Amitraz

DB11373

small molecule experimental vet_approved

Deskripsi

Amitraz is a non-systemic acaricide and insecticide. It was generated in 1969 by the Boots Co. in England. Amitraz presents insect repellent effects and hence, it can be used as an insecticide and pesticide. Its insecticide effect is due to its agonistic activity in the alpha-adrenergic system, its interaction with the octopamine receptors in the central nervous system and its driven inhibition of the synthesis of monoamine oxidases and prostaglandins. All the abovementioned effects are translated into the overexcitation, paralysis, and death in insects.

Amitraz presents a lower effect in mammals and thus, it is widely used in the treatment of mite- or tick-infestation of dogs.

Struktur Molekul 2D

Berat 293.406
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

672 Data
Valsartan Amitraz may decrease the antihypertensive activities of Valsartan.
Ramipril Amitraz may decrease the antihypertensive activities of Ramipril.
Reserpine Amitraz may decrease the antihypertensive activities of Reserpine.
Remikiren Amitraz may decrease the antihypertensive activities of Remikiren.
Torasemide Amitraz may decrease the antihypertensive activities of Torasemide.
Isradipine Amitraz may decrease the antihypertensive activities of Isradipine.
Olmesartan Amitraz may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Amitraz may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Amitraz may decrease the antihypertensive activities of Nitroprusside.
Diltiazem Amitraz may decrease the antihypertensive activities of Diltiazem.
Minoxidil Amitraz may decrease the antihypertensive activities of Minoxidil.
Treprostinil Amitraz may decrease the antihypertensive activities of Treprostinil.
Amlodipine Amitraz may decrease the antihypertensive activities of Amlodipine.
Nimodipine Amitraz may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Amitraz may decrease the antihypertensive activities of Nisoldipine.
Bendroflumethiazide Amitraz may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Amitraz may decrease the antihypertensive activities of Fosinopril.
Trandolapril Amitraz may decrease the antihypertensive activities of Trandolapril.
Metolazone Amitraz may decrease the antihypertensive activities of Metolazone.
Lercanidipine Amitraz may decrease the antihypertensive activities of Lercanidipine.
Benazepril Amitraz may decrease the antihypertensive activities of Benazepril.
Bosentan Amitraz may decrease the antihypertensive activities of Bosentan.
Enalapril Amitraz may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Amitraz may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Amitraz may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Amitraz may decrease the antihypertensive activities of Mecamylamine.
Losartan Amitraz may decrease the antihypertensive activities of Losartan.
Moexipril Amitraz may decrease the antihypertensive activities of Moexipril.
Eplerenone Amitraz may decrease the antihypertensive activities of Eplerenone.
Lisinopril Amitraz may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Amitraz may decrease the antihypertensive activities of Nitroglycerin.
Metyrosine Amitraz may decrease the antihypertensive activities of Metyrosine.
Hydroflumethiazide Amitraz may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Amitraz may decrease the antihypertensive activities of Cryptenamine.
Perindopril Amitraz may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Amitraz may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Amitraz may decrease the antihypertensive activities of Fenoldopam.
Indapamide Amitraz may decrease the antihypertensive activities of Indapamide.
Tadalafil Amitraz may decrease the antihypertensive activities of Tadalafil.
Eprosartan Amitraz may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Amitraz may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Amitraz may decrease the antihypertensive activities of Quinapril.
Telmisartan Amitraz may decrease the antihypertensive activities of Telmisartan.
Methyldopa Amitraz may decrease the antihypertensive activities of Methyldopa.
Hydrochlorothiazide Amitraz may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Amitraz may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Amitraz may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Amitraz may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Amitraz may decrease the antihypertensive activities of Deserpidine.
Pentolinium Amitraz may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Amitraz may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Amitraz may decrease the antihypertensive activities of Diazoxide.
Captopril Amitraz may decrease the antihypertensive activities of Captopril.
Epoprostenol Amitraz may decrease the antihypertensive activities of Epoprostenol.
Bepridil Amitraz may decrease the antihypertensive activities of Bepridil.
Hydralazine Amitraz may decrease the antihypertensive activities of Hydralazine.
Polythiazide Amitraz may decrease the antihypertensive activities of Polythiazide.
Cilazapril Amitraz may decrease the antihypertensive activities of Cilazapril.
Saprisartan Amitraz may decrease the antihypertensive activities of Saprisartan.
Spirapril Amitraz may decrease the antihypertensive activities of Spirapril.
Mibefradil Amitraz may decrease the antihypertensive activities of Mibefradil.
Tienilic acid Amitraz may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Amitraz may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Amitraz may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Amitraz may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Amitraz may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Amitraz may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Amitraz may decrease the antihypertensive activities of Pinacidil.
Temocapril Amitraz may decrease the antihypertensive activities of Temocapril.
Riociguat Amitraz may decrease the antihypertensive activities of Riociguat.
Macitentan Amitraz may decrease the antihypertensive activities of Macitentan.
Hexamethonium Amitraz may decrease the antihypertensive activities of Hexamethonium.
Aliskiren Amitraz may decrease the antihypertensive activities of Aliskiren.
Nicorandil Amitraz may decrease the antihypertensive activities of Nicorandil.
Efonidipine Amitraz may decrease the antihypertensive activities of Efonidipine.
Lacidipine Amitraz may decrease the antihypertensive activities of Lacidipine.
Manidipine Amitraz may decrease the antihypertensive activities of Manidipine.
Rauwolfia serpentina root Amitraz may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Amitraz may decrease the antihypertensive activities of Enalaprilat.
Selexipag Amitraz may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Amitraz may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Amitraz may decrease the antihypertensive activities of Imidapril.
BQ-123 Amitraz may decrease the antihypertensive activities of BQ-123.
Tetrahydropalmatine Amitraz may decrease the antihypertensive activities of Tetrahydropalmatine.
Cicletanine Amitraz may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Amitraz may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Amitraz may decrease the antihypertensive activities of Zofenopril.
Guanoxan Amitraz may decrease the antihypertensive activities of Guanoxan.
Delapril Amitraz may decrease the antihypertensive activities of Delapril.
Vincamine Amitraz may decrease the antihypertensive activities of Vincamine.
Linsidomine Amitraz may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Amitraz may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Amitraz may decrease the antihypertensive activities of Tolonidine.
Endralazine Amitraz may decrease the antihypertensive activities of Endralazine.
Cadralazine Amitraz may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Amitraz may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Amitraz may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Amitraz may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Amitraz may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Amitraz may decrease the antihypertensive activities of Guanoclor.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 24109378
    Lee S, Kim TH, Shin YW, Jeon Y, Kim J: Amitraz. Acta Crystallogr Sect E Struct Rep Online. 2013 Jul 24;69(Pt 8):o1300. doi: 10.1107/S1600536813019764. eCollection 2013.
  • PMID: 22576295
    Varma PV, Bhatt S, Bhat RY: Amitraz poisoning. Indian J Pediatr. 2013 Apr;80(4):349-50. doi: 10.1007/s12098-012-0772-2. Epub 2012 May 11.
  • PMID: 19809769
    Caprotta CG, Martinez M, Tiszler M, Guerra V: Amitraz poisoning. Arch Argent Pediatr. 2009 Oct;107(5):456-8. doi: 10.1590/S0325-00752009000500015.
  • PMID: 15822764
    Gursoy S, Kunt N, Kaygusuz K, Kafali H: Intravenous amitraz poisoning. Clin Toxicol (Phila). 2005;43(2):113-6.
  • PMID: 12029457
    Aydin K, Per H, Kurtoglu S, Poyrazoglu MH, Narin N, Aslan D: Amitraz poisoning in children. Eur J Pediatr. 2002 Jun;161(6):349-50. Epub 2002 Apr 16.
  • PMID: 11125712
    Yaramis A, Soker M, Bilici M: Amitraz poisoning in children. Hum Exp Toxicol. 2000 Aug;19(8):431-3.
  • PMID: 10885999
    Saha T, Chatterjee S, Saha K, Chowdhury A, Somchoudhury AK, Bhattacharyya A: Residues of amitraz, a new acaricide, on tea. Bull Environ Contam Toxicol. 2000 Aug;65(2):215-21.
  • PMID: 24288053
    Godara R, Parveen S, Katoch R, Yadav A, Verma PK, Katoch M, Kaur D, Ganai A, Raghuvanshi P, Singh NK: Acaricidal activity of extract of Artemisia absinthium against Rhipicephalus sanguineus of dogs. Parasitol Res. 2014 Feb;113(2):747-54. doi: 10.1007/s00436-013-3704-9. Epub 2013 Nov 28.
Menampilkan 8 dari 11 artikel.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Mitac

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul