Peringatan Keamanan

Highest dose tested was 360mg/kg/day in rats resulted in transient limb swelling.

Antithrombin Alfa

DB11166

biotech approved investigational

Deskripsi

Antithrombin Alfa is a recombinant antithrombin , an anticoagulant, that is used for the prevention of thromboembolic events in patients that have hereditary deficiency of antithrombin in high risk situations.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Dose of: 50IU/kg: 11.6 h 100IU/kg: 17.7 h
Volume Distribusi Dose of: 50IU/kg: 126.2 ml/kg 100IU/kg: 156.1 ml/kg Vd in hereditary deficient pregnant women in high risk situations had increased Vd of 14.3L.
Klirens (Clearance) Dose of: 50IU/kg: 9.6 ml/hr/kg 100IU/kg: 7.2 ml/hr/kg Cl in hereditary deficient pregnant women in high risk situations had increased Cl of 1.38L/h.

Absorpsi

Given IV so not absorbed.

Metabolisme

Not metabolized.

Rute Eliminasi

Irreversible complexes formed between antithrombin III and its target protease are rapidly removed by the liver.

Interaksi Makanan

1 Data
  • 1. Avoid herbs and supplements with anticoagulant/antiplatelet activity. Examples include garlic, ginger, bilberry, danshen, piracetam, and ginkgo biloba.

Interaksi Obat

640 Data
Apixaban Apixaban may increase the anticoagulant activities of Antithrombin Alfa.
Dabigatran etexilate Dabigatran etexilate may increase the anticoagulant activities of Antithrombin Alfa.
Dasatinib The risk or severity of bleeding and hemorrhage can be increased when Dasatinib is combined with Antithrombin Alfa.
Deferasirox The risk or severity of gastrointestinal bleeding can be increased when Antithrombin Alfa is combined with Deferasirox.
Ursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Cholic Acid.
Glycocholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Taurocholic acid.
Obeticholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Antithrombin Alfa is combined with Hyodeoxycholic Acid.
Edoxaban The risk or severity of bleeding can be increased when Edoxaban is combined with Antithrombin Alfa.
Ibrutinib The risk or severity of bleeding and hemorrhage can be increased when Ibrutinib is combined with Antithrombin Alfa.
Obinutuzumab The risk or severity of bleeding and hemorrhage can be increased when Antithrombin Alfa is combined with Obinutuzumab.
Rivaroxaban Antithrombin Alfa may increase the anticoagulant activities of Rivaroxaban.
Sugammadex The risk or severity of bleeding and hemorrhage can be increased when Antithrombin Alfa is combined with Sugammadex.
Tibolone Tibolone may increase the anticoagulant activities of Antithrombin Alfa.
Tipranavir The risk or severity of bleeding and hemorrhage can be increased when Tipranavir is combined with Antithrombin Alfa.
Urokinase Urokinase may increase the anticoagulant activities of Antithrombin Alfa.
Vitamin E Vitamin E may increase the anticoagulant activities of Antithrombin Alfa.
Vorapaxar The risk or severity of bleeding and hemorrhage can be increased when Vorapaxar is combined with Antithrombin Alfa.
Ginkgo biloba Ginkgo biloba may increase the anticoagulant activities of Antithrombin Alfa.
Ifosfamide The risk or severity of bleeding can be increased when Ifosfamide is combined with Antithrombin Alfa.
Quinine The therapeutic efficacy of Antithrombin Alfa can be increased when used in combination with Quinine.
Quinidine The therapeutic efficacy of Antithrombin Alfa can be increased when used in combination with Quinidine.
Tamoxifen The risk or severity of bleeding can be increased when Tamoxifen is combined with Antithrombin Alfa.
Toremifene The risk or severity of bleeding can be increased when Toremifene is combined with Antithrombin Alfa.
Pentoxifylline The therapeutic efficacy of Antithrombin Alfa can be increased when used in combination with Pentoxifylline.
Pentosan polysulfate Pentosan polysulfate may increase the anticoagulant activities of Antithrombin Alfa.
Levocarnitine The therapeutic efficacy of Antithrombin Alfa can be increased when used in combination with Levocarnitine.
Diethylstilbestrol Diethylstilbestrol may decrease the anticoagulant activities of Antithrombin Alfa.
Chlorotrianisene Chlorotrianisene may decrease the anticoagulant activities of Antithrombin Alfa.
Conjugated estrogens Conjugated estrogens may decrease the anticoagulant activities of Antithrombin Alfa.
Mestranol The risk or severity of adverse effects can be increased when Mestranol is combined with Antithrombin Alfa.
Estrone sulfate Estrone sulfate may decrease the anticoagulant activities of Antithrombin Alfa.
Quinestrol Quinestrol may decrease the anticoagulant activities of Antithrombin Alfa.
Hexestrol Hexestrol may decrease the anticoagulant activities of Antithrombin Alfa.
Synthetic Conjugated Estrogens, A Synthetic Conjugated Estrogens, A may decrease the anticoagulant activities of Antithrombin Alfa.
Synthetic Conjugated Estrogens, B Synthetic Conjugated Estrogens, B may decrease the anticoagulant activities of Antithrombin Alfa.
Polyestradiol phosphate Polyestradiol phosphate may decrease the anticoagulant activities of Antithrombin Alfa.
Esterified estrogens Esterified estrogens may decrease the anticoagulant activities of Antithrombin Alfa.
Zeranol Zeranol may decrease the anticoagulant activities of Antithrombin Alfa.
Equol Equol may decrease the anticoagulant activities of Antithrombin Alfa.
Methallenestril Methallenestril may decrease the anticoagulant activities of Antithrombin Alfa.
Epimestrol Epimestrol may decrease the anticoagulant activities of Antithrombin Alfa.
Moxestrol Moxestrol may decrease the anticoagulant activities of Antithrombin Alfa.
Estradiol acetate Estradiol acetate may decrease the anticoagulant activities of Antithrombin Alfa.
Estradiol benzoate Estradiol benzoate may decrease the anticoagulant activities of Antithrombin Alfa.
Estradiol cypionate Estradiol cypionate may decrease the anticoagulant activities of Antithrombin Alfa.
Estradiol valerate Estradiol valerate may decrease the anticoagulant activities of Antithrombin Alfa.
Biochanin A Biochanin A may decrease the anticoagulant activities of Antithrombin Alfa.
Formononetin Formononetin may decrease the anticoagulant activities of Antithrombin Alfa.
Estriol Estriol may decrease the anticoagulant activities of Antithrombin Alfa.
Limaprost The risk or severity of adverse effects can be increased when Limaprost is combined with Antithrombin Alfa.
Icosapent The risk or severity of bleeding and hemorrhage can be increased when Icosapent is combined with Antithrombin Alfa.
Mesalazine The risk or severity of bleeding can be increased when Mesalazine is combined with Antithrombin Alfa.
Indomethacin The risk or severity of bleeding and hemorrhage can be increased when Indomethacin is combined with Antithrombin Alfa.
Nabumetone The risk or severity of bleeding and hemorrhage can be increased when Nabumetone is combined with Antithrombin Alfa.
Ketorolac The risk or severity of bleeding and hemorrhage can be increased when Ketorolac is combined with Antithrombin Alfa.
Tenoxicam The risk or severity of bleeding and hemorrhage can be increased when Tenoxicam is combined with Antithrombin Alfa.
Celecoxib The risk or severity of bleeding and hemorrhage can be increased when Celecoxib is combined with Antithrombin Alfa.
Tolmetin The risk or severity of bleeding and hemorrhage can be increased when Tolmetin is combined with Antithrombin Alfa.
Rofecoxib The risk or severity of bleeding and hemorrhage can be increased when Rofecoxib is combined with Antithrombin Alfa.
Piroxicam The risk or severity of bleeding and hemorrhage can be increased when Piroxicam is combined with Antithrombin Alfa.
Fenoprofen The risk or severity of bleeding and hemorrhage can be increased when Fenoprofen is combined with Antithrombin Alfa.
Valdecoxib The risk or severity of bleeding and hemorrhage can be increased when Valdecoxib is combined with Antithrombin Alfa.
Diclofenac The risk or severity of bleeding and hemorrhage can be increased when Diclofenac is combined with Antithrombin Alfa.
Sulindac The risk or severity of bleeding and hemorrhage can be increased when Sulindac is combined with Antithrombin Alfa.
Flurbiprofen The risk or severity of bleeding and hemorrhage can be increased when Flurbiprofen is combined with Antithrombin Alfa.
Etodolac The risk or severity of bleeding and hemorrhage can be increased when Etodolac is combined with Antithrombin Alfa.
Mefenamic acid The risk or severity of bleeding and hemorrhage can be increased when Mefenamic acid is combined with Antithrombin Alfa.
Naproxen The risk or severity of bleeding and hemorrhage can be increased when Naproxen is combined with Antithrombin Alfa.
Sulfasalazine The risk or severity of bleeding and hemorrhage can be increased when Sulfasalazine is combined with Antithrombin Alfa.
Phenylbutazone The risk or severity of bleeding and hemorrhage can be increased when Phenylbutazone is combined with Antithrombin Alfa.
Meloxicam The risk or severity of bleeding and hemorrhage can be increased when Meloxicam is combined with Antithrombin Alfa.
Carprofen The risk or severity of bleeding and hemorrhage can be increased when Carprofen is combined with Antithrombin Alfa.
Diflunisal The risk or severity of bleeding and hemorrhage can be increased when Diflunisal is combined with Antithrombin Alfa.
Salicylic acid The risk or severity of bleeding and hemorrhage can be increased when Salicylic acid is combined with Antithrombin Alfa.
Meclofenamic acid The risk or severity of bleeding and hemorrhage can be increased when Meclofenamic acid is combined with Antithrombin Alfa.
Oxaprozin The risk or severity of bleeding and hemorrhage can be increased when Oxaprozin is combined with Antithrombin Alfa.
Ketoprofen The risk or severity of bleeding and hemorrhage can be increased when Ketoprofen is combined with Antithrombin Alfa.
Balsalazide The risk or severity of bleeding and hemorrhage can be increased when Balsalazide is combined with Antithrombin Alfa.
Olsalazine The risk or severity of bleeding can be increased when Olsalazine is combined with Antithrombin Alfa.
Lumiracoxib The risk or severity of bleeding and hemorrhage can be increased when Lumiracoxib is combined with Antithrombin Alfa.
Magnesium salicylate The risk or severity of bleeding and hemorrhage can be increased when Magnesium salicylate is combined with Antithrombin Alfa.
Salsalate The risk or severity of bleeding and hemorrhage can be increased when Salsalate is combined with Antithrombin Alfa.
Choline magnesium trisalicylate The risk or severity of bleeding and hemorrhage can be increased when Choline magnesium trisalicylate is combined with Antithrombin Alfa.
Antrafenine The risk or severity of bleeding and hemorrhage can be increased when Antrafenine is combined with Antithrombin Alfa.
Aminophenazone The risk or severity of bleeding and hemorrhage can be increased when Aminophenazone is combined with Antithrombin Alfa.
Antipyrine The risk or severity of bleeding and hemorrhage can be increased when Antipyrine is combined with Antithrombin Alfa.
Tiaprofenic acid The risk or severity of bleeding and hemorrhage can be increased when Tiaprofenic acid is combined with Antithrombin Alfa.
Etoricoxib The risk or severity of bleeding and hemorrhage can be increased when Etoricoxib is combined with Antithrombin Alfa.
Taxifolin The risk or severity of bleeding and hemorrhage can be increased when Taxifolin is combined with Antithrombin Alfa.
Oxyphenbutazone The risk or severity of bleeding and hemorrhage can be increased when Oxyphenbutazone is combined with Antithrombin Alfa.

Target Protein

Prothrombin F2
Coagulation factor X F10

Referensi & Sumber

Artikel (PubMed)
  • PMID: 19141163
    Patnaik MM, Moll S: Inherited antithrombin deficiency: a review. Haemophilia. 2008 Nov;14(6):1229-39. doi: 10.1111/j.1365-2516.2008.01830.x.

Contoh Produk & Brand

Produk: 6 • International brands: 0
Produk
  • Atryn
    Injection, powder, lyophilized, for solution • 1750 [iU]/10mL • Intravenous • US • Approved
  • ATryn
    Injection, powder, lyophilized, for solution • 525 [iU]/1mL • Intravenous • US • Approved
  • ATryn
    Injection, powder, lyophilized, for solution • 1750 [iU]/1mL • Intravenous • US • Approved
  • Atryn
    Injection, powder, for solution • 1750 IU • Intravenous • EU
  • Atryn
    Injection, powder, for solution • 1750 IU • Intravenous • EU
  • Atryn
    Injection, powder, for solution • 1750 IU • Intravenous • EU

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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