AS-8112

DB09207

small molecule experimental

Deskripsi

AS-8112 is a synthetic compound that acts as a selective antagonist at the dopamine receptor subtypes D2 and D3, and the serotonin receptor 5-HT3. It has been shown to exert potent antiemetic effects in animal studies and has been investigated for potential medical use.

Struktur Molekul 2D

Berat 399.333
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

25 Data
Tetrabenazine The risk or severity of adverse effects can be increased when AS-8112 is combined with Tetrabenazine.
Deutetrabenazine The risk or severity of adverse effects can be increased when AS-8112 is combined with Deutetrabenazine.
Apomorphine The therapeutic efficacy of Apomorphine can be decreased when used in combination with AS-8112.
Bromocriptine The therapeutic efficacy of Bromocriptine can be decreased when used in combination with AS-8112.
Levodopa The therapeutic efficacy of Levodopa can be decreased when used in combination with AS-8112.
Rotigotine The therapeutic efficacy of Rotigotine can be decreased when used in combination with AS-8112.
Piribedil The therapeutic efficacy of Piribedil can be decreased when used in combination with AS-8112.
Cabergoline The therapeutic efficacy of Cabergoline can be decreased when used in combination with AS-8112.
Dihydroergotamine The therapeutic efficacy of Dihydroergotamine can be decreased when used in combination with AS-8112.
Lisuride The therapeutic efficacy of Lisuride can be decreased when used in combination with AS-8112.
Fenoldopam The therapeutic efficacy of Fenoldopam can be decreased when used in combination with AS-8112.
Ergoloid mesylate The therapeutic efficacy of Ergoloid mesylate can be decreased when used in combination with AS-8112.
Pergolide The therapeutic efficacy of Pergolide can be decreased when used in combination with AS-8112.
Aripiprazole The therapeutic efficacy of Aripiprazole can be decreased when used in combination with AS-8112.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with AS-8112.
Brexpiprazole The therapeutic efficacy of Brexpiprazole can be decreased when used in combination with AS-8112.
Dihydroergocornine The therapeutic efficacy of Dihydroergocornine can be decreased when used in combination with AS-8112.
Dopexamine The therapeutic efficacy of Dopexamine can be decreased when used in combination with AS-8112.
Dihydrexidine The therapeutic efficacy of Dihydrexidine can be decreased when used in combination with AS-8112.
Dihydroergocryptine The therapeutic efficacy of Dihydroergocryptine can be decreased when used in combination with AS-8112.
Metergoline The therapeutic efficacy of Metergoline can be decreased when used in combination with AS-8112.
Ropinirole The therapeutic efficacy of Ropinirole can be decreased when used in combination with AS-8112.
Benzatropine The risk or severity of adverse effects can be increased when AS-8112 is combined with Benzatropine.
Pramipexole The therapeutic efficacy of Pramipexole can be decreased when used in combination with AS-8112.
Epicriptine The therapeutic efficacy of Epicriptine can be decreased when used in combination with AS-8112.

Target Protein

D(2) dopamine receptor DRD2
D(3) dopamine receptor DRD3
5HT3 serotonin receptor

Referensi & Sumber

Artikel (PubMed)
  • PMID: 11350861
    Yoshikawa T, Yoshida N, Oka M: The broad-spectrum anti-emetic activity of AS-8112, a novel dopamine D2, D3 and 5-HT3 receptors antagonist. Br J Pharmacol. 2001 May;133(2):253-60.
  • PMID: 11730730
    Yoshikawa T, Yoshida N, Oka M: Central antiemetic effects of AS-8112, a dopamine D2, D3, and 5-HT(3) receptor antagonist, in ferrets. Eur J Pharmacol. 2001 Nov 23;431(3):361-4.
  • PMID: 12593651
    Hirokawa Y, Fujiwara I, Suzuki K, Harada H, Yoshikawa T, Yoshida N, Kato S: Synthesis and structure-affinity relationships of novel N-(1-ethyl-4-methylhexahydro-1,4-diazepin-6-yl)pyridine-3-carboxamides with potent serotonin 5-HT3 and dopamine D2 receptor antagonistic activity. J Med Chem. 2003 Feb 27;46(5):702-15.

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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