Peringatan Keamanan

The acute oral LD50 in mice is 2314mg/kg MSDS.The most common adverse effects of tertacylines are gastrointestinal disturbances, and staining of teeth and bone. Some occurences of dental hypoplasia and bone deformity have been noted T28. In pregnant women tetracyclines may produce hepatotoxicity.

Chlortetracycline

DB09093

small molecule approved investigational vet_approved

Deskripsi

Chlortetracycline is a tetracycline antibiotic, and historically the first member of this class to be identified. It was discovered in 1945 by the scientist, Benjamin Minge Duggar, working at Lederle Laboratories under the supervision of Yellapragada Subbarow. He discovered that this antibiotic was the product of an actinomycete strain he cultured and obtained from a soil sample from a field in Missouri. The organism was named Streptomyces aureofaciens due to its gold-hued color.

Struktur Molekul 2D

Berat 478.88
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The half-life of Chlortetracycline is 5.6 hours [A1424].
Volume Distribusi Chlortetracycline has a volume of distribution of 100 liters [A1424].
Klirens (Clearance) -

Absorpsi

Chortetracycline reaches peak plasma concentation in about 3 hours A1424. Its oral bioavailability is 25-30%.

Metabolisme

Chlortetracycline is not known to undergo significant metabolism A1424.

Rute Eliminasi

Chlortetracycline is mainly eliminated in feces A1424. Renal function does not appear to affect the rate of elimination.

Interaksi Obat

43 Data
Methoxyflurane The risk or severity of renal failure can be increased when Methoxyflurane is combined with Chlortetracycline.
Magnesium Magnesium can cause a decrease in the absorption of Chlortetracycline resulting in a reduced serum concentration and potentially a decrease in efficacy.
Vibrio cholerae CVD 103-HgR strain live antigen The therapeutic efficacy of Vibrio cholerae CVD 103-HgR strain live antigen can be decreased when used in combination with Chlortetracycline.
Didanosine Didanosine can cause a decrease in the absorption of Chlortetracycline resulting in a reduced serum concentration and potentially a decrease in efficacy.
Collagenase clostridium histolyticum The therapeutic efficacy of Collagenase clostridium histolyticum can be decreased when used in combination with Chlortetracycline.
Acetylcysteine The therapeutic efficacy of Acetylcysteine can be decreased when used in combination with Chlortetracycline.
Estetrol The therapeutic efficacy of Estetrol can be decreased when used in combination with Chlortetracycline.
Palovarotene The risk or severity of pseudotumor cerebri can be increased when Chlortetracycline is combined with Palovarotene.
Lidocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Quinisocaine.
Cisatracurium Chlortetracycline may increase the neuromuscular blocking activities of Cisatracurium.
Ambroxol The risk or severity of methemoglobinemia can be increased when Chlortetracycline is combined with Ambroxol.
Fecal microbiota The therapeutic efficacy of Fecal microbiota can be decreased when used in combination with Chlortetracycline.

Target Protein

16S ribosomal RNA
30S ribosomal protein S3 rpsC
30S ribosomal protein S8 rpsH
30S ribosomal protein S19 rpsS
30S ribosomal protein S14 rpsN
30S ribosomal protein S7 rpsG
ADP-ribosylation factor 1 ARF1
Catalase katA
Ephrin type-B receptor 1 EPHB1
Pancreatic triacylglycerol lipase PNLIP
Protein-arginine deiminase type-4 PADI4

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16816396
    Agwuh KN, MacGowan A: Pharmacokinetics and pharmacodynamics of the tetracyclines including glycylcyclines. J Antimicrob Chemother. 2006 Aug;58(2):256-65. Epub 2006 Jul 1.
Textbook
  • ISBN: 978-0-7020-3471-8
    49, 50. (2012). In Rang and Dale's Pharmacology (7th ed., pp. 614, 629). Edinburgh: Elsevier/Churchill Livingstone.

Contoh Produk & Brand

Produk: 3 • International brands: 1
Produk
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International Brands
  • Aueromycin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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