Peringatan Keamanan

Both oral LD50 and dermal LD50 in rat is > 2000 mg/kg MSDS. In a developmental toxicity study of rats, the maternal and developmental no-observed-effect-level (NOEL) of bisoctrizole was the high dose level of 1000 mg/kg bw/day F90. Animal studies suggest that bisoctrizole mediates no phytotoxic effects F90.

Bisoctrizole

DB11262

small molecule approved

Deskripsi

Bisoctrizole, or methylene bis-benzotriazolyl tetramethylbutylphenol, is a broad-spectrum organic UV filter that is marketed as Tinosorb M A19212. It is a benzotriazole-based organic compound that absorbs, reflects, and scatters both UV-A and UV-B rays. Bisoctrizole is not approved by the FDA, but is approved in the EU and other parts of the world as a UV-filter in sunscreens, day care products and skin lightening products at a maximum concentration of 10% F90.

Struktur Molekul 2D

Berat 658.891
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) No pharmacokinetic data available.
Volume Distribusi No pharmacokinetic data available.
Klirens (Clearance) No pharmacokinetic data available.

Absorpsi

A rat and human dermal penetration study in vitro indicates that bisoctrizole displays minimal absorption through the skin, with only about 0.01% and 0.06 % of the applied dose penetration through the human and rat skin membrane, respectively F90. Despite low dermal uptake, potential bioaccumulation after repeated skin applications cannot be excluded F90.

Metabolisme

No pharmacokinetic data available.

Rute Eliminasi

No pharmacokinetic data available.

Interaksi Obat

0 Data
Tidak ada data.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 23320122
    Latha MS, Martis J, Shobha V, Sham Shinde R, Bangera S, Krishnankutty B, Bellary S, Varughese S, Rao P, Naveen Kumar BR: Sunscreening agents: a review. J Clin Aesthet Dermatol. 2013 Jan;6(1):16-26.

Contoh Produk & Brand

Produk: 26 • International brands: 0
Produk
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    Emulsion • - • Topical • Canada • OTC • Approved
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    Gel • - • Topical • US • OTC
  • Emulsion SPF 50+
    Emulsion • - • Topical • Canada • OTC • Approved
  • High Protection Emulsion
    Emulsion • - • Topical • Canada • OTC • Approved
  • High Protection Lotion
    Lotion • - • Topical • Canada • OTC • Approved
  • High Protection Lotion SPF 50+
    Lotion • - • Topical • Canada • OTC • Approved
  • High Protection Spray SPF 50+
    Lotion • - • Topical • Canada • OTC • Approved
  • iUNIK Centella Calming Daily Sunscreen
    Cream • - • Topical • US • OTC
Menampilkan 8 dari 26 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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