Peringatan Keamanan

Drometrizole trisiloxane is reported as having little to no absorption through the skin, which leads most national health agencies that approve its use in sunscreens (including the EU, Canada, Australia, Japan, and other countries) to consider it safe, given that most of their toxicity studies return little risk of adverse reactions as well A33069, L2780, L2781, L2782, L2783, F81.

Drometrizole trisiloxane

DB11585

small molecule approved

Deskripsi

Drometrizole trisiloxane is a photostable UVA and UVB light filter A33069, L2780, L2781, L2782, L2783, F81. The compound is a lipophilic benzotriazole derivative marketed as Meroxyl XL by L'Oreal, although sunscreens with drometrizole trisiloxane are currently only approved for use in the EU, Canada, Australia, and Japan, among other countries.

Despite being used elsewhere in the world with relatively few reports of adverse reactions, the FDA continues to cite that the existing scientific record is not sufficient to establish the compound as being generally recognized as safe and effective for over-the-counter sunscreen use L2795, F82.

Struktur Molekul 2D

Berat 501.849
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Drometrizole trisiloxane is reported as having little to no absorption through the skin [L2780, L2783]. The systemic presence of the compound is consequently expected to be minimal.
Volume Distribusi Drometrizole trisiloxane is reported as having little to no absorption through the skin [L2780, L2783]. The systemic presence of the compound is consequently expected to be minimal.
Klirens (Clearance) Drometrizole trisiloxane is reported as having little to no absorption through the skin [L2780, L2783]. The systemic presence of the compound is consequently expected to be minimal.

Absorpsi

Drometrizole trisiloxane is reported as having little to no absorption through the skin L2780, L2783. At this time, however, studies demonstrate that the components of most commonly used sunscreens are likely absorbed into the skin at least to some extent - although penetration to deeper tissues and the cutaneous circulation remains limited A33070. Despite the extensive use of sunscreen products around the world, there have been few reports of adverse effects related to their use A33070.

Metabolisme

Drometrizole trisiloxane is reported as having little to no absorption through the skin L2780, L2783. The systemic presence of the compound is consequently expected to be minimal.

Rute Eliminasi

Drometrizole trisiloxane is reported as having little to no absorption through the skin L2780, L2783. The systemic presence of the compound is consequently expected to be minimal.

Interaksi Obat

0 Data
Tidak ada data.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 18940542
    Gonzalez S, Fernandez-Lorente M, Gilaberte-Calzada Y: The latest on skin photoprotection. Clin Dermatol. 2008 Nov-Dec;26(6):614-26. doi: 10.1016/j.clindermatol.2007.09.010.
  • PMID: 11702366
    Benson HA: Assessment and clinical implications of absorption of sunscreens across skin. Am J Clin Dermatol. 2000 Jul-Aug;1(4):217-24.

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Sekuens Gen/Protein (FASTA)

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