Peringatan Keamanan

LD50 information for peginterferon beta-1a is not readily available in the literature. In clinical trials, no cases of overdoses occurred with the administration of interferon beta-1a at a dose of 75 ?g administered subcutaneously 3 times a week.L31428 In a case report, a 38-year-old patient attempted suicide with about 6 or 7 pre-filled syringes containing 44 mug (12 MIU) of subcutaneous interferon beta-1a; symptoms were limited to malaise and skin erythema, which resolved within 24 hours with no intervention. Laboratory test results were unremarkable.A191871 In the case of an overdose with interferon-beta 1a, prescribing information suggests to contact the local poison control centre.L31438

Peginterferon beta-1a

DB09122

biotech approved

Deskripsi

Multiple Sclerosis (MS) is a chronic and inflammatory autoimmune disease of the central nervous system, disrupting communication between the brain and other parts of the body. Most patients diagnosed with this illness experience their initial disease symptoms between the age of 20 to 40, often the most productive years of life. Symptoms may include but are not limited to fatigue, gait changes, bowel or bladder dysfunction, abnormal muscle twitching, vision disturbance, and depressing or mood swings.L5801 MS is one of the most common causes of neurological disability in young adults and is found to occur more frequently in women than in men.A176474,L5792

Peginterferon beta-1a is an interferon therapy used for the management of relapsing forms of MS. It was originally approved by the FDA in 2014 for subcutaneous use, and was approved for intramuscular use in January 2021.L31428 Currently, it is the only approved pegylated interferon for the management of MS with an proven ability to reduce relapses and delay the progression of disability resulting from MS.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The mean half life of peginterferon beta-1a is approximately 78 h in patients with MS[L31438], however, the half-life is highly variable and depends on duration of treatment and other factors.[A227983]
Volume Distribusi The volume of distribution of peginterferon beta-1a is about 481 L.[L31428] One pharmacokinetic study of patients administered interferon beta-1a revealed a volume of distribution in the range of 248-726 L, depending on the week of treatment.[A227983]
Klirens (Clearance) The average steady state clearance of peginterferon beta-1a is about 4.1 L/h.[L31428] One pharmacokinetic study revealed a clearance within the range of 3.68-7.89 L/h, depending on the week of treatment.[A227983]

Absorpsi

Peginterferon beta-1a is almost completely absorbed after subcutaneous administration. After 125 microgram subcutaneous doses of peginterferon beta-1a to patient with MS, a Cmax of 280 pg/mL was reached between 1 and 1.5 daysA227983, and the AUC over a 14 day dosing interval was 34.8 ng.hr/mL.L31428 The AUC ranges from 23.5-29.5 ng ml?1h, according to one pharmacokinetic study of patients with MS. Impairment of renal function may alter the Cmax and AUC of interferon beta-1a.A227983

Metabolisme

Peginterferon beta-1a is not extensively metabolized in the liver.L31428

Rute Eliminasi

Peginterferon beta-1a is mainly cleared through the kidneys.A227983,L31428

Interaksi Obat

555 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Peginterferon beta-1a.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Peginterferon beta-1a.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Peginterferon beta-1a.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Peginterferon beta-1a.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Peginterferon beta-1a.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Peginterferon beta-1a.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Peginterferon beta-1a.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Peginterferon beta-1a.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Peginterferon beta-1a.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Peginterferon beta-1a.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Peginterferon beta-1a.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Peginterferon beta-1a.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Peginterferon beta-1a.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Peginterferon beta-1a.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Peginterferon beta-1a.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Peginterferon beta-1a.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Peginterferon beta-1a.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Peginterferon beta-1a.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Peginterferon beta-1a.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Peginterferon beta-1a.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Peginterferon beta-1a.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Peginterferon beta-1a.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Peginterferon beta-1a.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Peginterferon beta-1a.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Peginterferon beta-1a.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Peginterferon beta-1a.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Peginterferon beta-1a.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Peginterferon beta-1a.
Flunisolide The risk or severity of adverse effects can be increased when Flunisolide is combined with Peginterferon beta-1a.
Bortezomib The risk or severity of adverse effects can be increased when Bortezomib is combined with Peginterferon beta-1a.
Cladribine Peginterferon beta-1a may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Peginterferon beta-1a.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Peginterferon beta-1a.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Peginterferon beta-1a.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Peginterferon beta-1a.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Peginterferon beta-1a.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Peginterferon beta-1a.
Bexarotene The risk or severity of adverse effects can be increased when Bexarotene is combined with Peginterferon beta-1a.
Vindesine The risk or severity of adverse effects can be increased when Vindesine is combined with Peginterferon beta-1a.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Peginterferon beta-1a.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Peginterferon beta-1a.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Peginterferon beta-1a.
Vinorelbine The risk or severity of adverse effects can be increased when Vinorelbine is combined with Peginterferon beta-1a.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Peginterferon beta-1a.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Beclomethasone dipropionate is combined with Peginterferon beta-1a.
Sorafenib The risk or severity of adverse effects can be increased when Sorafenib is combined with Peginterferon beta-1a.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Peginterferon beta-1a.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Peginterferon beta-1a.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Peginterferon beta-1a.
Betamethasone The risk or severity of adverse effects can be increased when Betamethasone is combined with Peginterferon beta-1a.
Teniposide The risk or severity of adverse effects can be increased when Teniposide is combined with Peginterferon beta-1a.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Peginterferon beta-1a.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Peginterferon beta-1a.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Peginterferon beta-1a.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Peginterferon beta-1a.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Peginterferon beta-1a.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Peginterferon beta-1a.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Peginterferon beta-1a.
Cyclophosphamide The risk or severity of adverse effects can be increased when Cyclophosphamide is combined with Peginterferon beta-1a.
Vincristine The risk or severity of adverse effects can be increased when Vincristine is combined with Peginterferon beta-1a.
Fluorouracil The risk or severity of adverse effects can be increased when Fluorouracil is combined with Peginterferon beta-1a.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Peginterferon beta-1a.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Peginterferon beta-1a.
Methotrexate The risk or severity of adverse effects can be increased when Methotrexate is combined with Peginterferon beta-1a.
Carbamazepine The risk or severity of adverse effects can be increased when Carbamazepine is combined with Peginterferon beta-1a.
Vinblastine The risk or severity of adverse effects can be increased when Vinblastine is combined with Peginterferon beta-1a.
Fluticasone propionate The risk or severity of adverse effects can be increased when Fluticasone propionate is combined with Peginterferon beta-1a.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Fluocinolone acetonide is combined with Peginterferon beta-1a.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Peginterferon beta-1a.
Imatinib The risk or severity of adverse effects can be increased when Imatinib is combined with Peginterferon beta-1a.
Triamcinolone The risk or severity of adverse effects can be increased when Triamcinolone is combined with Peginterferon beta-1a.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Peginterferon beta-1a.
Prednisone The risk or severity of adverse effects can be increased when Prednisone is combined with Peginterferon beta-1a.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Peginterferon beta-1a.
Fludrocortisone The risk or severity of adverse effects can be increased when Fludrocortisone is combined with Peginterferon beta-1a.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mycophenolate mofetil is combined with Peginterferon beta-1a.
Daunorubicin The risk or severity of adverse effects can be increased when Daunorubicin is combined with Peginterferon beta-1a.
Irinotecan The risk or severity of adverse effects can be increased when Irinotecan is combined with Peginterferon beta-1a.
Methimazole The risk or severity of adverse effects can be increased when Methimazole is combined with Peginterferon beta-1a.
Etoposide The risk or severity of adverse effects can be increased when Etoposide is combined with Peginterferon beta-1a.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Peginterferon beta-1a.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Peginterferon beta-1a.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Peginterferon beta-1a.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Peginterferon beta-1a.
Prednisolone The risk or severity of adverse effects can be increased when Prednisolone is combined with Peginterferon beta-1a.
Sirolimus The risk or severity of adverse effects can be increased when Sirolimus is combined with Peginterferon beta-1a.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Peginterferon beta-1a.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Peginterferon beta-1a.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Peginterferon beta-1a.
Methylprednisolone The risk or severity of adverse effects can be increased when Methylprednisolone is combined with Peginterferon beta-1a.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Peginterferon beta-1a.
Cytarabine The risk or severity of adverse effects can be increased when Cytarabine is combined with Peginterferon beta-1a.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Peginterferon beta-1a.
Doxorubicin The risk or severity of adverse effects can be increased when Doxorubicin is combined with Peginterferon beta-1a.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Peginterferon beta-1a.
Busulfan The risk or severity of adverse effects can be increased when Busulfan is combined with Peginterferon beta-1a.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Peginterferon beta-1a.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Peginterferon beta-1a.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Peginterferon beta-1a.
Thalidomide The risk or severity of adverse effects can be increased when Thalidomide is combined with Peginterferon beta-1a.

Target Protein

Interferon alpha/beta receptor 1 IFNAR1

Referensi & Sumber

Synthesis reference: Alessandra Del RioJoel Richard ; PEG-interferon-beta formulations. United States Patent US9138403B2. 2015-Sep-22
Artikel (PubMed)
  • PMID: 26195056
    Newsome SD, Guo S, Altincatal A, Proskorovsky I, Kinter E, Phillips G, You X, Sabatella G: Impact of peginterferon beta-1a and disease factors on quality of life in multiple sclerosis. Mult Scler Relat Disord. 2015 Jul;4(4):350-7. doi: 10.1016/j.msard.2015.06.004. Epub 2015 Jun 14.
  • PMID: 26036950
    Khan UT, Tanasescu R, Constantinescu CS: PEGylated IFNbeta-1a in the treatment of multiple sclerosis. Expert Opin Biol Ther. 2015 Jul;15(7):1077-84. doi: 10.1517/14712598.2015.1053206. Epub 2015 Jun 3.
  • PMID: 28367411
    Ghasemi N, Razavi S, Nikzad E: Multiple Sclerosis: Pathogenesis, Symptoms, Diagnoses and Cell-Based Therapy. Cell J. 2017 Apr-Jun;19(1):1-10. Epub 2016 Dec 21.
  • PMID: 25265472
    Hu X, Cui Y, White J, Zhu Y, Deykin A, Nestorov I, Hung S: Pharmacokinetics and pharmacodynamics of peginterferon beta-1a in patients with relapsing-remitting multiple sclerosis in the randomized ADVANCE study. Br J Clin Pharmacol. 2015 Mar;79(3):514-22. doi: 10.1111/bcp.12521.
  • PMID: 25666445
    Hoy SM: Peginterferon beta-1a: a review of its use in patients with relapsing-remitting multiple sclerosis. CNS Drugs. 2015 Feb;29(2):171-9. doi: 10.1007/s40263-015-0227-1.
  • PMID: 28638705
    Madsen C: The innovative development in interferon beta treatments of relapsing-remitting multiple sclerosis. Brain Behav. 2017 May 8;7(6):e00696. doi: 10.1002/brb3.696. eCollection 2017 Jun.
  • PMID: 2441659
    Pestka S, Langer JA, Zoon KC, Samuel CE: Interferons and their actions. Annu Rev Biochem. 1987;56:727-77. doi: 10.1146/annurev.bi.56.070187.003455.
  • PMID: 17562848
    Markowitz CE: Interferon-beta: mechanism of action and dosing issues. Neurology. 2007 Jun 12;68(24 Suppl 4):S8-11. doi: 10.1212/01.wnl.0000277703.74115.d2.
Menampilkan 8 dari 10 artikel.

Contoh Produk & Brand

Produk: 18 • International brands: 1
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International Brands
  • Plegridy — Biogen

Sekuens Gen/Protein (FASTA)

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