Peringatan Keamanan

The toxicity of this medication (7-8 times higher than that of procaine), has prevented this medication from being used on its own L1592.

Ester-type local anesthetics are much more likely to cause an allergic reaction compared to the amide-group local anesthetics because of the formation of PABA (Para-aminobenzoic acid) during the metabolic process. PABA may cause allergic reactions that range from urticaria to anaphylaxis. PABA is also formed during the metabolism of methylparaben (a common preservative) that is normally found in multi-dose vials including lidocaine (MDV) (amide-type local anesthetic) L1592, L1593.

Propoxycaine

DB09342

small molecule approved

Deskripsi

Propoxycaine is a local anesthetic of the ester type that has a rapid onset of action and a longer duration of action than procaine hydrochloride L1588. This drug was removed from the US market in 1996. Although no longer available in the United States, this medication was used in combination with procaine to aid in anesthesia during dental procedures L1592. Used in combination with procaine, it was the only dental local anesthetic available in cartridge form L1592.

Struktur Molekul 2D

Berat 294.395
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) Via the kidneys, primarily hydrolyzed [L1592].

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

This drug his hydrolyzed in both the plasma and the liver by plasma esterases L1593.

Rute Eliminasi

Renal L1592

Interaksi Obat

1043 Data
Hyaluronidase (ovine) Hyaluronidase (ovine) can cause an increase in the absorption of Propoxycaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase (human recombinant) Hyaluronidase (human recombinant) can cause an increase in the absorption of Propoxycaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase Hyaluronidase can cause an increase in the absorption of Propoxycaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Technetium Tc-99m tilmanocept Propoxycaine may decrease effectiveness of Technetium Tc-99m tilmanocept as a diagnostic agent.
Chloroprocaine The risk or severity of adverse effects can be increased when Propoxycaine is combined with Chloroprocaine.
Lidocaine The risk or severity of methemoglobinemia can be increased when Lidocaine is combined with Propoxycaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Ropivacaine is combined with Propoxycaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Bupivacaine is combined with Propoxycaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Cinchocaine is combined with Propoxycaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Dyclonine is combined with Propoxycaine.
Procaine The risk or severity of methemoglobinemia can be increased when Procaine is combined with Propoxycaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Prilocaine is combined with Propoxycaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Proparacaine is combined with Propoxycaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Meloxicam is combined with Propoxycaine.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Oxybuprocaine is combined with Propoxycaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Cocaine is combined with Propoxycaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Mepivacaine is combined with Propoxycaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Levobupivacaine is combined with Propoxycaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Diphenhydramine is combined with Propoxycaine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Benzocaine is combined with Propoxycaine.
Phenol The risk or severity of methemoglobinemia can be increased when Phenol is combined with Propoxycaine.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Tetrodotoxin is combined with Propoxycaine.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Benzyl alcohol is combined with Propoxycaine.
Capsaicin The risk or severity of methemoglobinemia can be increased when Capsaicin is combined with Propoxycaine.
Etidocaine The risk or severity of methemoglobinemia can be increased when Etidocaine is combined with Propoxycaine.
Articaine The risk or severity of methemoglobinemia can be increased when Articaine is combined with Propoxycaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Tetracaine is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Propoxycaine is combined with Quinisocaine.
Cetuximab The risk or severity of methemoglobinemia can be increased when Cetuximab is combined with Propoxycaine.
Denileukin diftitox The risk or severity of methemoglobinemia can be increased when Denileukin diftitox is combined with Propoxycaine.
Leuprolide The risk or severity of methemoglobinemia can be increased when Leuprolide is combined with Propoxycaine.
Peginterferon alfa-2a The risk or severity of methemoglobinemia can be increased when Peginterferon alfa-2a is combined with Propoxycaine.
Goserelin The risk or severity of methemoglobinemia can be increased when Goserelin is combined with Propoxycaine.
Asparaginase Escherichia coli The risk or severity of methemoglobinemia can be increased when Asparaginase Escherichia coli is combined with Propoxycaine.
Interferon alfa-2a The risk or severity of methemoglobinemia can be increased when Interferon alfa-2a is combined with Propoxycaine.
Aldesleukin The risk or severity of methemoglobinemia can be increased when Aldesleukin is combined with Propoxycaine.
Gemtuzumab ozogamicin The risk or severity of methemoglobinemia can be increased when Gemtuzumab ozogamicin is combined with Propoxycaine.
Pegaspargase The risk or severity of methemoglobinemia can be increased when Pegaspargase is combined with Propoxycaine.
Trastuzumab The risk or severity of methemoglobinemia can be increased when Trastuzumab is combined with Propoxycaine.
Rituximab The risk or severity of methemoglobinemia can be increased when Rituximab is combined with Propoxycaine.
Tositumomab The risk or severity of methemoglobinemia can be increased when Tositumomab is combined with Propoxycaine.
Alemtuzumab The risk or severity of methemoglobinemia can be increased when Alemtuzumab is combined with Propoxycaine.
Octreotide The risk or severity of methemoglobinemia can be increased when Octreotide is combined with Propoxycaine.
Interferon alfa-2b The risk or severity of methemoglobinemia can be increased when Interferon alfa-2b is combined with Propoxycaine.
Bevacizumab The risk or severity of methemoglobinemia can be increased when Bevacizumab is combined with Propoxycaine.
Masoprocol The risk or severity of methemoglobinemia can be increased when Masoprocol is combined with Propoxycaine.
Bortezomib The risk or severity of methemoglobinemia can be increased when Bortezomib is combined with Propoxycaine.
Pipobroman The risk or severity of methemoglobinemia can be increased when Pipobroman is combined with Propoxycaine.
Cladribine The risk or severity of methemoglobinemia can be increased when Cladribine is combined with Propoxycaine.
Cabergoline The risk or severity of methemoglobinemia can be increased when Cabergoline is combined with Propoxycaine.
Anagrelide The risk or severity of methemoglobinemia can be increased when Anagrelide is combined with Propoxycaine.
Carmustine The risk or severity of methemoglobinemia can be increased when Carmustine is combined with Propoxycaine.
Chlorotrianisene The risk or severity of methemoglobinemia can be increased when Chlorotrianisene is combined with Propoxycaine.
Amsacrine The risk or severity of methemoglobinemia can be increased when Amsacrine is combined with Propoxycaine.
Pamidronic acid The risk or severity of methemoglobinemia can be increased when Pamidronic acid is combined with Propoxycaine.
Bleomycin The risk or severity of methemoglobinemia can be increased when Bleomycin is combined with Propoxycaine.
Chlorambucil The risk or severity of methemoglobinemia can be increased when Chlorambucil is combined with Propoxycaine.
Raltitrexed The risk or severity of methemoglobinemia can be increased when Raltitrexed is combined with Propoxycaine.
Mitomycin The risk or severity of methemoglobinemia can be increased when Mitomycin is combined with Propoxycaine.
Bexarotene The risk or severity of methemoglobinemia can be increased when Bexarotene is combined with Propoxycaine.
Vindesine The risk or severity of methemoglobinemia can be increased when Vindesine is combined with Propoxycaine.
Valproic acid The risk or severity of methemoglobinemia can be increased when Valproic acid is combined with Propoxycaine.
Gefitinib The risk or severity of methemoglobinemia can be increased when Gefitinib is combined with Propoxycaine.
Floxuridine The risk or severity of methemoglobinemia can be increased when Floxuridine is combined with Propoxycaine.
Megestrol acetate The risk or severity of methemoglobinemia can be increased when Megestrol acetate is combined with Propoxycaine.
Tioguanine The risk or severity of methemoglobinemia can be increased when Tioguanine is combined with Propoxycaine.
Aminoglutethimide The risk or severity of methemoglobinemia can be increased when Aminoglutethimide is combined with Propoxycaine.
Vinorelbine The risk or severity of methemoglobinemia can be increased when Vinorelbine is combined with Propoxycaine.
Valrubicin The risk or severity of methemoglobinemia can be increased when Valrubicin is combined with Propoxycaine.
Sorafenib The risk or severity of methemoglobinemia can be increased when Sorafenib is combined with Propoxycaine.
Streptozocin The risk or severity of methemoglobinemia can be increased when Streptozocin is combined with Propoxycaine.
Trifluridine The risk or severity of methemoglobinemia can be increased when Trifluridine is combined with Propoxycaine.
Gemcitabine The risk or severity of methemoglobinemia can be increased when Gemcitabine is combined with Propoxycaine.
Teniposide The risk or severity of methemoglobinemia can be increased when Teniposide is combined with Propoxycaine.
Epirubicin The risk or severity of methemoglobinemia can be increased when Epirubicin is combined with Propoxycaine.
Lenalidomide The risk or severity of methemoglobinemia can be increased when Lenalidomide is combined with Propoxycaine.
Altretamine The risk or severity of methemoglobinemia can be increased when Altretamine is combined with Propoxycaine.
Flutamide The risk or severity of methemoglobinemia can be increased when Flutamide is combined with Propoxycaine.
Cisplatin The risk or severity of methemoglobinemia can be increased when Cisplatin is combined with Propoxycaine.
Alitretinoin The risk or severity of methemoglobinemia can be increased when Alitretinoin is combined with Propoxycaine.
Oxaliplatin The risk or severity of methemoglobinemia can be increased when Oxaliplatin is combined with Propoxycaine.
Erlotinib The risk or severity of methemoglobinemia can be increased when Erlotinib is combined with Propoxycaine.
Cyclophosphamide The risk or severity of methemoglobinemia can be increased when Cyclophosphamide is combined with Propoxycaine.
Toremifene The risk or severity of methemoglobinemia can be increased when Toremifene is combined with Propoxycaine.
Vincristine The risk or severity of methemoglobinemia can be increased when Vincristine is combined with Propoxycaine.
Fluorouracil The risk or severity of methemoglobinemia can be increased when Fluorouracil is combined with Propoxycaine.
Pentostatin The risk or severity of methemoglobinemia can be increased when Pentostatin is combined with Propoxycaine.
Methotrexate The risk or severity of methemoglobinemia can be increased when Methotrexate is combined with Propoxycaine.
Vinblastine The risk or severity of methemoglobinemia can be increased when Vinblastine is combined with Propoxycaine.
Medroxyprogesterone acetate The risk or severity of methemoglobinemia can be increased when Medroxyprogesterone acetate is combined with Propoxycaine.
Imatinib The risk or severity of methemoglobinemia can be increased when Imatinib is combined with Propoxycaine.
Clofarabine The risk or severity of methemoglobinemia can be increased when Clofarabine is combined with Propoxycaine.
Prednisone The risk or severity of methemoglobinemia can be increased when Prednisone is combined with Propoxycaine.

Target Protein

Voltage-gated sodium channel alpha subunit SCN1A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 19897799
    Hung CH, Liu KS, Shao DZ, Cheng KI, Chen YC, Chen YW: The systemic toxicity of equipotent proxymetacaine, oxybuprocaine, and bupivacaine during continuous intravenous infusion in rats. Anesth Analg. 2010 Jan 1;110(1):238-42. doi: 10.1213/ANE.0b013e3181bf6acf. Epub 2009 Nov 6.
  • PMID: 18407836
    Lee JH, Kim DI, Mun H, Lee SK, Park JS, Kim JH, Lee JH, Park YH, Jeon YC, Yoon UC, Bae MK, Jang HO, Wood WG, Yun I: The effect of propoxycaine.HCl on the physical properties of neuronal membranes. Chem Phys Lipids. 2008 Jul;154(1):19-25. doi: 10.1016/j.chemphyslip.2008.03.009. Epub 2008 Mar 22.

Contoh Produk & Brand

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