Peringatan Keamanan

Acute oral toxicity (LD50): 2650 mg/kg Rat MSDS.

Clove oil is considered safe in small quantities (< 1,500 ppm) as a food additive F108. The lethal oral dose is 3.75 g per kg body weight in humans F108.

Contact with skin or soft tissue may cause transient irritation, contact dermatitis, inflammation of the lips, and inflammation or ulceration of the mouth. The eugenol present in clove oil may act as an irritant to skin and mucous membranes; it may also cause hypersensitivity and is reported to inhibit prostaglandin synthesis. Patients may become sensitive to clove oil L2850.

After oral administration of 5-10 ml of clove oil in children below 2 years of age, life-threatening conditions were observed. Adverse effects included coma, acidosis, a generalized seizure, disordered blood clotting, and acute liver damage F108.

Overdose may lead to CNS depression, urinary abnormalities, anion-gap acidosis, deterioration of liver function, coma, seizure and low blood glucose levels. Treatment should be supportive and symptomatic; there have been reports in the literature that N-acetylcysteine has been successfully used as an antidote L2850.

There are no epidemiological studies of potential adverse human health effects related to exposure to clove leave oil or eugenol from any human exposure scenarios. Nor are there any studies of agricultural use, either in workers or those with bystander exposure or other applications. There are no occupational exposure standards for clove leaf oil or eugenol including OSHA PEL (Permissible Exposure Limit) or AGIHA TLVs (Threshold Limit Value) in air F108.

Clove oil

DB11338

biotech approved nutraceutical

Deskripsi

Clove oil is obtained by extraction from the dried flower buds of the clove plant. Traditionally, it has been used as a flavouring spice in foods, or as a fragrance. It is also found in topical analgesics. Clove oil has shown to exert some antimicrobial activities. The antioxidant and antimicrobial activity of clove is higher than that of many fruits, vegetables, and other spices A33133.

Clove is native of Indonesia but is now cultured in several parts of the world, including Brazil in the state of Bahia. This plant represents one of the richest source of phenolic compounds such as eugenol, eugenol acetate and gallic acid and has great potential for pharmaceutical, cosmetic, food and agricultural applications A33133.

Interestingly, clove oil has been studied for its potential benefit in treating neuropathic pain, as well as vaginal candidiasis with promising results A33137, A33144.

The FDA categorizes clove oil as generally recognized as safe (GRAS) for use in dental cement or as a food additive F108.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) In a pharmacokinetic study, average half-life values of eugenol in plasma and blood were long (14.0 and 18.3 h, respectively), suggesting a potential accumulation of the drug following repeated administrations [A33137].
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Clove oil is rapidly absorbed through the skin and is used in patented systems for dermal drug delivery to enhance drug uptake from skin patch delivery systems F108.

Metabolisme

In the rat, 20-30% of eugenol is metabolized to homovanillic acid and 4-hydroxy-3-methoxymandelic acid L2850. In a pharmacokinetic study in man, 95% of the ingested eugenol dose was recovered in the urine, most of which (greater than 99%) consisted of phenolic conjugates; 50% of the conjugated metabolites were eugenol-glucuronide and sulfate. Other metabolic routes observed were the epoxide-diol pathway, synthesis of a thiophenol and of a substituted propionic acid, allylic oxidation, and migration of the double bond A33147.

Rute Eliminasi

In a pharmacokinetic study, the metabolism of eugenol (the primary constituent of clove oil) was investigated in healthy male and female volunteers. It was quickly absorbed and metabolized after oral administration and was almost completely excreted in the urine within 24 hours of ingestion A33147.

Interaksi Obat

727 Data
Cyclosporine Cyclosporine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Icosapent Icosapent may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefotiam Cefotiam may decrease the excretion rate of Clove oil which could result in a higher serum level.
Mesalazine Mesalazine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefmenoxime Cefmenoxime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefmetazole Cefmetazole may decrease the excretion rate of Clove oil which could result in a higher serum level.
Pamidronic acid Pamidronic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Tenofovir disoproxil Tenofovir disoproxil may decrease the excretion rate of Clove oil which could result in a higher serum level.
Indomethacin Indomethacin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cidofovir Cidofovir may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefpiramide Cefpiramide may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftazidime Ceftazidime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Loracarbef Loracarbef may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefalotin Cefalotin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Nabumetone Nabumetone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ketorolac Ketorolac may decrease the excretion rate of Clove oil which could result in a higher serum level.
Tenoxicam Tenoxicam may decrease the excretion rate of Clove oil which could result in a higher serum level.
Celecoxib Celecoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefotaxime Cefotaxime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Tolmetin Tolmetin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Foscarnet Foscarnet may decrease the excretion rate of Clove oil which could result in a higher serum level.
Rofecoxib Rofecoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Piroxicam Piroxicam may decrease the excretion rate of Clove oil which could result in a higher serum level.
Methotrexate Methotrexate may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cephalexin Cephalexin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Fenoprofen Fenoprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Valaciclovir Valaciclovir may decrease the excretion rate of Clove oil which could result in a higher serum level.
Valdecoxib Valdecoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Diclofenac Diclofenac may decrease the excretion rate of Clove oil which could result in a higher serum level.
Sulindac Sulindac may decrease the excretion rate of Clove oil which could result in a higher serum level.
Bacitracin Bacitracin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Amphotericin B Amphotericin B may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cephaloglycin Cephaloglycin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Flurbiprofen Flurbiprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Adefovir dipivoxil Adefovir dipivoxil may decrease the excretion rate of Clove oil which could result in a higher serum level.
Pentamidine Pentamidine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Etodolac Etodolac may decrease the excretion rate of Clove oil which could result in a higher serum level.
Mefenamic acid Mefenamic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Acyclovir Acyclovir may decrease the excretion rate of Clove oil which could result in a higher serum level.
Naproxen Naproxen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Sulfasalazine Sulfasalazine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Phenylbutazone Phenylbutazone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Meloxicam Meloxicam may decrease the excretion rate of Clove oil which could result in a higher serum level.
Carprofen Carprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefaclor Cefaclor may decrease the excretion rate of Clove oil which could result in a higher serum level.
Diflunisal Diflunisal may decrease the excretion rate of Clove oil which could result in a higher serum level.
Tacrolimus Tacrolimus may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceforanide Ceforanide may decrease the excretion rate of Clove oil which could result in a higher serum level.
Salicylic acid Salicylic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Meclofenamic acid Meclofenamic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Acetylsalicylic acid Acetylsalicylic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Carboplatin Carboplatin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Oxaprozin Oxaprozin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ketoprofen Ketoprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Balsalazide Balsalazide may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ibuprofen Ibuprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefditoren Cefditoren may decrease the excretion rate of Clove oil which could result in a higher serum level.
Atazanavir Atazanavir may decrease the excretion rate of Clove oil which could result in a higher serum level.
Colistimethate Colistimethate may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefuroxime Cefuroxime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefapirin Cefapirin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefadroxil Cefadroxil may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefprozil Cefprozil may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftriaxone Ceftriaxone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Olsalazine Olsalazine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Lumiracoxib Lumiracoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefamandole Cefamandole may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefazolin Cefazolin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefonicid Cefonicid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefoperazone Cefoperazone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefotetan Cefotetan may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefoxitin Cefoxitin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftizoxime Ceftizoxime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefradine Cefradine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Magnesium salicylate Magnesium salicylate may decrease the excretion rate of Clove oil which could result in a higher serum level.
Salsalate Salsalate may decrease the excretion rate of Clove oil which could result in a higher serum level.
Choline magnesium trisalicylate Choline magnesium trisalicylate may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefepime Cefepime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefacetrile Cefacetrile may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftibuten Ceftibuten may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cefpodoxime Cefpodoxime may decrease the excretion rate of Clove oil which could result in a higher serum level.
Antrafenine Antrafenine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Aminophenazone Aminophenazone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Antipyrine Antipyrine may decrease the excretion rate of Clove oil which could result in a higher serum level.
Tiaprofenic acid Tiaprofenic acid may decrease the excretion rate of Clove oil which could result in a higher serum level.
Lopinavir Lopinavir may decrease the excretion rate of Clove oil which could result in a higher serum level.
Etoricoxib Etoricoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Hydrolyzed Cephalothin Hydrolyzed Cephalothin may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cephalothin Group Cephalothin Group may decrease the excretion rate of Clove oil which could result in a higher serum level.
Oxyphenbutazone Oxyphenbutazone may decrease the excretion rate of Clove oil which could result in a higher serum level.
Latamoxef Latamoxef may decrease the excretion rate of Clove oil which could result in a higher serum level.
Nimesulide Nimesulide may decrease the excretion rate of Clove oil which could result in a higher serum level.
Benoxaprofen Benoxaprofen may decrease the excretion rate of Clove oil which could result in a higher serum level.
Metamizole Metamizole may decrease the excretion rate of Clove oil which could result in a higher serum level.
Zomepirac Zomepirac may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftobiprole Ceftobiprole may decrease the excretion rate of Clove oil which could result in a higher serum level.
Cimicoxib Cimicoxib may decrease the excretion rate of Clove oil which could result in a higher serum level.
Ceftaroline fosamil Ceftaroline fosamil may decrease the excretion rate of Clove oil which could result in a higher serum level.
Lornoxicam Lornoxicam may decrease the excretion rate of Clove oil which could result in a higher serum level.
Aceclofenac Aceclofenac may decrease the excretion rate of Clove oil which could result in a higher serum level.

Target Protein

Vascular cell adhesion protein 1 VCAM1
C-X-C motif chemokine 10 CXCL10
Collagen alpha-1(I) chain COL1A1
Granulocyte-macrophage colony-stimulating factor receptor subunit alpha CSF2RA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 24031950
    Nunez L, Aquino MD: Microbicide activity of clove essential oil (Eugenia caryophyllata). Braz J Microbiol. 2012 Oct;43(4):1255-60. doi: 10.1590/S1517-83822012000400003. Epub 2012 Jun 1.
  • PMID: 25182278
    Cortes-Rojas DF, de Souza CR, Oliveira WP: Clove (Syzygium aromaticum): a precious spice. Asian Pac J Trop Biomed. 2014 Feb;4(2):90-6. doi: 10.1016/S2221-1691(14)60215-X.
  • PMID: 28407719
    Han X, Parker TL: Anti-inflammatory activity of clove (Eugenia caryophyllata) essential oil in human dermal fibroblasts. Pharm Biol. 2017 Dec;55(1):1619-1622. doi: 10.1080/13880209.2017.1314513.
  • PMID: 17321520
    Guenette SA, Ross A, Marier JF, Beaudry F, Vachon P: Pharmacokinetics of eugenol and its effects on thermal hypersensitivity in rats. Eur J Pharmacol. 2007 May 7;562(1-2):60-7. doi: 10.1016/j.ejphar.2007.01.044. Epub 2007 Feb 1.
  • PMID: 16390816
    Ahmad N, Alam MK, Shehbaz A, Khan A, Mannan A, Hakim SR, Bisht D, Owais M: Antimicrobial activity of clove oil and its potential in the treatment of vaginal candidiasis. J Drug Target. 2005 Dec;13(10):555-61. doi: 10.1080/10611860500422958 .
  • PMID: 1818340
    Pongprayoon U, Baeckstrom P, Jacobsson U, Lindstrom M, Bohlin L: Compounds inhibiting prostaglandin synthesis isolated from Ipomoea pes-caprae. Planta Med. 1991 Dec;57(6):515-8. doi: 10.1055/s-2006-960196.
  • PMID: 15922856
    Yoo CB, Han KT, Cho KS, Ha J, Park HJ, Nam JH, Kil UH, Lee KT: Eugenol isolated from the essential oil of Eugenia caryophyllata induces a reactive oxygen species-mediated apoptosis in HL-60 human promyelocytic leukemia cells. Cancer Lett. 2005 Jul 8;225(1):41-52. doi: 10.1016/j.canlet.2004.11.018. Epub 2004 Dec 15.
  • PMID: 2333717
    Fischer IU, von Unruh GE, Dengler HJ: The metabolism of eugenol in man. Xenobiotica. 1990 Feb;20(2):209-22.

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