Peringatan Keamanan

A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s T146.

Amylocaine

DB09088

small molecule approved withdrawn

Deskripsi

Despite the introduction of using cocaine injections for regional anesthesia in 1884, non-addictive substitutes were sought after immediately L1882. Finally, in 1903 the world's first synthetic and non-addictive local anesthetic, amylocaine, was synthesized and patented under the name Forneaucaine by Ernest Fourneau at the Pasteur Institute L1882. Elsewhere in English speaking countries it was referred to as Stovaine, given the meaning of the French word 'fourneau' as 'stove' in English L1882.

Although amylocaine could be administered topically or injected, it was most widely used for spinal anesthesia L1882. Even though it certainly possessed less severe side effects than cocaine L1882, the eventual development and clinical use of newer, more effective, and even safer local anesthetics like lidocaine, bupivicaine, and prilocaine in the 1940s and 1950s superseded and made the use of amylocaine obsolete.

Struktur Molekul 2D

Berat 235.327
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s [T146].
Volume Distribusi A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s [T146].
Klirens (Clearance) A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s [T146].

Absorpsi

A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s T146.

Metabolisme

A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s T146.

Rute Eliminasi

A lack of detailed information regarding the specificities of amylocaine relate to a lack of information on its pharmacokinetics at the time of its primary use in the early 1900s T146.

Interaksi Obat

0 Data
Tidak ada data.

Target Protein

Voltage-gated sodium channel alpha subunit SCN1A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 20771971
    Coleman RB: SPINAL ANAESTHESIA BY STOVAINE. Br Med J. 1925 Mar 21;1(3351):548-9.
  • PMID: 2157353
    Butterworth JF 4th, Strichartz GR: Molecular mechanisms of local anesthesia: a review. Anesthesiology. 1990 Apr;72(4):711-34.
Textbook
  • ISBN: 978-3-642-71112-1
    Gary R. Strichartz (1987). Local Anesthetics. Springer, Berlin, Heidelberg.

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Dentition Sirop De
    Syrup • 180 mg / 30 mL • Dental • Canada • OTC • Approved
  • Rhino Mex
    Liquid • - • Nasal • Canada • OTC • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul