Solithromycin

DB09308

small molecule investigational

Deskripsi

Solithromycin is a ketolide antibiotic undergoing clinical development for the treatment of community-acquired pneumonia (CAP) and other infections.

Struktur Molekul 2D

Berat 845.0088
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

315 Data
Eliglustat The metabolism of Eliglustat can be decreased when combined with Solithromycin.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Solithromycin.
Alfentanil The serum concentration of Alfentanil can be increased when it is combined with Solithromycin.
Buspirone The metabolism of Buspirone can be decreased when combined with Solithromycin.
Carbamazepine The metabolism of Carbamazepine can be decreased when combined with Solithromycin.
Cisapride The serum concentration of Cisapride can be increased when it is combined with Solithromycin.
Disopyramide Solithromycin may increase the QTc-prolonging activities of Disopyramide.
Estazolam The serum concentration of Estazolam can be increased when it is combined with Solithromycin.
Quinine The serum concentration of Quinine can be increased when it is combined with Solithromycin.
Quinidine The serum concentration of Quinidine can be increased when it is combined with Solithromycin.
Repaglinide The serum concentration of Repaglinide can be increased when it is combined with Solithromycin.
Sirolimus The metabolism of Sirolimus can be decreased when combined with Solithromycin.
Temsirolimus The metabolism of Temsirolimus can be decreased when combined with Solithromycin.
Terfenadine The serum concentration of Terfenadine can be increased when it is combined with Solithromycin.
Triazolam The serum concentration of Triazolam can be increased when it is combined with Solithromycin.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Solithromycin.
Colchicine The metabolism of Colchicine can be decreased when combined with Solithromycin.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Solithromycin.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Solithromycin.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Solithromycin.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Solithromycin.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with Solithromycin.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Solithromycin.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Solithromycin.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Solithromycin.
Alprazolam The serum concentration of Alprazolam can be increased when it is combined with Solithromycin.
Warfarin The serum concentration of Warfarin can be increased when it is combined with Solithromycin.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with Solithromycin.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with Solithromycin.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with Solithromycin.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with Solithromycin.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with Solithromycin.
Midazolam The serum concentration of Midazolam can be increased when it is combined with Solithromycin.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with Solithromycin.
Telaprevir The serum concentration of Telaprevir can be increased when it is combined with Solithromycin.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Solithromycin.
Vintafolide The serum concentration of Vintafolide can be increased when it is combined with Solithromycin.
Vincamine The serum concentration of Vincamine can be increased when it is combined with Solithromycin.
Acetyldigitoxin The serum concentration of Acetyldigitoxin can be increased when it is combined with Solithromycin.
Deslanoside The serum concentration of Deslanoside can be increased when it is combined with Solithromycin.
Ouabain The serum concentration of Ouabain can be increased when it is combined with Solithromycin.
Oleandrin The serum concentration of Oleandrin can be increased when it is combined with Solithromycin.
Cymarin The serum concentration of Cymarin can be increased when it is combined with Solithromycin.
Proscillaridin The serum concentration of Proscillaridin can be increased when it is combined with Solithromycin.
Metildigoxin The serum concentration of Metildigoxin can be increased when it is combined with Solithromycin.
Lanatoside C The serum concentration of Lanatoside C can be increased when it is combined with Solithromycin.
Gitoformate The serum concentration of Gitoformate can be increased when it is combined with Solithromycin.
Acetyldigoxin The serum concentration of Acetyldigoxin can be increased when it is combined with Solithromycin.
Peruvoside The serum concentration of Peruvoside can be increased when it is combined with Solithromycin.
Cyclosporine The metabolism of Cyclosporine can be decreased when combined with Solithromycin.
Dicoumarol The serum concentration of Dicoumarol can be increased when it is combined with Solithromycin.
Phenindione The serum concentration of Phenindione can be increased when it is combined with Solithromycin.
Coumarin The serum concentration of Coumarin can be increased when it is combined with Solithromycin.
Tioclomarol The serum concentration of Tioclomarol can be increased when it is combined with Solithromycin.
Ethyl biscoumacetate The serum concentration of Ethyl biscoumacetate can be increased when it is combined with Solithromycin.
Diphenadione The serum concentration of Diphenadione can be increased when it is combined with Solithromycin.
4-hydroxycoumarin The serum concentration of 4-hydroxycoumarin can be increased when it is combined with Solithromycin.
Fluindione The serum concentration of Fluindione can be increased when it is combined with Solithromycin.
Clorindione The serum concentration of Clorindione can be increased when it is combined with Solithromycin.
Oxtriphylline The metabolism of Oxtriphylline can be decreased when combined with Solithromycin.
Doxofylline The metabolism of Doxofylline can be decreased when combined with Solithromycin.
Bamifylline The metabolism of Bamifylline can be decreased when combined with Solithromycin.
Acefylline The metabolism of Acefylline can be decreased when combined with Solithromycin.
Bufylline The metabolism of Bufylline can be decreased when combined with Solithromycin.
Fenethylline The metabolism of Fenethylline can be decreased when combined with Solithromycin.
Proxyphylline The metabolism of Proxyphylline can be decreased when combined with Solithromycin.
Bromotheophylline The metabolism of Bromotheophylline can be decreased when combined with Solithromycin.
Pentoxifylline The metabolism of Pentoxifylline can be decreased when combined with Solithromycin.
8-azaguanine The metabolism of 8-azaguanine can be decreased when combined with Solithromycin.
7,9-Dimethylguanine The metabolism of 7,9-Dimethylguanine can be decreased when combined with Solithromycin.
Xanthine The metabolism of Xanthine can be decreased when combined with Solithromycin.
7-Deazaguanine The metabolism of 7-Deazaguanine can be decreased when combined with Solithromycin.
Guanine The metabolism of Guanine can be decreased when combined with Solithromycin.
9-Methylguanine The metabolism of 9-Methylguanine can be decreased when combined with Solithromycin.
Peldesine The metabolism of Peldesine can be decreased when combined with Solithromycin.
Hypoxanthine The metabolism of Hypoxanthine can be decreased when combined with Solithromycin.
9-Deazaguanine The metabolism of 9-Deazaguanine can be decreased when combined with Solithromycin.
Valomaciclovir The metabolism of Valomaciclovir can be decreased when combined with Solithromycin.
3-isobutyl-1-methyl-7H-xanthine The metabolism of 3-isobutyl-1-methyl-7H-xanthine can be decreased when combined with Solithromycin.
Uric acid The metabolism of Uric acid can be decreased when combined with Solithromycin.
6-O-benzylguanine The metabolism of 6-O-benzylguanine can be decreased when combined with Solithromycin.
Lisofylline The metabolism of Lisofylline can be decreased when combined with Solithromycin.
Lobucavir The metabolism of Lobucavir can be decreased when combined with Solithromycin.
Cafedrine The metabolism of Cafedrine can be decreased when combined with Solithromycin.
Theodrenaline The metabolism of Theodrenaline can be decreased when combined with Solithromycin.
Etamiphylline The metabolism of Etamiphylline can be decreased when combined with Solithromycin.
Pentifylline The metabolism of Pentifylline can be decreased when combined with Solithromycin.
Furafylline The metabolism of Furafylline can be decreased when combined with Solithromycin.
Theobromine The metabolism of Theobromine can be decreased when combined with Solithromycin.
Propentofylline The metabolism of Propentofylline can be decreased when combined with Solithromycin.
Caffeine The metabolism of Caffeine can be decreased when combined with Solithromycin.
8-chlorotheophylline The metabolism of 8-chlorotheophylline can be decreased when combined with Solithromycin.
Mercaptopurine The metabolism of Mercaptopurine can be decreased when combined with Solithromycin.
PCS-499 The metabolism of PCS-499 can be decreased when combined with Solithromycin.
Methylergometrine The serum concentration of Methylergometrine can be increased when it is combined with Solithromycin.
Lisuride The serum concentration of Lisuride can be increased when it is combined with Solithromycin.
Nicergoline The serum concentration of Nicergoline can be increased when it is combined with Solithromycin.
Ergoloid mesylate The serum concentration of Ergoloid mesylate can be increased when it is combined with Solithromycin.
Pergolide The serum concentration of Pergolide can be increased when it is combined with Solithromycin.
Ergometrine The serum concentration of Ergometrine can be increased when it is combined with Solithromycin.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15117934
    Reinert RR: Clinical efficacy of ketolides in the treatment of respiratory tract infections. J Antimicrob Chemother. 2004 Jun;53(6):918-27. Epub 2004 Apr 29.
  • PMID: 2017690
    Menache D: Replacement therapy in patients with hereditary antithrombin III deficiency. Semin Hematol. 1991 Jan;28(1):31-8.
  • PMID: 20211548
    Farrell DJ, Sader HS, Castanheira M, Biedenbach DJ, Rhomberg PR, Jones RN: Antimicrobial characterisation of CEM-101 activity against respiratory tract pathogens, including multidrug-resistant pneumococcal serogroup 19A isolates. Int J Antimicrob Agents. 2010 Jun;35(6):537-43. doi: 10.1016/j.ijantimicag.2010.01.026. Epub 2010 Mar 7.
  • PMID: 19884376
    McGhee P, Clark C, Kosowska-Shick KM, Nagai K, Dewasse B, Beachel L, Appelbaum PC: In vitro activity of CEM-101 against Streptococcus pneumoniae and Streptococcus pyogenes with defined macrolide resistance mechanisms. Antimicrob Agents Chemother. 2010 Jan;54(1):230-8. doi: 10.1128/AAC.01123-09. Epub 2009 Nov 2.
  • PMID: 20022192
    Putnam SD, Castanheira M, Moet GJ, Farrell DJ, Jones RN: CEM-101, a novel fluoroketolide: antimicrobial activity against a diverse collection of Gram-positive and Gram-negative bacteria. Diagn Microbiol Infect Dis. 2010 Apr;66(4):393-401. doi: 10.1016/j.diagmicrobio.2009.10.013.
  • PMID: 21075602
    Putnam SD, Sader HS, Farrell DJ, Biedenbach DJ, Castanheira M: Antimicrobial characterisation of solithromycin (CEM-101), a novel fluoroketolide: activity against staphylococci and enterococci. Int J Antimicrob Agents. 2011 Jan;37(1):39-45. doi: 10.1016/j.ijantimicag.2010.08.021.
  • PMID: 20855725
    Llano-Sotelo B, Dunkle J, Klepacki D, Zhang W, Fernandes P, Cate JH, Mankin AS: Binding and action of CEM-101, a new fluoroketolide antibiotic that inhibits protein synthesis. Antimicrob Agents Chemother. 2010 Dec;54(12):4961-70. doi: 10.1128/AAC.00860-10. Epub 2010 Sep 20.

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