Peringatan Keamanan

LD50 Mouse ip 300 mg/kg, LD50 Mouse sc 750 mg/kg

Pramocaine

DB09345

small molecule approved

Deskripsi

Pramocaine (also known as pramoxine or pramoxine HCI) is a topical anesthetic and antipruritic. It is used for many dermatological and anorectal/anogenital conditions including minor cuts/burns, insect bites, hives/rashes due to poison ivy exposure, hemorrhoids and other anorectal/anogenital disorders. Pramocaine is available by itself and in combination with other medications in various topical preparations. It works by preventing ionic fluctuations needed for neuron membrane depolarization and action potential propagation.

Struktur Molekul 2D

Berat 293.407
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

There is minimal absorption after topical administration and it is not given orally.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1590 Data
Buprenorphine Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Hydrocodone Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Magnesium sulfate The therapeutic efficacy of Pramocaine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Pramocaine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Mirtazapine Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Orphenadrine Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Pramipexole Pramocaine may increase the sedative activities of Pramipexole.
Ropinirole Pramocaine may increase the sedative activities of Ropinirole.
Rotigotine Pramocaine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Pramocaine.
Sodium oxybate The risk or severity of CNS depression can be increased when Sodium oxybate is combined with Pramocaine.
Suvorexant Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Thalidomide Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Pramocaine.
Ethanol Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Pramocaine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Fluvoxamine The risk or severity of adverse effects can be increased when Pramocaine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Pramocaine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Pramocaine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Pramocaine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Pramocaine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Pramocaine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Pramocaine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Pramocaine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Pramocaine is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Pramocaine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Pramocaine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Pramocaine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Pramocaine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Pramocaine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Pramocaine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Pramocaine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Pramocaine is combined with Alaproclate.
Technetium Tc-99m tilmanocept Pramocaine may decrease effectiveness of Technetium Tc-99m tilmanocept as a diagnostic agent.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with Pramocaine.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Pramocaine.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with Pramocaine.
Promazine The risk or severity of CNS depression can be increased when Promazine is combined with Pramocaine.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Pramocaine.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with Pramocaine.
Chlorpromazine The risk or severity of CNS depression can be increased when Chlorpromazine is combined with Pramocaine.
Gallamine triethiodide The risk or severity of CNS depression can be increased when Gallamine triethiodide is combined with Pramocaine.
Triflupromazine The risk or severity of CNS depression can be increased when Triflupromazine is combined with Pramocaine.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with Pramocaine.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Pramocaine.
Lamotrigine The risk or severity of methemoglobinemia can be increased when Lamotrigine is combined with Pramocaine.
Rocuronium The risk or severity of CNS depression can be increased when Rocuronium is combined with Pramocaine.
Scopolamine The risk or severity of CNS depression can be increased when Scopolamine is combined with Pramocaine.
Clidinium The risk or severity of CNS depression can be increased when Clidinium is combined with Pramocaine.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Pramocaine.
Brompheniramine The risk or severity of CNS depression can be increased when Brompheniramine is combined with Pramocaine.
Flupentixol The risk or severity of CNS depression can be increased when Flupentixol is combined with Pramocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Cocaine is combined with Pramocaine.
Quinidine The risk or severity of methemoglobinemia can be increased when Quinidine is combined with Pramocaine.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with Pramocaine.
Promethazine The risk or severity of CNS depression can be increased when Promethazine is combined with Pramocaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Diphenhydramine is combined with Pramocaine.
Doxacurium The risk or severity of CNS depression can be increased when Doxacurium is combined with Pramocaine.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Pramocaine.
Desipramine The risk or severity of CNS depression can be increased when Desipramine is combined with Pramocaine.
Quetiapine The risk or severity of CNS depression can be increased when Quetiapine is combined with Pramocaine.
Mivacurium The risk or severity of CNS depression can be increased when Mivacurium is combined with Pramocaine.
Aripiprazole The risk or severity of CNS depression can be increased when Aripiprazole is combined with Pramocaine.
Chlorprothixene The risk or severity of CNS depression can be increased when Chlorprothixene is combined with Pramocaine.
Metocurine The risk or severity of CNS depression can be increased when Metocurine is combined with Pramocaine.
Pancuronium The risk or severity of CNS depression can be increased when Pancuronium is combined with Pramocaine.
Pipecuronium The risk or severity of CNS depression can be increased when Pipecuronium is combined with Pramocaine.
Rapacuronium The risk or severity of CNS depression can be increased when Rapacuronium is combined with Pramocaine.
Pizotifen The risk or severity of CNS depression can be increased when Pizotifen is combined with Pramocaine.
Benactyzine The risk or severity of CNS depression can be increased when Benactyzine is combined with Pramocaine.
Dosulepin The risk or severity of CNS depression can be increased when Dosulepin is combined with Pramocaine.
Emepronium The risk or severity of CNS depression can be increased when Pramocaine is combined with Emepronium.
Zopiclone The risk or severity of adverse effects can be increased when Pramocaine is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Pramocaine.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Pramocaine.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with Pramocaine.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Pramocaine.
Lorazepam The risk or severity of methemoglobinemia can be increased when Lorazepam is combined with Pramocaine.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Pramocaine.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Pramocaine.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with Pramocaine.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Pramocaine.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Pramocaine.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with Pramocaine.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with Pramocaine.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Pramocaine.
Butalbital The risk or severity of methemoglobinemia can be increased when Butalbital is combined with Pramocaine.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with Pramocaine.

Target Protein

Voltage-gated sodium channel alpha subunit SCN1A

Referensi & Sumber

Link

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