Brilaroxazine

DB09226

small molecule investigational

Deskripsi

Brilaroxazine (RP5063) is an investigational atypical antipsychotic which is under development by Reviva Pharmaceuticals for the treatment of schizophrenia and schizoaffective disorder. Reviva Pharmaceuticals also intends to investigate RP5063 for the treatment of bipolar disorder, major depressive disorder, psychosis/agitation associated with Alzheimer's disease, Parkinson's disease psychosis, attention deficit hyperactivity disorder (ADD/ADHD), and autism. As of May 2015, it is in phase III clinical trials for schizophrenia.

Struktur Molekul 2D

Berat 450.36
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

770 Data
Buprenorphine Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Hydrocodone Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Magnesium sulfate The therapeutic efficacy of Brilaroxazine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Brilaroxazine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Mirtazapine Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Orphenadrine Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Pramipexole Brilaroxazine may increase the sedative activities of Pramipexole.
Ropinirole Brilaroxazine may increase the sedative activities of Ropinirole.
Rotigotine Brilaroxazine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Brilaroxazine.
Sodium oxybate Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Thalidomide Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Brilaroxazine may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Brilaroxazine.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Brilaroxazine.
Sulpiride Brilaroxazine may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Brilaroxazine.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Brilaroxazine.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Brilaroxazine.
Mequitazine Brilaroxazine may increase the arrhythmogenic activities of Mequitazine.
Tetrabenazine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Tetrabenazine.
Deutetrabenazine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Deutetrabenazine.
Dicoumarol The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with (S)-Warfarin.
Ethanol Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Brilaroxazine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Brilaroxazine.
Zimelidine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Brilaroxazine.
Indalpine The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Brilaroxazine is combined with Alaproclate.
Carbidopa The therapeutic efficacy of Carbidopa can be decreased when used in combination with Brilaroxazine.
Benzatropine The therapeutic efficacy of Benzatropine can be decreased when used in combination with Brilaroxazine.
Cabergoline The therapeutic efficacy of Cabergoline can be decreased when used in combination with Brilaroxazine.
Tolcapone The therapeutic efficacy of Tolcapone can be decreased when used in combination with Brilaroxazine.
Metixene The therapeutic efficacy of Metixene can be decreased when used in combination with Brilaroxazine.
Trihexyphenidyl The therapeutic efficacy of Trihexyphenidyl can be decreased when used in combination with Brilaroxazine.
Procyclidine The therapeutic efficacy of Procyclidine can be decreased when used in combination with Brilaroxazine.
Profenamine The therapeutic efficacy of Profenamine can be decreased when used in combination with Brilaroxazine.
Entacapone The therapeutic efficacy of Entacapone can be decreased when used in combination with Brilaroxazine.
Lisuride The therapeutic efficacy of Lisuride can be decreased when used in combination with Brilaroxazine.
Apomorphine The therapeutic efficacy of Apomorphine can be decreased when used in combination with Brilaroxazine.
Biperiden The therapeutic efficacy of Biperiden can be decreased when used in combination with Brilaroxazine.
Amantadine The therapeutic efficacy of Amantadine can be decreased when used in combination with Brilaroxazine.
Memantine The therapeutic efficacy of Memantine can be decreased when used in combination with Brilaroxazine.
Pergolide The therapeutic efficacy of Pergolide can be decreased when used in combination with Brilaroxazine.
Bromocriptine The therapeutic efficacy of Bromocriptine can be decreased when used in combination with Brilaroxazine.
Levodopa The therapeutic efficacy of Levodopa can be decreased when used in combination with Brilaroxazine.
Rasagiline The therapeutic efficacy of Rasagiline can be decreased when used in combination with Brilaroxazine.
3,5-Dinitrocatechol The therapeutic efficacy of 3,5-Dinitrocatechol can be decreased when used in combination with Brilaroxazine.
Etilevodopa The therapeutic efficacy of Etilevodopa can be decreased when used in combination with Brilaroxazine.
Safinamide The therapeutic efficacy of Safinamide can be decreased when used in combination with Brilaroxazine.
Ifenprodil The therapeutic efficacy of Ifenprodil can be decreased when used in combination with Brilaroxazine.
Dexetimide The therapeutic efficacy of Dexetimide can be decreased when used in combination with Brilaroxazine.
Opicapone The therapeutic efficacy of Opicapone can be decreased when used in combination with Brilaroxazine.
Piribedil The therapeutic efficacy of Piribedil can be decreased when used in combination with Brilaroxazine.
Benserazide The therapeutic efficacy of Benserazide can be decreased when used in combination with Brilaroxazine.
Tropatepine The therapeutic efficacy of Tropatepine can be decreased when used in combination with Brilaroxazine.
Melevodopa The therapeutic efficacy of Melevodopa can be decreased when used in combination with Brilaroxazine.
Dihydroergocryptine The therapeutic efficacy of Dihydroergocryptine can be decreased when used in combination with Brilaroxazine.

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