Peringatan Keamanan

The most common adverse effects with the combination cream are localized reactions such as: erythema (47%), skin discoloration (16%), and edema (14%). Systemic adverse events were less common, occurring at a rate of <1% and included vomiting, headache, dizziness, and fever. Similar to other amide and ester anesthetics, CNS excitation and/or depression may occur. It is not well known at which plasma concentration systemic toxicity occurs with tetracaine; however, the threshold is thought to be much lower than that of lidocaine which is 1000 ng/mL.

Tetracaine

DB09085

small molecule approved vet_approved

Deskripsi

Tetracaine is an ester local anaesthetic currently available in combination with lidocaine as a cream and patch.

Struktur Molekul 2D

Berat 264.369
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Tetracaine is hydrolyzed rapidly in the plasma; therefore, half-life has not been determined.
Volume Distribusi Tetracaine is rapidly hydrolyzed in the plasma; therefore, volume of distribution could not be determined.
Klirens (Clearance) Tetracaine is hydrolyzed rapidly in the plasma; therefore, clearance has not been determined.

Absorpsi

Systemic absorption of anaesthetic from the combination cream is directly related to the duration and surface area of application. Although peak plasma concentrations for lidocaine were measured, plasma levels for tetracaine could not be determined due to low levels (<0.9 ng/mL)

Metabolisme

Tetracaine is rapidly hydrolyzed by plasma esterases to the following primary metabolites: para-aminobenzoic acid and diethylaminoethanol. The activity of both metabolites is unspecified.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1608 Data
Buprenorphine Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Hydrocodone Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Magnesium sulfate The therapeutic efficacy of Tetracaine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Tetracaine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Mirtazapine Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Orphenadrine Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Pramipexole Tetracaine may increase the sedative activities of Pramipexole.
Ropinirole Tetracaine may increase the sedative activities of Ropinirole.
Rotigotine Tetracaine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Tetracaine.
Sodium oxybate Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Thalidomide Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Prilocaine The risk or severity of methemoglobinemia can be increased when Tetracaine is combined with Prilocaine.
Hyaluronidase (ovine) Hyaluronidase (ovine) can cause an increase in the absorption of Tetracaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase (human recombinant) Hyaluronidase (human recombinant) can cause an increase in the absorption of Tetracaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase Hyaluronidase can cause an increase in the absorption of Tetracaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Tetracaine.
Ethanol Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Tetracaine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Fluvoxamine The risk or severity of adverse effects can be increased when Tetracaine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Tetracaine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Tetracaine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Tetracaine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Tetracaine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Tetracaine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Tetracaine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Tetracaine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Tetracaine is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Tetracaine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Tetracaine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Tetracaine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Tetracaine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Tetracaine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Tetracaine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Tetracaine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Tetracaine is combined with Alaproclate.
Dapsone The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Tetracaine.
Technetium Tc-99m tilmanocept Tetracaine may decrease effectiveness of Technetium Tc-99m tilmanocept as a diagnostic agent.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with Tetracaine.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Tetracaine.
Clozapine The risk or severity of CNS depression can be increased when Clozapine is combined with Tetracaine.
Promazine The risk or severity of CNS depression can be increased when Promazine is combined with Tetracaine.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Tetracaine.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with Tetracaine.
Chlorpromazine The risk or severity of CNS depression can be increased when Chlorpromazine is combined with Tetracaine.
Gallamine triethiodide The risk or severity of CNS depression can be increased when Gallamine triethiodide is combined with Tetracaine.
Triflupromazine The risk or severity of CNS depression can be increased when Triflupromazine is combined with Tetracaine.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with Tetracaine.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Tetracaine.
Lamotrigine The risk or severity of methemoglobinemia can be increased when Lamotrigine is combined with Tetracaine.
Rocuronium The risk or severity of CNS depression can be increased when Rocuronium is combined with Tetracaine.
Scopolamine The risk or severity of CNS depression can be increased when Scopolamine is combined with Tetracaine.
Clidinium The risk or severity of CNS depression can be increased when Clidinium is combined with Tetracaine.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Tetracaine.
Brompheniramine The risk or severity of CNS depression can be increased when Brompheniramine is combined with Tetracaine.
Flupentixol The risk or severity of CNS depression can be increased when Flupentixol is combined with Tetracaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Cocaine is combined with Tetracaine.
Quinidine The risk or severity of methemoglobinemia can be increased when Quinidine is combined with Tetracaine.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with Tetracaine.
Promethazine The risk or severity of CNS depression can be increased when Promethazine is combined with Tetracaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Diphenhydramine is combined with Tetracaine.
Doxacurium The risk or severity of CNS depression can be increased when Doxacurium is combined with Tetracaine.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Tetracaine.
Desipramine The risk or severity of CNS depression can be increased when Desipramine is combined with Tetracaine.
Quetiapine The risk or severity of CNS depression can be increased when Quetiapine is combined with Tetracaine.
Mivacurium The risk or severity of CNS depression can be increased when Mivacurium is combined with Tetracaine.
Aripiprazole The risk or severity of CNS depression can be increased when Aripiprazole is combined with Tetracaine.
Chlorprothixene The risk or severity of CNS depression can be increased when Chlorprothixene is combined with Tetracaine.
Metocurine The risk or severity of CNS depression can be increased when Metocurine is combined with Tetracaine.
Pancuronium The risk or severity of CNS depression can be increased when Pancuronium is combined with Tetracaine.
Pipecuronium The risk or severity of CNS depression can be increased when Pipecuronium is combined with Tetracaine.
Rapacuronium The risk or severity of CNS depression can be increased when Rapacuronium is combined with Tetracaine.
Pizotifen The risk or severity of CNS depression can be increased when Pizotifen is combined with Tetracaine.
Benactyzine The risk or severity of CNS depression can be increased when Benactyzine is combined with Tetracaine.
Dosulepin The risk or severity of CNS depression can be increased when Tetracaine is combined with Dosulepin.
Emepronium The risk or severity of CNS depression can be increased when Tetracaine is combined with Emepronium.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Tetracaine.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Tetracaine.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with Tetracaine.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Tetracaine.
Lorazepam The risk or severity of methemoglobinemia can be increased when Lorazepam is combined with Tetracaine.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Tetracaine.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Tetracaine.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with Tetracaine.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Tetracaine.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with Tetracaine.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with Tetracaine.

Target Protein

Ryanodine receptor 1 RYR1
Sodium channel protein type 10 subunit alpha SCN10A
Ryanodine receptor 2 RYR2
Voltage-gated sodium channel alpha subunit SCN1A

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 136 • International brands: 1
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Menampilkan 8 dari 136 produk.
International Brands
  • Pontocaine HCl

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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