when Bectumomab is combined with Fasinumab.
Oregovomab The risk or severity of adverse effects can be increased when Oregovomab is combined with Fasinumab.
IGN311 The risk or severity of adverse effects can be increased when IGN311 is combined with Fasinumab.
Adecatumumab The risk or severity of adverse effects can be increased when Adecatumumab is combined with Fasinumab.
Labetuzumab The risk or severity of adverse effects can be increased when Labetuzumab is combined with Fasinumab.
Matuzumab The risk or severity of adverse effects can be increased when Matuzumab is combined with Fasinumab.
Fontolizumab The risk or severity of adverse effects can be increased when Fontolizumab is combined with Fasinumab.
Bavituximab The risk or severity of adverse effects can be increased when Bavituximab is combined with Fasinumab.
CR002 The risk or severity of adverse effects can be increased when CR002 is combined with Fasinumab.
Rozrolimupab The risk or severity of adverse effects can be increased when Rozrolimupab is combined with Fasinumab.
Girentuximab The risk or severity of adverse effects can be increased when Girentuximab is combined with Fasinumab.
Obiltoxaximab The risk or severity of adverse effects can be increased when Obiltoxaximab is combined with Fasinumab.
XTL-001 The risk or severity of adverse effects can be increased when XTL-001 is combined with Fasinumab.
NAV 1800 The risk or severity of adverse effects can be increased when NAV 1800 is combined with Fasinumab.
Briakinumab The risk or severity of adverse effects can be increased when Briakinumab is combined with Fasinumab.
Otelixizumab The risk or severity of adverse effects can be increased when Otelixizumab is combined with Fasinumab.
AMG 108 The risk or severity of adverse effects can be increased when AMG 108 is combined with Fasinumab.
Iratumumab The risk or severity of adverse effects can be increased when Iratumumab is combined with Fasinumab.
Enokizumab The risk or severity of adverse effects can be increased when Enokizumab is combined with Fasinumab.
Ramucirumab The risk or severity of adverse effects can be increased when Ramucirumab is combined with Fasinumab.
Farletuzumab The risk or severity of adverse effects can be increased when Farletuzumab is combined with Fasinumab.
Veltuzumab The risk or severity of adverse effects can be increased when Veltuzumab is combined with Fasinumab.
Ustekinumab The risk or severity of adverse effects can be increased when Ustekinumab is combined with Fasinumab.
Trastuzumab emtansine The risk or severity of adverse effects can be increased when Trastuzumab emtansine is combined with Fasinumab.
PRO-542 The risk or severity of adverse effects can be increased when PRO-542 is combined with Fasinumab.
TNX-901 The risk or severity of adverse effects can be increased when TNX-901 is combined with Fasinumab.
Inotuzumab ozogamicin The risk or severity of adverse effects can be increased when Inotuzumab ozogamicin is combined with Fasinumab.
RI 624 The risk or severity of adverse effects can be increased when RI 624 is combined with Fasinumab.
Stamulumab The risk or severity of adverse effects can be increased when MYO-029 is combined with Fasinumab.
CT-011 The risk or severity of adverse effects can be increased when CT-011 is combined with Fasinumab.
Leronlimab The risk or severity of adverse effects can be increased when Leronlimab is combined with Fasinumab.
Glembatumumab vedotin The risk or severity of adverse effects can be increased when Glembatumumab vedotin is combined with Fasinumab.
Olaratumab The risk or severity of adverse effects can be increased when Olaratumab is combined with Fasinumab.
IPH 2101 The risk or severity of adverse effects can be increased when IPH 2101 is combined with Fasinumab.
TB-402 The risk or severity of adverse effects can be increased when TB-402 is combined with Fasinumab.
Caplacizumab The risk or severity of adverse effects can be increased when Caplacizumab is combined with Fasinumab.
IMC-1C11 The risk or severity of adverse effects can be increased when IMC-1C11 is combined with Fasinumab.
Eldelumab The risk or severity of adverse effects can be increased when Eldelumab is combined with Fasinumab.
Lumiliximab The risk or severity of adverse effects can be increased when Lumiliximab is combined with Fasinumab.

Target Protein

Beta-nerve growth factor NGF

Referensi & Sumber

Artikel (PubMed)
  • PMID: 33459118
    Kaplon H, Reichert JM: Antibodies to watch in 2021. MAbs. 2021 Jan-Dec;13(1):1860476. doi: 10.1080/19420862.2020.1860476.
  • PMID: 33293475
    Cao Z, Zhou J, Long Z, Li Y, Sun J, Luo Y, Wang W: Targeting nerve growth factor, a new option for treatment of osteoarthritis: a network meta-analysis of comparative efficacy and safety with traditional drugs. Aging (Albany NY). 2020 Dec 3;13(1):1051-1070. doi: 10.18632/aging.202232. Epub 2020 Dec 3.
  • PMID: 34234542
    Bimonte S, Cascella M, Forte CA, Esposito G, Cuomo A: The Role of Anti-Nerve Growth Factor Monoclonal Antibodies in the Control of Chronic Cancer and Non-Cancer Pain. J Pain Res. 2021 Jun 28;14:1959-1967. doi: 10.2147/JPR.S302004. eCollection 2021.
  • PMID: 23028238
    Kumar V, Mahal BA: NGF - the TrkA to successful pain treatment. J Pain Res. 2012;5:279-87. doi: 10.2147/JPR.S33408. Epub 2012 Aug 17.

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