Triptolide

DB12025

small molecule investigational

Deskripsi

Triptolide has been used in trials studying the treatment of HIV, Crohn's Disease, Intestinal Diseases, Gastrointestinal Diseases, and Digestive System Diseases, among others.

Struktur Molekul 2D

Berat 360.406
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

390 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Triptolide.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Triptolide.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Triptolide.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Triptolide.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Triptolide.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Triptolide.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Triptolide.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Triptolide.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Triptolide.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Triptolide.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Triptolide.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Triptolide.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Triptolide.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Triptolide.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Triptolide.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Triptolide.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Triptolide.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Triptolide.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Triptolide.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Triptolide.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Triptolide.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Triptolide.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Triptolide.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Triptolide.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Triptolide.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Triptolide.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Triptolide.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Triptolide.
Bortezomib The risk or severity of adverse effects can be increased when Bortezomib is combined with Triptolide.
Cladribine Triptolide may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Triptolide.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Triptolide.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Triptolide.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Triptolide.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Triptolide.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Triptolide.
Bexarotene The risk or severity of adverse effects can be increased when Bexarotene is combined with Triptolide.
Vindesine The risk or severity of adverse effects can be increased when Vindesine is combined with Triptolide.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Triptolide.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Triptolide.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Triptolide.
Vinorelbine The risk or severity of adverse effects can be increased when Vinorelbine is combined with Triptolide.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Triptolide.
Sorafenib The risk or severity of adverse effects can be increased when Sorafenib is combined with Triptolide.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Triptolide.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Triptolide.
Teniposide The risk or severity of adverse effects can be increased when Teniposide is combined with Triptolide.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Triptolide.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Triptolide.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Triptolide.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Triptolide.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Triptolide.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Triptolide.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Triptolide.
Cyclophosphamide The risk or severity of adverse effects can be increased when Cyclophosphamide is combined with Triptolide.
Vincristine The risk or severity of adverse effects can be increased when Vincristine is combined with Triptolide.
Fluorouracil The risk or severity of adverse effects can be increased when Fluorouracil is combined with Triptolide.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Triptolide.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Triptolide.
Methotrexate The risk or severity of adverse effects can be increased when Methotrexate is combined with Triptolide.
Vinblastine The risk or severity of adverse effects can be increased when Vinblastine is combined with Triptolide.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Triptolide.
Imatinib The risk or severity of adverse effects can be increased when Imatinib is combined with Triptolide.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Triptolide.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Triptolide.
Daunorubicin The risk or severity of adverse effects can be increased when Daunorubicin is combined with Triptolide.
Irinotecan The risk or severity of adverse effects can be increased when Irinotecan is combined with Triptolide.
Methimazole The risk or severity of adverse effects can be increased when Methimazole is combined with Triptolide.
Etoposide The risk or severity of adverse effects can be increased when Etoposide is combined with Triptolide.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Triptolide.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Triptolide.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Triptolide.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Triptolide.
Sirolimus The risk or severity of adverse effects can be increased when Sirolimus is combined with Triptolide.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Triptolide.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Triptolide.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Triptolide.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Triptolide.
Cytarabine The risk or severity of adverse effects can be increased when Cytarabine is combined with Triptolide.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Triptolide.
Doxorubicin The risk or severity of adverse effects can be increased when Doxorubicin is combined with Triptolide.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Triptolide.
Busulfan The risk or severity of adverse effects can be increased when Busulfan is combined with Triptolide.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Triptolide.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Triptolide.
Melphalan The risk or severity of adverse effects can be increased when Melphalan is combined with Triptolide.
Fludarabine The risk or severity of adverse effects can be increased when Fludarabine is combined with Triptolide.
Flucytosine The risk or severity of adverse effects can be increased when Flucytosine is combined with Triptolide.
Capecitabine The risk or severity of adverse effects can be increased when Capecitabine is combined with Triptolide.
Procarbazine The risk or severity of adverse effects can be increased when Procarbazine is combined with Triptolide.
Arsenic trioxide The risk or severity of adverse effects can be increased when Arsenic trioxide is combined with Triptolide.
Idarubicin The risk or severity of adverse effects can be increased when Idarubicin is combined with Triptolide.
Ifosfamide The risk or severity of adverse effects can be increased when Ifosfamide is combined with Triptolide.
Estramustine The risk or severity of adverse effects can be increased when Estramustine is combined with Triptolide.
Mitoxantrone The risk or severity of adverse effects can be increased when Mitoxantrone is combined with Triptolide.
Lomustine The risk or severity of adverse effects can be increased when Lomustine is combined with Triptolide.
Paclitaxel The risk or severity of adverse effects can be increased when Paclitaxel is combined with Triptolide.
Docetaxel The risk or severity of adverse effects can be increased when Docetaxel is combined with Triptolide.
Dasatinib The risk or severity of adverse effects can be increased when Dasatinib is combined with Triptolide.
Eculizumab The risk or severity of adverse effects can be increased when Eculizumab is combined with Triptolide.

Target Protein

Transcription factor RelB RELB
Nuclear factor NF-kappa-B p105 subunit NFKB1
Nuclear factor NF-kappa-B p100 subunit NFKB2
Transcription factor p65 RELA
Proto-oncogene c-Rel REL

Referensi & Sumber

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