Isosorbide

DB09401

small molecule approved investigational

Deskripsi

Isosorbide was previously available in an oral formulation for the reduction of intraocular pressure. It was approved by the FDA in 1980, but has since been discontinued. Currently, isosorbide is an organic nitrate currently available in the isosorbide mononitrate and isosorbide dinitrate forms, and is used for the prevention of angina. Refer to these drug entries for more information.

Struktur Molekul 2D

Berat 146.1412
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Isosorbide is rapidly absorbed after oral administration.L34064 Refer to isosorbide mononitrate for detailed absorption information.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

712 Data
Dapoxetine Dapoxetine may increase the orthostatic hypotensive and hypotensive activities of Isosorbide.
Riociguat Isosorbide may increase the hypotensive activities of Riociguat.
Rosiglitazone The risk or severity of adverse effects can be increased when Isosorbide is combined with Rosiglitazone.
Molsidomine Molsidomine may increase the hypotensive activities of Isosorbide.
Tadalafil The risk or severity of hypotension can be increased when Tadalafil is combined with Isosorbide.
Vardenafil The risk or severity of hypotension can be increased when Vardenafil is combined with Isosorbide.
Dipyridamole The risk or severity of hypotension can be increased when Dipyridamole is combined with Isosorbide.
Ibudilast The risk or severity of hypotension can be increased when Ibudilast is combined with Isosorbide.
Avanafil Avanafil may increase the hypotensive activities of Isosorbide.
Udenafil The risk or severity of hypotension can be increased when Udenafil is combined with Isosorbide.
Doxofylline The risk or severity of hypotension can be increased when Doxofylline is combined with Isosorbide.
Mirodenafil The risk or severity of hypotension can be increased when Mirodenafil is combined with Isosorbide.
Fostamatinib The risk or severity of hypotension can be increased when Fostamatinib is combined with Isosorbide.
Ethanol Ethanol may increase the hypotensive and vasodilatory activities of Isosorbide.
Sodium phosphate, monobasic Isosorbide may increase the nephrotoxic activities of Sodium phosphate, monobasic.
Acemetacin The therapeutic efficacy of Isosorbide can be decreased when used in combination with Acemetacin.
Patent Blue The therapeutic efficacy of Isosorbide can be decreased when used in combination with Patent Blue.
Lactulose The risk or severity of dehydration can be increased when Isosorbide is combined with Lactulose.
Mannitol The risk or severity of dehydration can be increased when Isosorbide is combined with Mannitol.
Lubiprostone The risk or severity of dehydration can be increased when Isosorbide is combined with Lubiprostone.
Tegaserod The risk or severity of dehydration can be increased when Isosorbide is combined with Tegaserod.
Magnesium oxide The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium oxide.
Magnesium cation The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium cation.
Sorbitol The risk or severity of dehydration can be increased when Isosorbide is combined with Sorbitol.
Dantron The risk or severity of dehydration can be increased when Isosorbide is combined with Dantron.
Oxyphenisatin The risk or severity of dehydration can be increased when Isosorbide is combined with Oxyphenisatin.
Phenolphthalein The risk or severity of dehydration can be increased when Isosorbide is combined with Phenolphthalein.
Emodin The risk or severity of dehydration can be increased when Isosorbide is combined with Emodin.
Linaclotide The risk or severity of dehydration can be increased when Isosorbide is combined with Linaclotide.
Bisacodyl The risk or severity of dehydration can be increased when Isosorbide is combined with Bisacodyl.
Magnesium hydroxide The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium hydroxide.
Bisoxatin The risk or severity of dehydration can be increased when Isosorbide is combined with Bisoxatin.
Picosulfuric acid The risk or severity of dehydration can be increased when Isosorbide is combined with Picosulfuric acid.
Magnesium trisilicate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium trisilicate.
Polyethylene glycol The risk or severity of dehydration can be increased when Isosorbide is combined with Polyethylene glycol.
Polycarbophil The risk or severity of dehydration can be increased when Isosorbide is combined with Polycarbophil.
Magnesium acetate tetrahydrate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium acetate tetrahydrate.
Monopotassium phosphate The risk or severity of dehydration can be increased when Isosorbide is combined with Monopotassium phosphate.
Dipotassium phosphate The risk or severity of dehydration can be increased when Isosorbide is combined with Dipotassium phosphate.
Glycerin The risk or severity of dehydration can be increased when Isosorbide is combined with Glycerin.
Sodium sulfate The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium sulfate.
Magnesium carbonate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium carbonate.
Potassium lactate The risk or severity of dehydration can be increased when Isosorbide is combined with Potassium lactate.
Sodium fluorophosphate The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium fluorophosphate.
Mineral oil The risk or severity of dehydration can be increased when Isosorbide is combined with Mineral oil.
Carboxymethylcellulose The risk or severity of dehydration can be increased when Isosorbide is combined with Carboxymethylcellulose.
Docusate The risk or severity of dehydration can be increased when Isosorbide is combined with Docusate.
Plantago seed The risk or severity of dehydration can be increased when Isosorbide is combined with Plantago seed.
Magnesium citrate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium citrate.
Castor oil The risk or severity of dehydration can be increased when Isosorbide is combined with Castor oil.
Magnesium glycinate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium glycinate.
Methylcellulose The risk or severity of dehydration can be increased when Isosorbide is combined with Methylcellulose.
Sennosides The risk or severity of dehydration can be increased when Isosorbide is combined with Sennosides.
Lactitol The risk or severity of dehydration can be increased when Isosorbide is combined with Lactitol.
Plecanatide The risk or severity of dehydration can be increased when Isosorbide is combined with Plecanatide.
Gluconic Acid The risk or severity of dehydration can be increased when Isosorbide is combined with Gluconic Acid.
Magnesium peroxide The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium peroxide.
Pentaerithrityl The risk or severity of dehydration can be increased when Isosorbide is combined with Pentaerithrityl.
Sodium tartrate The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium tartrate.
Magnesium acetate The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium acetate.
Deacetylbisacodyl The risk or severity of dehydration can be increased when Isosorbide is combined with Deacetylbisacodyl.
Sodium ascorbate The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium ascorbate.
Potassium sulfate The risk or severity of dehydration can be increased when Isosorbide is combined with Potassium sulfate.
Sodium phosphate, dibasic The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium phosphate, dibasic.
Sodium phosphate, monobasic, unspecified form The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium phosphate, monobasic, unspecified form.
Sodium phosphate, dibasic, unspecified form The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium phosphate, dibasic, unspecified form.
Magnesium The risk or severity of dehydration can be increased when Isosorbide is combined with Magnesium.
Sodium cation The risk or severity of dehydration can be increased when Isosorbide is combined with Sodium cation.
Plantago ovata seed The risk or severity of dehydration can be increased when Isosorbide is combined with Plantago ovata seed.
Oxyphenisatin acetate The risk or severity of dehydration can be increased when Isosorbide is combined with Oxyphenisatin acetate.
Calcium polycarbophil The risk or severity of dehydration can be increased when Isosorbide is combined with Calcium polycarbophil.
Konjac mannan The risk or severity of dehydration can be increased when Isosorbide is combined with Konjac mannan.
Alloin The risk or severity of dehydration can be increased when Isosorbide is combined with Alloin.
Frangula purshiana bark The risk or severity of dehydration can be increased when Isosorbide is combined with Frangula purshiana bark.
Dehydrocholic acid The risk or severity of dehydration can be increased when Isosorbide is combined with Dehydrocholic acid.
Sulfate ion The risk or severity of dehydration can be increased when Isosorbide is combined with Sulfate ion.
Piperacillin Isosorbide may increase the excretion rate of Piperacillin which could result in a lower serum level and potentially a reduction in efficacy.
Ampicillin Isosorbide may increase the excretion rate of Ampicillin which could result in a lower serum level and potentially a reduction in efficacy.
Oxacillin Isosorbide may increase the excretion rate of Oxacillin which could result in a lower serum level and potentially a reduction in efficacy.
Amoxicillin Isosorbide may increase the excretion rate of Amoxicillin which could result in a lower serum level and potentially a reduction in efficacy.
Procaine benzylpenicillin Isosorbide may increase the excretion rate of Procaine benzylpenicillin which could result in a lower serum level and potentially a reduction in efficacy.
Prucalopride The risk or severity of dehydration can be increased when Isosorbide is combined with Prucalopride.
Diflunisal Isosorbide may increase the excretion rate of Diflunisal which could result in a lower serum level and potentially a reduction in efficacy.
Ibuprofen Isosorbide may increase the excretion rate of Ibuprofen which could result in a lower serum level and potentially a reduction in efficacy.
Naloxone Isosorbide may increase the excretion rate of Naloxone which could result in a lower serum level and potentially a reduction in efficacy.
Dexketoprofen Isosorbide may increase the excretion rate of Dexketoprofen which could result in a lower serum level and potentially a reduction in efficacy.
Leuprolide Isosorbide may increase the excretion rate of Leuprolide which could result in a lower serum level and potentially a reduction in efficacy.
Goserelin Isosorbide may increase the excretion rate of Goserelin which could result in a lower serum level and potentially a reduction in efficacy.
Salmon calcitonin Isosorbide may increase the excretion rate of Salmon calcitonin which could result in a lower serum level and potentially a reduction in efficacy.
Desmopressin Isosorbide may increase the excretion rate of Desmopressin which could result in a lower serum level and potentially a reduction in efficacy.
Aldesleukin Isosorbide may increase the excretion rate of Aldesleukin which could result in a lower serum level and potentially a reduction in efficacy.
Daptomycin Isosorbide may increase the excretion rate of Daptomycin which could result in a lower serum level and potentially a reduction in efficacy.
Tositumomab Isosorbide may increase the excretion rate of Tositumomab which could result in a lower serum level and potentially a reduction in efficacy.
Cyanocobalamin Isosorbide may increase the excretion rate of Cyanocobalamin which could result in a lower serum level and potentially a reduction in efficacy.
Folic acid Isosorbide may increase the excretion rate of Folic acid which could result in a lower serum level and potentially a reduction in efficacy.
Pyridoxine Isosorbide may increase the excretion rate of Pyridoxine which could result in a lower serum level and potentially a reduction in efficacy.
Fluvoxamine Isosorbide may increase the excretion rate of Fluvoxamine which could result in a lower serum level and potentially a reduction in efficacy.
Baclofen Isosorbide may increase the excretion rate of Baclofen which could result in a lower serum level and potentially a reduction in efficacy.
Amphetamine Isosorbide may increase the excretion rate of Amphetamine which could result in a lower serum level and potentially a reduction in efficacy.
Cevimeline Isosorbide may increase the excretion rate of Cevimeline which could result in a lower serum level and potentially a reduction in efficacy.

Target Protein

Guanylate cyclase GUCY1A1

Referensi & Sumber

Synthesis reference: Bonnin, I., Mereau, R., Tassaing, T., & De Oliveira Vigier, K. (2020). One-pot synthesis of isosorbide from cellulose or lignocellulosic biomass: a challenge?. Beilstein journal of organic chemistry, 16, 1713–1721. https://doi.org/10.3762/bjoc.16.143
Artikel (PubMed)
  • PMID: 32491771
    Balasubramanian S, Chowdhury YS: Isosorbide .
  • PMID: 31424733
    Lee PM, Gerriets V: Nitrates .
  • PMID: 3300979
    Chasseaud LF: Isosorbide 5-mononitrate pharmacokinetics. Cardiology. 1987;74 Suppl 1:6-11. doi: 10.1159/000174255.
  • PMID: 2905390
    Romanin C, Kukovetz WR: Guanylate cyclase activation by organic nitrates is not mediated via nitrite. J Mol Cell Cardiol. 1988 May;20(5):389-96. doi: 10.1016/s0022-2828(88)80130-5.
  • PMID: 2895614
    Schroder H, Noack E: Structure-activity relationship of organic nitrates for activation of guanylate cyclase. Arch Int Pharmacodyn Ther. 1987 Dec;290(2):235-46.
  • PMID: 2886220
    Kukovetz WR, Holzmann S, Romanin C: Mechanism of vasodilation by nitrates: role of cyclic GMP. Cardiology. 1987;74 Suppl 1:12-9. doi: 10.1159/000174258.
  • PMID: -
    Kulshrestha O.P. and Mittal, R.N.: Isosorbide and intraocular pressure British Journal of Ophthalmology.
  • PMID: 9076203
    Hessemer V, Schmidt KG: Influence of the vasodilator drug isosorbide dinitrate on ocular circulation. Arch Ophthalmol. 1997 Mar;115(3):324-7. doi: 10.1001/archopht.1997.01100150326003.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Ismotic
    Solution • 450 mg/1mL • Oral • US • Approved

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