Peringatan Keamanan

The toxic effects of normethadone are similar to those of other opioids. It can produce respiratory depression, depression of central nervous system function, and constipation FDA Label.

Normethadone

DB11609

small molecule approved illicit

Deskripsi

Normethadone is used as an opioid antitussive in combination with DB11610. It is marketed in Canada by Valeant under the tradename Cophylac.

Struktur Molekul 2D

Berat 295.426
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol. Ingesting alcohol may cause additive CNS depressive effects.

Interaksi Obat

915 Data
Buprenorphine Normethadone may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Hydrocodone Normethadone may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Magnesium sulfate The therapeutic efficacy of Normethadone can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Normethadone may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Normethadone may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Orphenadrine Normethadone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Normethadone may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Pramipexole Normethadone may increase the sedative activities of Pramipexole.
Ropinirole Normethadone may increase the sedative activities of Ropinirole.
Rotigotine Normethadone may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Normethadone.
Sodium oxybate Normethadone may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Normethadone may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Thalidomide Normethadone may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Normethadone may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Alvimopan The risk or severity of adverse effects can be increased when Normethadone is combined with Alvimopan.
Desmopressin The risk or severity of hyponatremia can be increased when Normethadone is combined with Desmopressin.
Morphine The risk or severity of adverse effects can be increased when Morphine is combined with Normethadone.
Codeine The risk or severity of adverse effects can be increased when Codeine is combined with Normethadone.
Hydromorphone The risk or severity of adverse effects can be increased when Hydromorphone is combined with Normethadone.
Meperidine The risk or severity of adverse effects can be increased when Meperidine is combined with Normethadone.
Oxycodone The risk or severity of adverse effects can be increased when Oxycodone is combined with Normethadone.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Dextropropoxyphene is combined with Normethadone.
Naltrexone The therapeutic efficacy of Normethadone can be decreased when used in combination with Naltrexone.
Sufentanil The risk or severity of adverse effects can be increased when Sufentanil is combined with Normethadone.
Alfentanil The risk or severity of adverse effects can be increased when Alfentanil is combined with Normethadone.
Fentanyl The risk or severity of adverse effects can be increased when Fentanyl is combined with Normethadone.
Levorphanol The risk or severity of adverse effects can be increased when Levorphanol is combined with Normethadone.
Remifentanil The risk or severity of adverse effects can be increased when Remifentanil is combined with Normethadone.
Diphenoxylate The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Normethadone.
Oxymorphone The risk or severity of adverse effects can be increased when Oxymorphone is combined with Normethadone.
Dezocine The risk or severity of adverse effects can be increased when Dezocine is combined with Normethadone.
Methadyl acetate The risk or severity of adverse effects can be increased when Methadyl acetate is combined with Normethadone.
Dihydroetorphine The risk or severity of adverse effects can be increased when Dihydroetorphine is combined with Normethadone.
Diamorphine The risk or severity of adverse effects can be increased when Diamorphine is combined with Normethadone.
Bezitramide The risk or severity of adverse effects can be increased when Bezitramide is combined with Normethadone.
Ethylmorphine The risk or severity of adverse effects can be increased when Ethylmorphine is combined with Normethadone.
Etorphine The risk or severity of adverse effects can be increased when Etorphine is combined with Normethadone.
Dextromoramide The risk or severity of adverse effects can be increased when Dextromoramide is combined with Normethadone.
Desomorphine The risk or severity of adverse effects can be increased when Desomorphine is combined with Normethadone.
Carfentanil The risk or severity of adverse effects can be increased when Carfentanil is combined with Normethadone.
Dihydrocodeine The risk or severity of adverse effects can be increased when Dihydrocodeine is combined with Normethadone.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Alphacetylmethadol is combined with Normethadone.
Dihydromorphine The risk or severity of adverse effects can be increased when Dihydromorphine is combined with Normethadone.
Ketobemidone The risk or severity of adverse effects can be increased when Ketobemidone is combined with Normethadone.
DPDPE The risk or severity of adverse effects can be increased when DPDPE is combined with Normethadone.
Lofentanil The risk or severity of adverse effects can be increased when Lofentanil is combined with Normethadone.
Opium The risk or severity of adverse effects can be increased when Opium is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Normethadone is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Normethadone is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Normethadone is combined with Nicomorphine.
Meptazinol The therapeutic efficacy of Normethadone can be decreased when used in combination with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Normethadone is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Normethadone is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Normethadone is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Normethadone is combined with Carfentanil, C-11.
Naloxegol The risk or severity of adverse effects can be increased when Naloxegol is combined with Normethadone.
Benzhydrocodone The risk or severity of adverse effects can be increased when Normethadone is combined with Benzhydrocodone.
Pegvisomant The therapeutic efficacy of Pegvisomant can be decreased when used in combination with Normethadone.
Succinylcholine The risk or severity of bradycardia can be increased when Succinylcholine is combined with Normethadone.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Normethadone.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Normethadone.
Mirtazapine Normethadone may increase the serotonergic activities of Mirtazapine.
Fluvoxamine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Fluvoxamine.
Citalopram The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Citalopram.
Duloxetine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Duloxetine.
Paroxetine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Paroxetine.
Sertraline The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Sertraline.
Sibutramine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Sibutramine.
Nefazodone The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Nefazodone.
Zimelidine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Zimelidine.
Dapoxetine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Dapoxetine.
Milnacipran The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Normethadone.
Seproxetine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Levomilnacipran.
Indalpine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Indalpine.
Ritanserin The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Ritanserin.
Alaproclate The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Alaproclate.
Ethanol Normethadone may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Normethadone may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Normethadone.
Phentermine Phentermine may increase the analgesic activities of Normethadone.
Pseudoephedrine Pseudoephedrine may increase the analgesic activities of Normethadone.
Benzphetamine Benzphetamine may increase the analgesic activities of Normethadone.
Diethylpropion Diethylpropion may increase the analgesic activities of Normethadone.
Lisdexamfetamine The risk or severity of serotonin syndrome can be increased when Normethadone is combined with Lisdexamfetamine.
Mephentermine Mephentermine may increase the analgesic activities of Normethadone.
MMDA MMDA may increase the analgesic activities of Normethadone.
Midomafetamine Midomafetamine may increase the analgesic activities of Normethadone.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may increase the analgesic activities of Normethadone.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may increase the analgesic activities of Normethadone.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 1852031
    Adcock JJ: Peripheral opioid receptors and the cough reflex. Respir Med. 1991 Jan;85 Suppl A:43-6.

Contoh Produk & Brand

Produk: 3 • International brands: 0
Produk
  • Cophylac
    Solution / drops • - • Oral • Canada • Approved
  • Cophylac
    Solution / drops • - • Oral • Canada • Approved
  • Cophylac Drops
    Solution / drops • - • Oral • Canada • Approved

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