Medetomidine

DB11428

small molecule experimental vet_approved

Deskripsi

Medetomidine is a synthetic compound used as a surgical anesthetic and analgesic. It is normally found as its hydrochloride salt, medetomidine hydrochloride. Medetomidine is an intravenously available alpha-2 adrenergic agonist. The drug has been developed by Orion Pharma. In the United States, it is currently approved for its veterinary use in dogs and distributed by Pfizer Animal Health. In Canada, medetomidine is distributed by Novartis Animal Health. The marketed product is a racemic mixture of two stereoisomers from which dexmedetomidine is the main active isomer.

Struktur Molekul 2D

Berat 200.2795
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1144 Data
Valsartan Medetomidine may decrease the antihypertensive activities of Valsartan.
Ramipril Medetomidine may decrease the antihypertensive activities of Ramipril.
Remikiren Medetomidine may decrease the antihypertensive activities of Remikiren.
Torasemide Medetomidine may decrease the antihypertensive activities of Torasemide.
Isradipine Medetomidine may decrease the antihypertensive activities of Isradipine.
Olmesartan Medetomidine may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Medetomidine may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Medetomidine may decrease the antihypertensive activities of Nitroprusside.
Diltiazem Medetomidine may decrease the antihypertensive activities of Diltiazem.
Minoxidil Medetomidine may decrease the antihypertensive activities of Minoxidil.
Treprostinil Medetomidine may decrease the antihypertensive activities of Treprostinil.
Amlodipine Medetomidine may decrease the antihypertensive activities of Amlodipine.
Nimodipine Medetomidine may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Medetomidine may decrease the antihypertensive activities of Nisoldipine.
Bendroflumethiazide Medetomidine may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Medetomidine may decrease the antihypertensive activities of Fosinopril.
Trandolapril Medetomidine may decrease the antihypertensive activities of Trandolapril.
Metolazone Medetomidine may decrease the antihypertensive activities of Metolazone.
Lercanidipine Medetomidine may decrease the antihypertensive activities of Lercanidipine.
Benazepril Medetomidine may decrease the antihypertensive activities of Benazepril.
Bosentan Medetomidine may decrease the antihypertensive activities of Bosentan.
Enalapril Medetomidine may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Medetomidine may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Medetomidine may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Medetomidine may decrease the antihypertensive activities of Mecamylamine.
Losartan Medetomidine may decrease the antihypertensive activities of Losartan.
Moexipril Medetomidine may decrease the antihypertensive activities of Moexipril.
Eplerenone Medetomidine may decrease the antihypertensive activities of Eplerenone.
Lisinopril Medetomidine may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Medetomidine may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Medetomidine may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Medetomidine may decrease the antihypertensive activities of Cryptenamine.
Perindopril Medetomidine may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Medetomidine may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Medetomidine may decrease the antihypertensive activities of Fenoldopam.
Indapamide Medetomidine may decrease the antihypertensive activities of Indapamide.
Tadalafil Medetomidine may decrease the antihypertensive activities of Tadalafil.
Eprosartan Medetomidine may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Medetomidine may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Medetomidine may decrease the antihypertensive activities of Quinapril.
Telmisartan Medetomidine may decrease the antihypertensive activities of Telmisartan.
Methyldopa Medetomidine may decrease the antihypertensive activities of Methyldopa.
Hydrochlorothiazide Medetomidine may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Medetomidine may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Medetomidine may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Medetomidine may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Medetomidine may decrease the antihypertensive activities of Deserpidine.
Pentolinium Medetomidine may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Medetomidine may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Medetomidine may decrease the antihypertensive activities of Diazoxide.
Captopril Medetomidine may decrease the antihypertensive activities of Captopril.
Epoprostenol Medetomidine may decrease the antihypertensive activities of Epoprostenol.
Bepridil Medetomidine may decrease the antihypertensive activities of Bepridil.
Hydralazine Medetomidine may decrease the antihypertensive activities of Hydralazine.
Polythiazide Medetomidine may decrease the antihypertensive activities of Polythiazide.
Cilazapril Medetomidine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Medetomidine may decrease the antihypertensive activities of Saprisartan.
Spirapril Medetomidine may decrease the antihypertensive activities of Spirapril.
Mibefradil Medetomidine may decrease the antihypertensive activities of Mibefradil.
Tienilic acid Medetomidine may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Medetomidine may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Medetomidine may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Medetomidine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Medetomidine may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Medetomidine may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Medetomidine may decrease the antihypertensive activities of Pinacidil.
Temocapril Medetomidine may decrease the antihypertensive activities of Temocapril.
Riociguat Medetomidine may decrease the antihypertensive activities of Riociguat.
Macitentan Medetomidine may decrease the antihypertensive activities of Macitentan.
Aliskiren Medetomidine may decrease the antihypertensive activities of Aliskiren.
Nicorandil Medetomidine may decrease the antihypertensive activities of Nicorandil.
Efonidipine Medetomidine may decrease the antihypertensive activities of Efonidipine.
Lacidipine Medetomidine may decrease the antihypertensive activities of Lacidipine.
Manidipine Medetomidine may decrease the antihypertensive activities of Manidipine.
Rauwolfia serpentina root Medetomidine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Medetomidine may decrease the antihypertensive activities of Enalaprilat.
Selexipag Medetomidine may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Medetomidine may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Medetomidine may decrease the antihypertensive activities of Imidapril.
BQ-123 Medetomidine may decrease the antihypertensive activities of BQ-123.
Cicletanine Medetomidine may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Medetomidine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Medetomidine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Medetomidine may decrease the antihypertensive activities of Guanoxan.
Delapril Medetomidine may decrease the antihypertensive activities of Delapril.
Vincamine Medetomidine may decrease the antihypertensive activities of Vincamine.
Linsidomine Medetomidine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Medetomidine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Medetomidine may decrease the antihypertensive activities of Tolonidine.
Endralazine Medetomidine may decrease the antihypertensive activities of Endralazine.
Cadralazine Medetomidine may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Medetomidine may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Medetomidine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Medetomidine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Medetomidine may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Medetomidine may decrease the antihypertensive activities of Guanoclor.
Muzolimine Medetomidine may decrease the antihypertensive activities of Muzolimine.
Xipamide Medetomidine may decrease the antihypertensive activities of Xipamide.
Candesartan Medetomidine may decrease the antihypertensive activities of Candesartan.
Dexniguldipine Medetomidine may decrease the antihypertensive activities of Dexniguldipine.

Target Protein

Alpha-2A adrenergic receptor ADRA2A
Alpha-1B adrenergic receptor ADRA1B
Alpha-1D adrenergic receptor ADRA1D
Alpha-2B adrenergic receptor ADRA2B
Alpha-1A adrenergic receptor ADRA1A
Alpha-2C adrenergic receptor ADRA2C

Referensi & Sumber

Artikel (PubMed)
  • PMID: 8966714
    Hellebrekers LJ: Medetomidine. Tijdschr Diergeneeskd. 1996 Nov 1;121(21):634.
  • PMID: 8212947
    Mohammad FK, Zangana IK, Abdul-Latif AR: Medetomidine sedation in sheep. Zentralbl Veterinarmed A. 1993 Jun;40(5):328-31.
  • PMID: 1763477
    Jones P, Hoare C: Medetomidine in horses. Vet Rec. 1991 Nov 23;129(21):476.
  • PMID: 2571277
    Salonen JS: Pharmacokinetics of medetomidine. Acta Vet Scand Suppl. 1989;85:49-54.
  • PMID: 2316155
    Crighton M: Diuresis following medetomidine. Vet Rec. 1990 Feb 24;126(8):201.
  • PMID: 2309424
    Manners H: Anaesthesia following medetomidine. Vet Rec. 1990 Feb 17;126(7):174.
  • PMID: 2571266
    Vaha-Vahe T: The clinical efficacy of medetomidine. Acta Vet Scand Suppl. 1989;85:151-3.
  • PMID: 9278121
    Ko JC, Heaton-Jones TG, Nicklin CF: Evaluation of the sedative and cardiorespiratory effects of medetomidine, medetomidine-butorphanol, medetomidine-ketamine, and medetomidine-butorphanol-ketamine in ferrets. J Am Anim Hosp Assoc. 1997 Sep-Oct;33(5):438-48.
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Sekuens Gen/Protein (FASTA)

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