Peringatan Keamanan

Oral LD50 of racepinephrine hydrochloride in mouse is 90 mg/kg MSDS.

Overdosage of epinephrine may cause extremely elevated arterial pressure, which may further lead to cerebrovascular hemorrhage, particularly in elderly patients. Peripheral vascular constriction in conjunction with cardiac stimulation may produce pulmonary oedema. Treatment consists of rapidly acting vasodilators or alpha-adrenergic blocking drugs and/or respiratory support. Transient bradycardia followed by tachycardia may also be observed, and may be accompanied by potentially fatal cardiac arrhythmias. remature ventricular contractions may appear within one minute after injection and may be followed by multifocal ventricular tachycardia (prefibrillation rhythm). Subsidence of the ventricular effects may be followed by atrial tachycardia and occasionally by atrioventricular block. In case of arrhythmias, treatment should involve administration of a beta­ adrenergic blocking drug such as propranolol. Overdosage may also produce extreme pallor and coldness of the skin, metabolic acidosis, and kidney failure, which should each be treated with suitable corrective measures FDA Label.

Racepinephrine

DB11124

small molecule approved

Deskripsi

Racepinephrine is a racemic mixture consisting of d-DB00668 and l-DB00668 enantiomers. Epinephrine is a non-selective ?- and ?-adrenergic receptor agonist. It is a bronchodilator used in the temporary relief of mild symptoms of intermittent asthma including wheezing, tightness of chest and shortness of breath. It is an active ingredient in oral inhalation over-the-counter products as racepinephrine hydrochloride.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for [DB00668].
Volume Distribusi To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for [DB00668].
Klirens (Clearance) To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for [DB00668].

Absorpsi

To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for DB00668.

Metabolisme

To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for DB00668.

Rute Eliminasi

To refer to the pharmacokinetic data of L-epinephrine, refer to the drug entry for DB00668.

Interaksi Makanan

1 Data
  • 1. Avoid caffeine.

Interaksi Obat

921 Data
Valsartan Racepinephrine may decrease the antihypertensive activities of Valsartan.
Ramipril Racepinephrine may decrease the antihypertensive activities of Ramipril.
Reserpine Racepinephrine may decrease the antihypertensive activities of Reserpine.
Remikiren Racepinephrine may decrease the antihypertensive activities of Remikiren.
Isradipine Racepinephrine may decrease the antihypertensive activities of Isradipine.
Olmesartan Racepinephrine may decrease the antihypertensive activities of Olmesartan.
Nitroprusside Racepinephrine may decrease the antihypertensive activities of Nitroprusside.
Diltiazem Racepinephrine may decrease the antihypertensive activities of Diltiazem.
Minoxidil Racepinephrine may decrease the antihypertensive activities of Minoxidil.
Treprostinil Racepinephrine may decrease the antihypertensive activities of Treprostinil.
Amlodipine Racepinephrine may decrease the antihypertensive activities of Amlodipine.
Nimodipine Racepinephrine may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Racepinephrine may decrease the antihypertensive activities of Nisoldipine.
Fosinopril Racepinephrine may decrease the antihypertensive activities of Fosinopril.
Trandolapril Racepinephrine may decrease the antihypertensive activities of Trandolapril.
Lercanidipine Racepinephrine may decrease the antihypertensive activities of Lercanidipine.
Benazepril Racepinephrine may decrease the antihypertensive activities of Benazepril.
Bosentan Racepinephrine may decrease the antihypertensive activities of Bosentan.
Enalapril Racepinephrine may decrease the antihypertensive activities of Enalapril.
Candoxatril Racepinephrine may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Racepinephrine may decrease the antihypertensive activities of Mecamylamine.
Losartan Racepinephrine may decrease the antihypertensive activities of Losartan.
Moexipril Racepinephrine may decrease the antihypertensive activities of Moexipril.
Lisinopril Racepinephrine may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Racepinephrine may decrease the antihypertensive activities of Nitroglycerin.
Metyrosine Racepinephrine may decrease the antihypertensive activities of Metyrosine.
Cryptenamine Racepinephrine may decrease the antihypertensive activities of Cryptenamine.
Perindopril Racepinephrine may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Racepinephrine may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Racepinephrine may decrease the antihypertensive activities of Fenoldopam.
Tadalafil Racepinephrine may decrease the antihypertensive activities of Tadalafil.
Eprosartan Racepinephrine may decrease the antihypertensive activities of Eprosartan.
Quinapril Racepinephrine may decrease the antihypertensive activities of Quinapril.
Telmisartan Racepinephrine may decrease the antihypertensive activities of Telmisartan.
Methyldopa Racepinephrine may decrease the antihypertensive activities of Methyldopa.
Irbesartan Racepinephrine may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Racepinephrine may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Racepinephrine may decrease the antihypertensive activities of Deserpidine.
Pentolinium Racepinephrine may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Racepinephrine may decrease the antihypertensive activities of Trimethaphan.
Captopril Racepinephrine may decrease the antihypertensive activities of Captopril.
Epoprostenol Racepinephrine may decrease the antihypertensive activities of Epoprostenol.
Bepridil Racepinephrine may decrease the antihypertensive activities of Bepridil.
Hydralazine Racepinephrine may decrease the antihypertensive activities of Hydralazine.
Cilazapril Racepinephrine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Racepinephrine may decrease the antihypertensive activities of Saprisartan.
Spirapril Racepinephrine may decrease the antihypertensive activities of Spirapril.
Mibefradil Racepinephrine may decrease the antihypertensive activities of Mibefradil.
Debrisoquine Racepinephrine may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Racepinephrine may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Racepinephrine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Racepinephrine may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Racepinephrine may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Racepinephrine may decrease the antihypertensive activities of Pinacidil.
Temocapril Racepinephrine may decrease the antihypertensive activities of Temocapril.
Riociguat Racepinephrine may decrease the antihypertensive activities of Riociguat.
Macitentan Racepinephrine may decrease the antihypertensive activities of Macitentan.
Hexamethonium Racepinephrine may decrease the antihypertensive activities of Hexamethonium.
Aliskiren Racepinephrine may decrease the antihypertensive activities of Aliskiren.
Nicorandil Racepinephrine may decrease the antihypertensive activities of Nicorandil.
Lacidipine Racepinephrine may decrease the antihypertensive activities of Lacidipine.
Manidipine Racepinephrine may decrease the antihypertensive activities of Manidipine.
Rauwolfia serpentina root Racepinephrine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Racepinephrine may decrease the antihypertensive activities of Enalaprilat.
Selexipag Racepinephrine may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Racepinephrine may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Racepinephrine may decrease the antihypertensive activities of Imidapril.
BQ-123 Racepinephrine may decrease the antihypertensive activities of BQ-123.
Tetrahydropalmatine Racepinephrine may decrease the antihypertensive activities of Tetrahydropalmatine.
Dihydralazine Racepinephrine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Racepinephrine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Racepinephrine may decrease the antihypertensive activities of Guanoxan.
Delapril Racepinephrine may decrease the antihypertensive activities of Delapril.
Vincamine Racepinephrine may decrease the antihypertensive activities of Vincamine.
Linsidomine Racepinephrine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Racepinephrine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Racepinephrine may decrease the antihypertensive activities of Tolonidine.
Endralazine Racepinephrine may decrease the antihypertensive activities of Endralazine.
Cadralazine Racepinephrine may decrease the antihypertensive activities of Cadralazine.
Bietaserpine Racepinephrine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Racepinephrine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Racepinephrine may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Racepinephrine may decrease the antihypertensive activities of Guanoclor.
Candesartan Racepinephrine may decrease the antihypertensive activities of Candesartan.
Dexniguldipine Racepinephrine may decrease the antihypertensive activities of Dexniguldipine.
Tocopherylquinone Racepinephrine may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Racepinephrine may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Racepinephrine may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Racepinephrine may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Racepinephrine may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Racepinephrine may decrease the antihypertensive activities of Quinaprilat.
Felodipine Racepinephrine may decrease the antihypertensive activities of Felodipine.
Levamlodipine Racepinephrine may decrease the antihypertensive activities of Levamlodipine.
Azilsartan medoxomil Racepinephrine may decrease the antihypertensive activities of Azilsartan medoxomil.
Diazoxide Racepinephrine may decrease the antihypertensive activities of Diazoxide.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Racepinephrine.
Benzylpenicilloyl polylysine Racepinephrine may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Desmopressin The risk or severity of hypertension can be increased when Desmopressin is combined with Racepinephrine.
Cyclosporine The risk or severity of hypertension can be increased when Cyclosporine is combined with Racepinephrine.
Icosapent The risk or severity of hypertension can be increased when Icosapent is combined with Racepinephrine.

Target Protein

Alpha-1A adrenergic receptor ADRA1A
Alpha-1B adrenergic receptor ADRA1B
Alpha-2A adrenergic receptor ADRA2A
Alpha-2B adrenergic receptor ADRA2B
Alpha-2C adrenergic receptor ADRA2C
Alpha-1D adrenergic receptor ADRA1D
Beta-1 adrenergic receptor ADRB1
Beta-2 adrenergic receptor ADRB2
Beta-3 adrenergic receptor ADRB3

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15876347
    Langley JM, Smith MB, LeBlanc JC, Joudrey H, Ojah CR, Pianosi P: Racemic epinephrine compared to salbutamol in hospitalized young children with bronchiolitis; a randomized controlled clinical trial ISRCTN46561076. BMC Pediatr. 2005 May 5;5(1):7. doi: 10.1186/1471-2431-5-7.
  • PMID: 7767427
    Reijonen T, Korppi M, Pitkakangas S, Tenhola S, Remes K: The clinical efficacy of nebulized racemic epinephrine and albuterol in acute bronchiolitis. Arch Pediatr Adolesc Med. 1995 Jun;149(6):686-92.
Textbook
  • ISBN: 978-0-7020-3471-8
    14. (2012). In Rang and Dale's Pharmacology (7th ed., pp. 174-175, 181-182). Edinburgh: Elsevier/Churchill Livingstone.

Contoh Produk & Brand

Produk: 50 • International brands: 0
Produk
  • Asthmanefrin
    Solution • 11.25 mg/0.5mL • Respiratory (inhalation) • US • OTC
  • Blue Gel Anesthetic
    Gel • - • Topical • US • OTC
  • Cord No2 Gingival Retraction
    Packing • 0.5 mg / 2.54 cm • Dental • Canada • Approved
  • Cord No3
    Packing • 0.5 mg / 2.54 cm • Dental • Canada • Approved
  • Cotton Coil
    Packing • 3 mg / 2.54 cm • Dental • Canada • Approved
  • Crown Pak Retraction Cord
    Packing • 0.5 mg / 2.54 cm • Dental • Canada • Approved
  • Epi-Mist
    Aerosol, spray • .594 mg/.120mL • Respiratory (inhalation) • US • OTC
  • Epidri 6%
    - • 2.1 mg • Dental • Canada • Approved
Menampilkan 8 dari 50 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul