Peringatan Keamanan

In an acute oral toxicity study in mouse, LD50 was >2000 mg/kg MSDS. Single oral doses of curcumin at 1-5 g/kg bw induced no toxic effects in rats F114. There has been no cases of overdose reported F114.

Curcumin

DB11672

small molecule approved investigational

Deskripsi

Curcumin, also known as diferuloylmethane, is an active component in the golden spice turmeric (Curcuma longa) and in Curcuma xanthorrhiza oil. It is a highly pleiotropic molecule that exhibits antibacterial, anti-inflammatory, hypoglycemic, antioxidant, wound-healing, and antimicrobial activities A33166. Due to these properties, curcumin has been investigated for the treatment and supportive care of clinical conditions including proteinuria, breast cancer, multiple myeloma, depression, and Non Small Cell Lung Cancer (NSCLC). Despite proven efficacy against numerous experimental models, poor bioavailability due to poor absorption, rapid metabolism, and rapid systemic elimination have been shown to limit the therapeutic efficacy of curcumin A33166. Curcumin is under investigation for the treatment and supportive care of various clinical conditions including mucositis, rectal cancer, prostate cancer, chronic schizophrenia, and Mild Cognitive Impairment (MCI) A33166.

Struktur Molekul 2D

Berat 368.3799
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) No pharmacokinetic data available.
Volume Distribusi Following oral administration of radio-labelled curcumin to rats, radioactivity was detected in the liver and kidneys [F114].
Klirens (Clearance) No pharmacokinetic data available.

Absorpsi

Curcumin displays poor absorption into the gastrointestinal tract. In a rat study, oral administration of a single dose of 2 g of curcumin resulted in a plasma concentration of less than 5 ?g/mL, indicating poor absorption from the gut F114.

Metabolisme

Initially, curcumin undergoes rapid intestinal metabolism to form curcumin glucuronide and curcumin sulfate via O-conjugation. Other metabolites formed include tetrahydrocurcumin, hexahydrocurcumin, and hexahydrocurcuminol via reduction F114. Curcumin may also undergo intensive second metabolism in the liver where the major metabolites were glucuronides of tetrahydrocurcumin and hexahydrocurcumin, with dihydroferulic acid and traces of ferulic acid as further metabolites F114. Hepatic metabolites are expected to be excreted in the bile F114. Certain curcumin metabolites, such as tetrahydrocurcumin, retain anti-inflammatory and antioxidant properties F114.

Rute Eliminasi

Following oral administration of curcumin to rats at a dose of 1 g/kg bw, about 75% of dose was excreted in the faeces and only traces of the compound was detected in the urine F114. When a single 400 mg dose of curcumin was administered orally to rats, about 60% was absorbed and 40% was excreted unchanged in the faeces over an period of 5 days F114. Intraperitoneal administration resulted in fecal excretion of 73% and biliary excretion of 11% F114.

Interaksi Obat

1022 Data
Voxelotor The serum concentration of Voxelotor can be increased when it is combined with Curcumin.
Levamlodipine The serum concentration of Levamlodipine can be increased when it is combined with Curcumin.
Haloperidol The serum concentration of Haloperidol can be increased when it is combined with Curcumin.
Oliceridine The serum concentration of Oliceridine can be increased when it is combined with Curcumin.
Relugolix The serum concentration of Relugolix can be increased when it is combined with Curcumin.
Tepotinib The serum concentration of Tepotinib can be increased when it is combined with Curcumin.
Pexidartinib The metabolism of Pexidartinib can be decreased when combined with Curcumin.
Pretomanid The metabolism of Pretomanid can be decreased when combined with Curcumin.
Lefamulin The serum concentration of Lefamulin can be increased when it is combined with Curcumin.
Colchicine The serum concentration of Colchicine can be increased when it is combined with Curcumin.
Dronedarone The metabolism of Dronedarone can be decreased when combined with Curcumin.
Elexacaftor The serum concentration of Elexacaftor can be increased when it is combined with Curcumin.
Zanubrutinib The metabolism of Zanubrutinib can be decreased when combined with Curcumin.
Enfortumab vedotin The serum concentration of Enfortumab vedotin can be increased when it is combined with Curcumin.
Darolutamide The serum concentration of Darolutamide can be increased when it is combined with Curcumin.
Lumateperone The serum concentration of Lumateperone can be increased when it is combined with Curcumin.
Ubrogepant The serum concentration of Ubrogepant can be increased when it is combined with Curcumin.
Ranolazine The metabolism of Ranolazine can be decreased when combined with Curcumin.
Rimegepant The metabolism of Rimegepant can be decreased when combined with Curcumin.
Osilodrostat The serum concentration of Osilodrostat can be increased when it is combined with Curcumin.
Neratinib The serum concentration of Neratinib can be increased when it is combined with Curcumin.
Lovastatin The serum concentration of Lovastatin can be increased when it is combined with Curcumin.
Pemigatinib The metabolism of Pemigatinib can be decreased when combined with Curcumin.
Ripretinib The serum concentration of Ripretinib can be increased when it is combined with Curcumin.
Bortezomib The metabolism of Bortezomib can be decreased when combined with Curcumin.
Lurbinectedin The serum concentration of Lurbinectedin can be increased when it is combined with Curcumin.
Pralsetinib The serum concentration of Pralsetinib can be increased when it is combined with Curcumin.
Voclosporin The metabolism of Voclosporin can be decreased when combined with Curcumin.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Curcumin.
Avanafil The metabolism of Avanafil can be decreased when combined with Curcumin.
Silodosin The excretion of Silodosin can be decreased when combined with Curcumin.
Pimavanserin The metabolism of Pimavanserin can be decreased when combined with Curcumin.
Ticagrelor The metabolism of Ticagrelor can be decreased when combined with Curcumin.
Infigratinib The metabolism of Infigratinib can be decreased when combined with Curcumin.
Ibrexafungerp The serum concentration of Ibrexafungerp can be increased when it is combined with Curcumin.
Finerenone The serum concentration of the active metabolites of Finerenone can be increased when Finerenone is used in combination with Curcumin.
Methysergide The serum concentration of Methysergide can be increased when it is combined with Curcumin.
Cabergoline The metabolism of Cabergoline can be decreased when combined with Curcumin.
Dihydroergotamine The metabolism of Dihydroergotamine can be decreased when combined with Curcumin.
Methylergometrine The serum concentration of Methylergometrine can be increased when it is combined with Curcumin.
Lisuride The serum concentration of Lisuride can be increased when it is combined with Curcumin.
Ergotamine The metabolism of Ergotamine can be decreased when combined with Curcumin.
Nicergoline The serum concentration of Nicergoline can be increased when it is combined with Curcumin.
Ergoloid mesylate The serum concentration of Ergoloid mesylate can be increased when it is combined with Curcumin.
Pergolide The serum concentration of Pergolide can be increased when it is combined with Curcumin.
Bromocriptine The serum concentration of Bromocriptine can be increased when it is combined with Curcumin.
Ergometrine The serum concentration of Ergometrine can be increased when it is combined with Curcumin.
Lysergic acid diethylamide The serum concentration of Lysergic acid diethylamide can be increased when it is combined with Curcumin.
Dihydroergocornine The serum concentration of Dihydroergocornine can be increased when it is combined with Curcumin.
Dihydroergocristine The serum concentration of Dihydroergocristine can be increased when it is combined with Curcumin.
Dihydroergocryptine The serum concentration of Dihydroergocryptine can be increased when it is combined with Curcumin.
Terguride The serum concentration of Terguride can be increased when it is combined with Curcumin.
Metergoline The serum concentration of Metergoline can be increased when it is combined with Curcumin.
Simvastatin The risk or severity of myopathy and rhabdomyolysis can be increased when Curcumin is combined with Simvastatin.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Curcumin.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Curcumin.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Curcumin.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Curcumin.
Afatinib The serum concentration of Afatinib can be increased when it is combined with Curcumin.
Bosutinib The serum concentration of Bosutinib can be increased when it is combined with Curcumin.
Brentuximab vedotin The serum concentration of Brentuximab vedotin can be increased when it is combined with Curcumin.
Edoxaban The serum concentration of Edoxaban can be increased when it is combined with Curcumin.
Ledipasvir The serum concentration of Ledipasvir can be increased when it is combined with Curcumin.
Naloxegol The serum concentration of Naloxegol can be increased when it is combined with Curcumin.
Pazopanib The serum concentration of Pazopanib can be increased when it is combined with Curcumin.
Prucalopride The serum concentration of Prucalopride can be increased when it is combined with Curcumin.
Topotecan The serum concentration of Topotecan can be increased when it is combined with Curcumin.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Curcumin.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Curcumin.
Everolimus The serum concentration of Everolimus can be increased when it is combined with Curcumin.
Rifaximin The serum concentration of Rifaximin can be increased when it is combined with Curcumin.
Brexpiprazole The metabolism of Brexpiprazole can be decreased when combined with Curcumin.
Trastuzumab emtansine The metabolism of Trastuzumab emtansine can be decreased when combined with Curcumin.
Almotriptan The metabolism of Almotriptan can be decreased when combined with Curcumin.
Axitinib The metabolism of Axitinib can be decreased when combined with Curcumin.
Bedaquiline The metabolism of Bedaquiline can be decreased when combined with Curcumin.
Cabazitaxel The metabolism of Cabazitaxel can be decreased when combined with Curcumin.
Cabozantinib The metabolism of Cabozantinib can be decreased when combined with Curcumin.
Ceritinib The metabolism of Ceritinib can be decreased when combined with Curcumin.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Curcumin.
Daclatasvir The metabolism of Daclatasvir can be decreased when combined with Curcumin.
Dasatinib The metabolism of Dasatinib can be decreased when combined with Curcumin.
Erlotinib The metabolism of Erlotinib can be decreased when combined with Curcumin.
Fentanyl The metabolism of Fentanyl can be decreased when combined with Curcumin.
Fesoterodine The metabolism of Fesoterodine can be decreased when combined with Curcumin.
Flibanserin The metabolism of Flibanserin can be decreased when combined with Curcumin.
Guanfacine The metabolism of Guanfacine can be decreased when combined with Curcumin.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Curcumin.
Irinotecan The serum concentration of the active metabolites of Irinotecan can be decreased when Irinotecan is used in combination with Curcumin.
Lapatinib The metabolism of Lapatinib can be decreased when combined with Curcumin.
Milnacipran The metabolism of Milnacipran can be decreased when combined with Curcumin.
Levomilnacipran The metabolism of Levomilnacipran can be decreased when combined with Curcumin.
Maraviroc The metabolism of Maraviroc can be decreased when combined with Curcumin.
Mifepristone The metabolism of Mifepristone can be decreased when combined with Curcumin.
Nilotinib The metabolism of Nilotinib can be decreased when combined with Curcumin.
Olaparib The metabolism of Olaparib can be decreased when combined with Curcumin.
Palbociclib The metabolism of Palbociclib can be decreased when combined with Curcumin.
Panobinostat The metabolism of Panobinostat can be decreased when combined with Curcumin.
Ponatinib The metabolism of Ponatinib can be decreased when combined with Curcumin.
Quetiapine The serum concentration of Quetiapine can be increased when it is combined with Curcumin.

Target Protein

Cytochrome P450 3A4 CYP3A4
Nitric oxide synthase, inducible NOS2
Carbonic anhydrase 14 CA14
Carbonic anhydrase 1 CA1
Collagenase 3 MMP13
DNA (cytosine-5)-methyltransferase 3B DNMT3B
Xanthine dehydrogenase/oxidase XDH
Prostaglandin G/H synthase 1 PTGS1
Matrix metalloproteinase-9 MMP9
Prostaglandin G/H synthase 2 PTGS2
Carbonic anhydrase 4 CA4
Amyloid-beta precursor protein APP
Carbonic anhydrase 2 CA2
Carbonic anhydrase 12 CA12
Carbonic anhydrase 6 CA6
Carbonic anhydrase 9 CA9
Peroxisome proliferator-activated receptor gamma PPARG
Vitamin D3 receptor VDR
ATP-binding cassette sub-family C member 5 ABCC5
Carbonyl reductase [NADPH] 1 CBR1
Glutathione S-transferase P GSTP1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 23143785
    Gupta SC, Patchva S, Aggarwal BB: Therapeutic roles of curcumin: lessons learned from clinical trials. AAPS J. 2013 Jan;15(1):195-218. doi: 10.1208/s12248-012-9432-8. Epub 2012 Nov 10.
  • PMID: 27834897
    Lopes-Rodrigues V, Sousa E, Vasconcelos MH: Curcumin as a Modulator of P-Glycoprotein in Cancer: Challenges and Perspectives. Pharmaceuticals (Basel). 2016 Nov 10;9(4). pii: ph9040071. doi: 10.3390/ph9040071.

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