Peringatan Keamanan

The EU has published a statement of caution that antiperspirant should not be applied to damaged or irritated skin, yet it is common to shave the underarm area before applying antiperspirant F48.

The possible health risks of aluminum containing antiperspirant use are not well studied. Although it has been suggested that deodorant and/or antiperspirant use is associated with incidence or age of breast cancer diagnosis A32464, a causal relationship between aluminium product use and breast cancer has not been established A32967, A32971.

The oral toxicity of aluminium compounds for which data are available (bromide, nitrate, chloride and sulfate) is moderate to low, with LD50 values in the range of 162 to 750 mg Al/kg in rats, and from 164 to 980 mg Al/kg in mice, depending on the type of aluminium compound studied F48.

Aluminum zirconium octachlorohydrex gly

DB11200

small molecule approved

Deskripsi

Aluminum zirconium octachlorohydrex gly is complex that consists of aluminum zirconium octachlorohydrate and glycine. It is an active antiperspirant agent L2705, L2706. It diffuses into the sweat pores and prevents perspiration (sweat) from leaving the pores. The anhydrous form of the compound also has water-absorbing properties. Currently, the FDA allows the inclusion of this substance in concentrations of up to 20% in antiperspirants L2012.

Interestingly, this chemical has been studied in relation to its possible impact on the microbiome of the human underarms A32967.

Struktur Molekul 2D

Berat 263.74
Wujud -

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

A preliminary study of the dermal absorption of aluminium from antiperspirants using aluminum-26 was performed. After repeated exposure for 6 days to aluminum chlorohydrate 21 % (about 13 mg of aluminium) to each axilla under occlusive dressing in two volunteers (one man and a woman), on skin previously tape stripped twice, blood and urine samples were obtained. Aluminium was detected in the blood 6 hours after the primary application and remained detectable for 15 days therafter. The results of this study estimate that the proportion of aluminium is absorbed averaged 0.012%. The shortcomings of this study are that it was not done in accordance with good practice (GCP) and it was performed using only 2 volunteers L2703.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

0 Data
Tidak ada data.

Target Protein

Sweat ducts

Referensi & Sumber

Artikel (PubMed)
  • PMID: 7673497
    Reynolds K, Darrigrand A, Roberts D, Knapik J, Pollard J, Duplantis K, Jones B: Effects of an antiperspirant with emollients on foot-sweat accumulation and blister formation while walking in the heat. J Am Acad Dermatol. 1995 Oct;33(4):626-30.
  • PMID: 26855863
    Urban J, Fergus DJ, Savage AM, Ehlers M, Menninger HL, Dunn RR, Horvath JE: The effect of habitual and experimental antiperspirant and deodorant product use on the armpit microbiome. PeerJ. 2016 Feb 2;4:e1605. doi: 10.7717/peerj.1605. eCollection 2016.
  • PMID: 16045991
    Darbre PD: Aluminium, antiperspirants and breast cancer. J Inorg Biochem. 2005 Sep;99(9):1912-9. doi: 10.1016/j.jinorgbio.2005.06.001.
  • PMID: 27755864
    Allam MF: Breast Cancer and Deodorants/Antiperspirants: a Systematic Review. Cent Eur J Public Health. 2016 Sep;24(3):245-247. doi: 10.21101/cejph.a4475.

Contoh Produk & Brand

Produk: 1654 • International brands: 0
Produk
  • 24 Hour High Performance Antiperspirant
    Stick • 18.6 mL/100mL • Topical • US • OTC
  • 5 Day
    Liquid • 20 g/100mL • Topical • US • OTC
  • Active Antiperspirant and Deodorant for Men
    Cream • 17.8 g/100g • Topical • US • OTC
  • Adidas 24H Anti Perspirant Deep Energy 2.8
    Stick • 12.6 g/79g • Topical • US • OTC
  • Adidas 24H Anti Perspirant Dynamic Pulse 2.8
    Stick • 12.6 g/79g • Topical • US • OTC
  • Adidas 24H Anti Perspirant Pure Game 2.8
    Stick • 12.6 g/79g • Topical • US • OTC
  • Adidas Action 3 Control
    Stick • 14.2 g/79g • Topical • US • OTC
  • Adidas Action 3 Fresh
    Stick • 18 mg/100g • Topical • US • OTC
Menampilkan 8 dari 1654 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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