Xylazine

DB11477

small molecule vet_approved

Deskripsi

Xylazine is a clonidine analog used as a non-opioid tranquilizer in veterinary medicine and as an emetic, especially in cats.A9095,L42675,A251420 It acts as an agonist at ?2 adrenoceptors; however, its affinity is lower than the one reported for other ?2 adrenergic receptor agonists such as detomidine and medetomidine.A32545 Xylazine is not approved for human use and requires a veterinary licence for its purchase and use.L42680 The intentional and unintentional use of xylazine is a cause for concern due to its side effects.A9096 The use of xylazine can lead to hypotension and bradycardiaA9092,A9093, and when combined with central nervous system depressants, such as benzodiazepines or alcohol, it can significantly depress vital functions and increase the risk of overdose and death.L42675 Xylazine is sometimes used as an adulterant and combined with opioids and recreational drugs; however, it has no antidote, and the use of naloxone has no effect on xylazine.L42675,L42680

Struktur Molekul 2D

Berat 220.33
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1150 Data
Valsartan Xylazine may decrease the antihypertensive activities of Valsartan.
Ramipril Xylazine may decrease the antihypertensive activities of Ramipril.
Remikiren Xylazine may decrease the antihypertensive activities of Remikiren.
Torasemide Xylazine may decrease the antihypertensive activities of Torasemide.
Isradipine Xylazine may decrease the antihypertensive activities of Isradipine.
Olmesartan Xylazine may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Xylazine may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Xylazine may decrease the antihypertensive activities of Nitroprusside.
Diltiazem Xylazine may decrease the antihypertensive activities of Diltiazem.
Minoxidil Xylazine may decrease the antihypertensive activities of Minoxidil.
Treprostinil Xylazine may decrease the antihypertensive activities of Treprostinil.
Amlodipine Xylazine may decrease the antihypertensive activities of Amlodipine.
Nimodipine Xylazine may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Xylazine may decrease the antihypertensive activities of Nisoldipine.
Bendroflumethiazide Xylazine may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Xylazine may decrease the antihypertensive activities of Fosinopril.
Trandolapril Xylazine may decrease the antihypertensive activities of Trandolapril.
Metolazone Xylazine may decrease the antihypertensive activities of Metolazone.
Lercanidipine Xylazine may decrease the antihypertensive activities of Lercanidipine.
Benazepril Xylazine may decrease the antihypertensive activities of Benazepril.
Bosentan Xylazine may decrease the antihypertensive activities of Bosentan.
Enalapril Xylazine may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Xylazine may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Xylazine may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Xylazine may decrease the antihypertensive activities of Mecamylamine.
Losartan Xylazine may decrease the antihypertensive activities of Losartan.
Moexipril Xylazine may decrease the antihypertensive activities of Moexipril.
Eplerenone Xylazine may decrease the antihypertensive activities of Eplerenone.
Lisinopril Xylazine may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Xylazine may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Xylazine may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Xylazine may decrease the antihypertensive activities of Cryptenamine.
Perindopril Xylazine may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Xylazine may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Xylazine may decrease the antihypertensive activities of Fenoldopam.
Indapamide Xylazine may decrease the antihypertensive activities of Indapamide.
Tadalafil Xylazine may decrease the antihypertensive activities of Tadalafil.
Eprosartan Xylazine may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Xylazine may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Xylazine may decrease the antihypertensive activities of Quinapril.
Telmisartan Xylazine may decrease the antihypertensive activities of Telmisartan.
Methyldopa Xylazine may decrease the antihypertensive activities of Methyldopa.
Hydrochlorothiazide Xylazine may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Xylazine may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Xylazine may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Xylazine may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Xylazine may decrease the antihypertensive activities of Deserpidine.
Pentolinium Xylazine may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Xylazine may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Xylazine may decrease the antihypertensive activities of Diazoxide.
Captopril Xylazine may decrease the antihypertensive activities of Captopril.
Epoprostenol Xylazine may decrease the antihypertensive activities of Epoprostenol.
Bepridil Xylazine may decrease the antihypertensive activities of Bepridil.
Hydralazine Xylazine may decrease the antihypertensive activities of Hydralazine.
Polythiazide Xylazine may decrease the antihypertensive activities of Polythiazide.
Cilazapril Xylazine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Xylazine may decrease the antihypertensive activities of Saprisartan.
Spirapril Xylazine may decrease the antihypertensive activities of Spirapril.
Mibefradil Xylazine may decrease the antihypertensive activities of Mibefradil.
Tienilic acid Xylazine may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Xylazine may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Xylazine may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Xylazine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Xylazine may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Xylazine may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Xylazine may decrease the antihypertensive activities of Pinacidil.
Temocapril Xylazine may decrease the antihypertensive activities of Temocapril.
Riociguat Xylazine may decrease the antihypertensive activities of Riociguat.
Macitentan Xylazine may decrease the antihypertensive activities of Macitentan.
Aliskiren Xylazine may decrease the antihypertensive activities of Aliskiren.
Nicorandil Xylazine may decrease the antihypertensive activities of Nicorandil.
Efonidipine Xylazine may decrease the antihypertensive activities of Efonidipine.
Lacidipine Xylazine may decrease the antihypertensive activities of Lacidipine.
Manidipine Xylazine may decrease the antihypertensive activities of Manidipine.
Rauwolfia serpentina root Xylazine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Xylazine may decrease the antihypertensive activities of Enalaprilat.
Selexipag Xylazine may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Xylazine may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Xylazine may decrease the antihypertensive activities of Imidapril.
BQ-123 Xylazine may decrease the antihypertensive activities of BQ-123.
Cicletanine Xylazine may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Xylazine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Xylazine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Xylazine may decrease the antihypertensive activities of Guanoxan.
Delapril Xylazine may decrease the antihypertensive activities of Delapril.
Vincamine Xylazine may decrease the antihypertensive activities of Vincamine.
Linsidomine Xylazine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Xylazine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Xylazine may decrease the antihypertensive activities of Tolonidine.
Endralazine Xylazine may decrease the antihypertensive activities of Endralazine.
Cadralazine Xylazine may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Xylazine may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Xylazine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Xylazine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Xylazine may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Xylazine may decrease the antihypertensive activities of Guanoclor.
Muzolimine Xylazine may decrease the antihypertensive activities of Muzolimine.
Xipamide Xylazine may decrease the antihypertensive activities of Xipamide.
Candesartan Xylazine may decrease the antihypertensive activities of Candesartan.
Dexniguldipine Xylazine may decrease the antihypertensive activities of Dexniguldipine.

Target Protein

Alpha-2B adrenergic receptor ADRA2B
Alpha-2C adrenergic receptor ADRA2C
Alpha-2 adrenergic receptors ADRA2A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16031828
    Beasley M: Xylazine. N Z Vet J. 1995 Jun;43(3):125.
  • PMID: 16031851
    Fyffe JJ: Xylazine. N Z Vet J. 1995 Oct;43(5):204-5.
  • PMID: 3963565
    Haskins SC, Patz JD, Farver TB: Xylazine and xylazine-ketamine in dogs. Am J Vet Res. 1986 Mar;47(3):636-41.
  • PMID: 17423135
    Haigh JC: Misuse of xylazine. Can Vet J. 1988 Oct;29(10):782-4.
  • PMID: 9597647
    Schwartz DD, Clark TP: Affinity of detomidine, medetomidine and xylazine for alpha-2 adrenergic receptor subtypes. J Vet Pharmacol Ther. 1998 Apr;21(2):107-11.
  • PMID: 7349332
    Colby ED, McCarthy LE, Borison HL: Emetic action of xylazine on the chemoreceptor trigger zone for vomiting in cats. J Vet Pharmacol Ther. 1981 Jun;4(2):93-6. doi: 10.1111/j.1365-2885.1981.tb00716.x.

Contoh Produk & Brand

Produk: 0 • International brands: 4
International Brands
  • Anased
  • Chanazine
  • Rompun
  • Sedazine

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul