Thiostrepton

DB11467

small molecule vet_approved

Deskripsi

Thiostrepton is a natural cyclic oligopeptide antibiotic, derived from several strains of streptomycetes including Streptomyces azureus and Streptomyces laurentii. Thiostrepton is a natural product of the ribosomally synthesized and post-translationally modified peptide class.

Struktur Molekul 2D

Berat 1664.89
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

55 Data
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Thiostrepton.
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Thiostrepton.
Typhoid vaccine The therapeutic efficacy of Typhoid vaccine can be decreased when used in combination with Thiostrepton.
Dicoumarol The risk or severity of bleeding can be increased when Thiostrepton is combined with Dicoumarol.
Phenindione The risk or severity of bleeding can be increased when Thiostrepton is combined with Phenindione.
Warfarin The risk or severity of bleeding can be increased when Thiostrepton is combined with Warfarin.
Phenprocoumon The risk or severity of bleeding can be increased when Thiostrepton is combined with Phenprocoumon.
Acenocoumarol The risk or severity of bleeding can be increased when Thiostrepton is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of bleeding can be increased when Thiostrepton is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of bleeding can be increased when Thiostrepton is combined with Coumarin.
(R)-warfarin The risk or severity of bleeding can be increased when Thiostrepton is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of bleeding can be increased when Thiostrepton is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of bleeding can be increased when Thiostrepton is combined with Fluindione.
Clorindione The risk or severity of bleeding can be increased when Thiostrepton is combined with Clorindione.
Diphenadione The risk or severity of bleeding can be increased when Thiostrepton is combined with Diphenadione.
Tioclomarol The risk or severity of bleeding can be increased when Thiostrepton is combined with Tioclomarol.
(S)-Warfarin The risk or severity of bleeding can be increased when Thiostrepton is combined with (S)-Warfarin.
Lactulose The therapeutic efficacy of Lactulose can be decreased when used in combination with Thiostrepton.
Vibrio cholerae CVD 103-HgR strain live antigen The therapeutic efficacy of Vibrio cholerae CVD 103-HgR strain live antigen can be decreased when used in combination with Thiostrepton.
Estetrol The therapeutic efficacy of Estetrol can be decreased when used in combination with Thiostrepton.
Lidocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Quinisocaine.
Cisatracurium Thiostrepton may increase the neuromuscular blocking activities of Cisatracurium.
Ambroxol The risk or severity of methemoglobinemia can be increased when Thiostrepton is combined with Ambroxol.
Fecal microbiota The therapeutic efficacy of Fecal microbiota can be decreased when used in combination with Thiostrepton.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 5416649
    Bodanszky M, Scozzie JA, Muramatsu I: Dehydroalanine residues in thiostrepton. J Antibiot (Tokyo). 1970 Jan;23(1):9-12.
  • PMID: 11266162
    Godoy-Alcantar C, Rivera IL, Yatsimirsky AK: Anion recognition by thiostrepton. Bioorg Med Chem Lett. 2001 Mar 12;11(5):651-4.
  • PMID: 5409975
    Anderson B, Hodgkin DC, Viswamitra MA: The structure of thiostrepton. Nature. 1970 Jan 17;225(5229):233-5.
  • PMID: 13486397
    COHN I Jr, LONGACRE AB: Thiostrepton and thiostrepton-neomycin for preoperative preparation of the colon. Surgery. 1957 Nov;42(5):865-73.
  • PMID: 440414
    Cundliffe E, Thompson J: Ribose methylation and resistance to thiostrepton. Nature. 1979 Apr 26;278(5707):859-61.
  • PMID: 9109400
    Clough B, Strath M, Preiser P, Denny P, Wilson IR: Thiostrepton binds to malarial plastid rRNA. FEBS Lett. 1997 Apr 7;406(1-2):123-5.
  • PMID: 908663
    Trejo WH, Dean LD, Pluscec J, Meyers E, Brown WE: Streptomyces laurentii, a new species producing thiostrepton. J Antibiot (Tokyo). 1977 Aug;30(8):639-43.
  • PMID: 15199170
    Cameron DM, Thompson J, Gregory ST, March PE, Dahlberg AE: Thiostrepton-resistant mutants of Thermus thermophilus. Nucleic Acids Res. 2004 Jun 15;32(10):3220-7. Print 2004.
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