Rabusertib

DB11662

small molecule investigational

Deskripsi

Rabusertib has been used in trials studying the treatment of Cancer, Solid Tumors, Advanced Cancer, Pancreatic Neoplasms, and Non Small Cell Lung Cancer.

Struktur Molekul 2D

Berat 436.31
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

39 Data
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Rabusertib.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Rabusertib.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Rabusertib.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Rabusertib.
Lidocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Quinisocaine.
Nelarabine The risk or severity of adverse effects can be increased when Nelarabine is combined with Rabusertib.
Ambroxol The risk or severity of methemoglobinemia can be increased when Rabusertib is combined with Ambroxol.
Etrasimod The risk or severity of immunosuppression can be increased when Rabusertib is combined with Etrasimod.

Target Protein

Serine/threonine-protein kinase Chk1 CHEK1

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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