Brodalumab

DB11776

biotech approved investigational

Deskripsi

Brodalumab has been used in trials studying the treatment of Asthma, Psoriasis, Crohn's Disease, Psoriatic Arthritis, and Rheumatoid Arthritis. Brodalumab was FDA approved in February, 2017 as Siliq for the treatment of moderate-to-severe plaque psoriasis.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi 4.62 L.
Klirens (Clearance) 0.223 L/day.

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

670 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Brodalumab.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Brodalumab.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Brodalumab.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Brodalumab.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Brodalumab.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Brodalumab.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Brodalumab.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Brodalumab.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Brodalumab.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Brodalumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Brodalumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Brodalumab.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Brodalumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Brodalumab.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Brodalumab.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Brodalumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Brodalumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Brodalumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Brodalumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Brodalumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Brodalumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Brodalumab.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Brodalumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Brodalumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Brodalumab.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Brodalumab.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Brodalumab.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Brodalumab.
Flunisolide The risk or severity of adverse effects can be increased when Flunisolide is combined with Brodalumab.
Bortezomib The risk or severity of adverse effects can be increased when Bortezomib is combined with Brodalumab.
Cladribine Brodalumab may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Brodalumab.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Brodalumab.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Brodalumab.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Brodalumab.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Brodalumab.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Brodalumab.
Bexarotene The risk or severity of adverse effects can be increased when Bexarotene is combined with Brodalumab.
Vindesine The risk or severity of adverse effects can be increased when Vindesine is combined with Brodalumab.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Brodalumab.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Brodalumab.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Brodalumab.
Vinorelbine The risk or severity of adverse effects can be increased when Vinorelbine is combined with Brodalumab.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Brodalumab.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Beclomethasone dipropionate is combined with Brodalumab.
Sorafenib The risk or severity of adverse effects can be increased when Sorafenib is combined with Brodalumab.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Brodalumab.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Brodalumab.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Brodalumab.
Betamethasone The risk or severity of adverse effects can be increased when Betamethasone is combined with Brodalumab.
Teniposide The risk or severity of adverse effects can be increased when Teniposide is combined with Brodalumab.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Brodalumab.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Brodalumab.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Brodalumab.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Brodalumab.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Brodalumab.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Brodalumab.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Brodalumab.
Cyclophosphamide The risk or severity of adverse effects can be increased when Cyclophosphamide is combined with Brodalumab.
Vincristine The risk or severity of adverse effects can be increased when Vincristine is combined with Brodalumab.
Fluorouracil The risk or severity of adverse effects can be increased when Fluorouracil is combined with Brodalumab.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Brodalumab.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Brodalumab.
Methotrexate The risk or severity of adverse effects can be increased when Methotrexate is combined with Brodalumab.
Carbamazepine The risk or severity of adverse effects can be increased when Carbamazepine is combined with Brodalumab.
Vinblastine The risk or severity of adverse effects can be increased when Vinblastine is combined with Brodalumab.
Fluticasone propionate The risk or severity of adverse effects can be increased when Fluticasone propionate is combined with Brodalumab.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Fluocinolone acetonide is combined with Brodalumab.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Brodalumab.
Imatinib The risk or severity of adverse effects can be increased when Imatinib is combined with Brodalumab.
Triamcinolone The risk or severity of adverse effects can be increased when Triamcinolone is combined with Brodalumab.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Brodalumab.
Prednisone The risk or severity of adverse effects can be increased when Prednisone is combined with Brodalumab.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Brodalumab.
Fludrocortisone The risk or severity of adverse effects can be increased when Fludrocortisone is combined with Brodalumab.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mycophenolate mofetil is combined with Brodalumab.
Daunorubicin The risk or severity of adverse effects can be increased when Daunorubicin is combined with Brodalumab.
Irinotecan The risk or severity of adverse effects can be increased when Irinotecan is combined with Brodalumab.
Methimazole The risk or severity of adverse effects can be increased when Methimazole is combined with Brodalumab.
Etoposide The risk or severity of adverse effects can be increased when Etoposide is combined with Brodalumab.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Brodalumab.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Brodalumab.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Brodalumab.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Brodalumab.
Prednisolone The risk or severity of adverse effects can be increased when Prednisolone is combined with Brodalumab.
Sirolimus The risk or severity of adverse effects can be increased when Sirolimus is combined with Brodalumab.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Brodalumab.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Brodalumab.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Brodalumab.
Methylprednisolone The risk or severity of adverse effects can be increased when Methylprednisolone is combined with Brodalumab.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Brodalumab.
Cytarabine The risk or severity of adverse effects can be increased when Cytarabine is combined with Brodalumab.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Brodalumab.
Doxorubicin The risk or severity of adverse effects can be increased when Doxorubicin is combined with Brodalumab.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Brodalumab.
Busulfan The risk or severity of adverse effects can be increased when Busulfan is combined with Brodalumab.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Brodalumab.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Brodalumab.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Brodalumab.
Thalidomide The risk or severity of adverse effects can be increased when Thalidomide is combined with Brodalumab.

Target Protein

Interleukin-17 receptor A IL17RA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 27577550
    Greig SL: Brodalumab: First Global Approval. Drugs. 2016 Sep;76(14):1403-12. doi: 10.1007/s40265-016-0634-8.
  • PMID: 24846347
    Endres CJ, Salinger DH, Kock K, Gastonguay MR, Martin DA, Klekotka P, Nirula A, Gibbs MA: Population pharmacokinetics of brodalumab in healthy adults and adults with psoriasis from single and multiple dose studies. J Clin Pharmacol. 2014 Nov;54(11):1230-8. doi: 10.1002/jcph.334. Epub 2014 May 27.

Contoh Produk & Brand

Produk: 4 • International brands: 0
Produk
  • Kyntheum
    Injection, solution • 210 mg • Subcutaneous • EU • Approved
  • Kyntheum
    Injection, solution • 210 mg • Subcutaneous • EU • Approved
  • Siliq
    Injection • 210 mg/1 • Subcutaneous • US • Approved
  • Siliq
    Solution • 210 mg / 1.5 mL • Subcutaneous • Canada • Approved

Sekuens Gen/Protein (FASTA)

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